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4CEB | 1.75 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | ZSV, GOL, EDO, ACY, SO4 | Kd = 1080 uM | 575.629, 92.094, 62.068, 60.052, 96.063 |
3CKT | 1.65 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | YDP, CL | Ki = 0.48 uM | 603.753, 35.453 |
2ZGA | 1.65 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | YDP | Ki = 0.48 uM | 603.753 |
4CIE | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | Y7N, ACY, CL, SO4 | 422.474, 60.052, 35.453, 96.063 | |
1BV7 | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | XV6 | Ki = 0.5 nM | 758.908 |
1BV9 | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | XV6 | Ki = 1.1 nM | 758.908 |
1BWA | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | XV6 | Ki = 2.5 nM | 758.908 |
1QBR | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | XV6 | Ki = 0.027 nM | 758.908 |
1K6P | 2.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | XN3, ACT | Kd = 44 nM | 656.811, 59.044 |
1K6V | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | XN2, ACT | Kd = 120 nM | 670.837, 59.044 |
1K6T | 2.25 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | XN1, ACT | Kd = 24 nM | 627.816, 59.044 |
1HVR | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | XK2 | Ki = 0.31 nM | 606.752 |
4CIG | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | X0P, ACT, SO4 | Kd = 214 uM | 498.57, 59.044, 96.063 |
4CFA | 2.05 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | WOP, SO4 | 475.493, 96.063 | |
4CJQ | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | VXO, SO4, ACT | Kd = 256 uM | 436.5, 96.063, 59.044 |
4CER | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | VL4, CL, SO4 | 496.552, 35.453, 96.063 | |
1MT7 | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | VAL SER GLN ASN TYR PRO ILE VAL GLN ASN, ACT | 904.056, 59.044 | |
8HVP | 2.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | VAL SER GLN ASN LOV ILE VAL | Ki < 1 nM | 872.075 |
4PHV | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | VAC | ic50 = 0.67 nM | 618.761 |
1HPO | 2.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | UNI | Ki = 0.6 nM | 504.597 |
1S1T | 2.4 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.49 | UC1, PO4 | 335.848, 94.971 | |
4CHO | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | U2Z, EDO, ACT, GOL, SO4 | 217.267, 62.068, 59.044, 92.094, 96.063 | |
1A9M | 2.3 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | U0E | Ki = 119 nM | 596.762 |
1AXA | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | U0E | 596.762 | |
1GNM | 2.3 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | U0E | Ki = 560 nM | 596.762 |