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1MT8 | 2.15 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | LYS ALA ARG VAL LEU ALA GLU ALA MET SER, ACT | 916.136, 59.044 | |
1ZTZ | 2.15 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | CB5, ALA GLY ALA ALA | Ki = 66 nM | 323.749, 273.313 |
4CFD | 2.15 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | CL, ACT, S8Y, SO4 | 35.453, 59.044, 441.477, 96.063 | |
4CGJ | 2.15 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | NZL, ACT, SO4 | 424.49, 59.044, 96.063 | |
4QJ2 | 2.13 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, SO4, ARG PRO GLY ASN PHE LEU GLN SER ARG PRO, PO4 | 92.094, 96.063, 975.119, 94.971 | |
6OOU | 2.13 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 017, SO4 | 547.664, 96.063 | |
6OPY | 2.13 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME HYDROLASES | 017 | Ki = 156.4 nM | 547.664 |
1EC1 | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | BEE | Ki = 1.2 nM | 778.977 |
1ODW | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 0E8 | Ki = 100 nM | 543.695 |
1OHR | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 1UN | Ki = 2 nM | 567.782 |
1QBT | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 146 | Ki = 0.024 nM | 824.924 |
1QS4 | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | MG, 100 | ic50 = 2.3 uM | 24.305, 289.677 |
1T7K | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | BH0 | Ki = 1.37 nM | 598.669 |
2BQV | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | A1A | Ki = 9 nM | 588.694 |
2P3B | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 3TL | Ki = 3.3 nM | 909.077 |
2P3C | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | ACY, 3TL | Ki = 24 nM | 60.052, 909.077 |
2QI0 | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, MZ3 | Ki = 42 nM | 94.971, 582.706 |
3BGR | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.49 | T27, EDO | 366.419, 62.068 | |
3VQB | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | FBG, SO4, CD | 198.148, 96.063, 112.411 | |
3VQP | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | CL, DBJ, SO4, CD | 35.453, 166.174, 96.063, 112.411 | |
4CE9 | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | O3N, ACY, SO4, GOL | 550.643, 60.052, 96.063, 92.094 | |
4CF9 | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | ACT, EE2, 5EY, SO4, EDO | 59.044, 396.39, 396.39, 96.063, 62.068 | |
4DVS | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | NON-ENZYME OTHER | 0LY, NAG, EPE | 382.295, 221.208, 238.305 | |
4PHV | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | VAC | ic50 = 0.67 nM | 618.761 |
5U6E | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | NON-ENZYME OTHER | 82M, EPE, NAG | 408.878, 238.305, 221.208 | |
6NUJ | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | L3D | 442.506 | |
6OPW | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME HYDROLASES | 017, SO4 | Ki = 23.2 nM | 547.664, 96.063 |
6OPS | 2.08 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 017 | 547.664 | |
4CGI | 2.07 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | NZL, ACT, SO4 | Kd = 752 uM | 424.49, 59.044, 96.063 |
1EBK | 2.06 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 0Q4 | 833.053 | |
1ZSR | 2.06 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 0ZT | Ki = 0.15 nM | 703.824 |
3U7S | 2.05 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | BME, 017 | Ki = 3700 pM | 78.133, 547.664 |
4CFA | 2.05 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | WOP, SO4 | 475.493, 96.063 | |
4GZF | 2.05 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | ILO VAL DC0 GLU ALA NLE | ic50 = 4.4 nM | 832.057 |
4M8X | 2.05 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | KGQ | Ki = 0.063 nM | 728.787 |
5HGM | 2.04 | HUMAN IMMUNODEFICIENCY VIRUS 1 | NON-ENZYME OTHER | DTP | 491.182 | |
6OXR | 2.04 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NJA | 576.701 | |
2AZB | 2.03 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 3TL | ic50 = 64 nM | 909.077 |
6OPX | 2.03 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME HYDROLASES | 017 | Ki = 172.7 nM | 547.664 |
1ZP8 | 2.02 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | AB2 | Ki = 1.7 nM | 663.784 |
1ZPA | 2.02 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | A83 | Ki = 4 nM | 720.878 |
1EBZ | 2.01 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | BEC | Ki = 0.4 nM | 633.731 |
2AZC | 2.01 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 3TL | ic50 = 183 nM | 909.077 |
5TYS | 2.01 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 7OA | ic50 = 0.019 nM | 706.82 |
6DH5 | 2.01 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | A60, SO4 | 575.717, 96.063 | |
1A30 | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GLU ASP LEU | Ki = 50 uM | 373.362 |
1A8K | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 0Q4 | 833.053 | |
1A94 | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 0Q4 | Ki = 14 nM | 833.053 |
1AJV | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NMB | Ki = 19.1 nM | 574.687 |
1AJX | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | AH1 | Ki = 12.2 nM | 538.633 |
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