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4PHV | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | VAC | ic50 = 0.67 nM | 618.761 |
4Q1W | 1.85 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | ACT, 017, PO4 | Ki = 2 pM | 59.044, 547.664, 94.971 |
4Q1X | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, 017, GOL | Ki = 7 pM | 94.971, 547.664, 92.094 |
4Q1Y | 1.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | ACT, 017, PO4 | Ki = 45 pM | 59.044, 547.664, 94.971 |
4QJ2 | 2.13 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, SO4, ARG PRO GLY ASN PHE LEU GLN SER ARG PRO, PO4 | 92.094, 96.063, 975.119, 94.971 | |
4RZ8 | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS 1 | NON-ENZYME OTHER | EPE, NAG, 3ZM | ic50 ~ 270 nM | 238.305, 221.208, 444.978 |
4TSX | 1.94 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | SO4, LF0 | Kd = 10.3 uM | 96.063, 405.486 |
4TVG | 2.18 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | K97, IVA VAL VAL STA ALA STA, GOL | 260.288, 696.992, 92.094 | |
4TVH | 2.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 3TL, BME, K97 | 909.077, 78.133, 260.288 | |
4U7Q | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 3EM | Ki = 180 pM | 797.959 |
4U7V | 1.38 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | BME, 3EN | Ki = 3.2 uM | 78.133, 524.675 |
4XRQ | 1.95 | HUMAN IMMUNODEFICIENCY VIRUS 1 | NON-ENZYME OTHER | 1B0 | Kd = 0.232 uM | 425.522 |
5COK | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 52U | 576.701 | |
5CON | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 52W | 592.701 | |
5COO | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 52Z | 622.727 | |
5COP | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 53F | 607.716 | |
5DGU | 1.22 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 5B7, NA, CL, ACT | Ki = 0.0045 nM | 606.727, 22.99, 35.453, 59.044 |
5DGW | 1.62 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 5B5, NA, CL | Ki = 0.009 nM | 619.769, 22.99, 35.453 |
5HGM | 2.04 | HUMAN IMMUNODEFICIENCY VIRUS 1 | NON-ENZYME OTHER | DTP | 491.182 | |
5HRN | 1.75 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.49 | 65P, CAC, SO4, EDO | 534.594, 136.989, 96.063, 62.068 | |
5HRP | 1.81 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | 65P, CAC, EDO, SO4 | 534.594, 136.989, 62.068, 96.063 | |
5HRR | 1.88 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | EDO, 65P, CAC, SO4 | 62.068, 534.594, 136.989, 96.063 | |
5HRS | 1.86 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | EDO, 65P, CAC, SO4 | 62.068, 534.594, 136.989, 96.063 | |
5IVQ | 1.57 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 6EH, CL | 425.521, 35.453 | |
5IVR | 1.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 6EG, CL | 566.69, 35.453 | |
5IVS | 1.46 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 6EF, CL | ic50 = 6.1 nM | 650.763, 35.453 |
5IVT | 1.15 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | ACT, CL, 6EE | ic50 = 0.8 nM | 59.044, 35.453, 674.034 |
5JFP | 1.49 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 6KK, CL, NA | Ki = 0.48 nM | 620.797, 35.453, 22.99 |
5JFU | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 6KQ, CL | Ki = 8.5 nM | 654.813, 35.453 |
5JG1 | 1.16 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, NA, CL, 6KR | Ki = 1.9 nM | 92.094, 22.99, 35.453, 634.824 |
5KAO | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | G43 | 627.146 | |
5KGW | 2.34 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | 7SK, SO4 | 393.475, 96.063 | |
5KQX | 2.4 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | ROC | Ki = 3.6 nM | 670.841 |
5KQY | 1.65 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 017 | Ki = 0.51 nM | 547.664 |
5KQZ | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 0Q4 | 833.053 | |
5KR0 | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 478, GOL | Ki = 0.71 nM | 505.627, 92.094 |
5KR1 | 1.6 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 017 | Ki = 0.32 nM | 547.664 |
5KR2 | 1.78 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | ROC | Ki = 3.3 nM | 670.841 |
5KRS | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | DMS, 6XI | 78.133, 193.222 | |
5KRT | 1.65 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | 6W6 | 262.113 | |
5OI2 | 2.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | SO4, 9VN, MG | ic50 = 0.17 uM | 96.063, 413.573, 24.305 |
5OI5 | 2.4 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | MG, 9VK | ic50 = 0.19 uM | 24.305, 413.573 |
5OI8 | 2.35 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | 9VN, SO4, MG | ic50 = 0.21 uM | 413.573, 96.063, 24.305 |
5OIA | 2.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | 9VK, SO4, MG | ic50 = 0.17 uM | 413.573, 96.063, 24.305 |
5T2Z | 1.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME HYDROLASES | 017 | 547.664 | |
5TKK | 1.55 | HUMAN IMMUNODEFICIENCY VIRUS 1 | NON-ENZYME OTHER | ALA VAL GLY ILE GLY ALA VAL PHE | 471.579 | |
5TYR | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 7O7 | ic50 = 0.26 nM | 670.839 |
5TYS | 2.01 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 7OA | ic50 = 0.019 nM | 706.82 |
5U6E | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | NON-ENZYME OTHER | 82M, EPE, NAG | 408.878, 238.305, 221.208 | |
5ULT | 1.53 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | CL, NA, 8FM | Ki = 0.014 nM | 35.453, 22.99, 588.712 |
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