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6O5A | 1.67 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME HYDROLASES | GOL, 2NC | Ki = 514 nM | 92.094, 770.983 |
2RKG | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, AB1 | Ki = 8.2 nM | 92.094, 628.801 |
6DV4 | 1.14 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, ACT, GA5, CL, NA | Ki = 1.6 nM | 92.094, 59.044, 695.865, 35.453, 22.99 |
2AVM | 1.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, ACY, 2NC | Ki = 2 uM | 92.094, 60.052, 770.983 |
2FLE | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, AI | Ki = 14 nM | 92.094, 801.029 |
1XL2 | 1.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, CL, 189 | Ki = 1.5 uM | 92.094, 35.453, 577.777 |
5UPZ | 1.27 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, CL, 8HD, NA | Ki = 0.63 nM | 92.094, 35.453, 662.796, 22.99 |
2O4S | 1.54 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, CL, AB1 | Kd = 31 pM | 92.094, 35.453, 628.801 |
2O4L | 1.33 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, CL, TPV | Kd = 608 pM | 92.094, 35.453, 602.664 |
2QD7 | 1.11 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, DMS, 065, PO4 | Ki = 0.8 nM | 92.094, 78.133, 576.658, 94.971 |
4E43 | 1.54 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, DMS, BME, ASN LEU LEU GLN LYS LYS, ACT | 92.094, 78.133, 78.133, 729.945, 59.044 | |
4CF8 | 1.65 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | GOL, EDO, CL, ACY, SO4, V7H | 92.094, 62.068, 35.453, 60.052, 96.063, 504.531 | |
4OVL | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | GOL, EDO, SO4, 1TD, ACY | 92.094, 62.068, 96.063, 265.263, 60.052 | |
6OTG | 1.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, FMT, 4UY | Ki = 31.4 nM | 92.094, 46.025, 591.716 |
6DJ7 | 1.31 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, G10, ACT, CL, NA | Ki = 1.9 nM | 92.094, 583.645, 59.044, 35.453, 22.99 |
2PWC | 1.78 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, G3G, CL | Ki = 0.27 uM | 92.094, 591.744, 35.453 |
2R43 | 1.58 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, G3G, CL | Ki = 1 uM | 92.094, 591.744, 35.453 |
2PWR | 1.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, G4G, CL | Ki = 0.26 uM | 92.094, 647.764, 35.453 |
6VCE | 1.18 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, G6R, NA, CL | ic50 = 79 pM | 92.094, 704.847, 22.99, 35.453 |
6DV0 | 1.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, GA8, CL, NA | Ki = 0.38 nM | 92.094, 697.904, 35.453, 22.99 |
6DJ5 | 1.75 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, NA, G52, CL | 92.094, 22.99, 604.712, 35.453 | |
4QJ2 | 2.13 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, SO4, ARG PRO GLY ASN PHE LEU GLN SER ARG PRO, PO4 | 92.094, 96.063, 975.119, 94.971 | |
2O4N | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, TPV | Kd = 15010 pM | 92.094, 602.664 |
4CJK | 1.75 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | H39, CL, SO4, ACT | 386.442, 35.453, 96.063, 59.044 | |
4CHZ | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | H75, EDO, ACT, CL, SO4 | 293.159, 62.068, 59.044, 35.453, 96.063 | |
2BBB | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | HH1 | ic50 = 2.4 nM | 623.738 |
2UXZ | 1.75 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | HI1 | Ki = 3.3 nM | 709.67 |
4CJT | 1.71 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | HLR, GOL, SO4, ACT | 134.135, 92.094, 96.063, 59.044 | |
2UY0 | 1.76 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | HV1 | Ki = 120 nM | 723.653 |
6E7J | 1.3 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | HWY, NA, CL | Ki = 0.33 nM | 651.77, 22.99, 35.453 |
6ES8 | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS 1 | NON-ENZYME OTHER | IHP | 660.035 | |
1KJH | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | ILE ARG LYS ILE LEU PHE LEU ASP GLY ILE, ACT | 1146.42, 59.044 | |
4GZF | 2.05 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | ILO VAL DC0 GLU ALA NLE | ic50 = 4.4 nM | 832.057 |
4GYE | 2.27 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | ILO VAL PUK GLU ALA NLE | 866.074 | |
1BDQ | 2.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | IM1 | Ki = 460 nM | 534.69 |
1TCX | 2.3 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | IM1 | Ki = 112 nM | 534.69 |
7UPJ | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | INU | Ki = 3.2 nM | 479.588 |
4E91 | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS 1 | NON-ENZYME OTHER | IOD, 0OF, 0OE | 126.904, 517.498, 522.985 | |
3NU9 | 1.85 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | IOD, 478 | Ki = 0.9 nM | 126.904, 505.627 |
3NUJ | 1.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | IOD, 478 | Ki = 0.41 nM | 126.904, 505.627 |
3NUO | 1.35 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | IOD, 478 | Ki = 0.16 nM | 126.904, 505.627 |
3S43 | 1.26 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | IOD, GOL, 478 | Ki = 2.53 nM | 126.904, 92.094, 505.627 |
4EJL | 2.45 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | IOP, DMS, GOL, PEG | Kd = 7.2 uM | 189.211, 78.133, 92.094, 106.12 |
4EJK | 1.79 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | IOP, IVA VAL VAL STA ALA STA | Kd = 5.3 uM | 189.211, 696.992 |
4CF1 | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | IY7, ACT, SO4 | 496.552, 59.044, 96.063 | |
6EB1 | 2.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | J3M | ic50 = 4.65 uM | 467.556 |
6EB2 | 2.49 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | J3P | ic50 = 0.48 uM | 547.644 |
6MCS | 1.52 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | JDV | 688.83 | |
6OGQ | 1.41 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME HYDROLASES | JDV, SO4, PEG, GOL | ic50 = 26 nM | 688.83, 96.063, 106.12, 92.094 |
6MCR | 1.48 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | JDY, EDO | 688.83, 62.068 |
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