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2I4W | 1.55 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | KGQ | Ki = 2.6 pM | 728.787 |
2I4X | 1.55 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | KGQ | Ki = 1.9 pM | 728.787 |
4M8X | 2.05 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | KGQ | Ki = 0.063 nM | 728.787 |
4M8Y | 2.22 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | KGQ | Ki = 0.11 nM | 728.787 |
1U8G | 2.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | KI2 PHE GLU GLU NH2 | 732.767 | |
6NCJ | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | KJJ, SO4, EDO | ic50 = 0.024 uM | 572.709, 96.063, 62.068 |
1HPX | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | KNI | Ki = 5.5 pM | 667.839 |
3FX5 | 0.93 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | KNI, GOL | Ki < 1 nM | 667.839, 92.094 |
3A2O | 0.88 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | KNJ, GOL | Ki = 0.83 nM | 568.727, 92.094 |
6KMP | 1.31 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | KVS | 800.986 | |
1NPV | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | L27 | ic50 = 5.7 nM | 595.685 |
6NUJ | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | L3D | 442.506 | |
1C70 | 2.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | L75 | Ki = 0.05 nM | 652.822 |
3OU3 | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | LEU ASN PHE PRO ILE SER PRO | 786.928 | |
1NPW | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | LGZ | ic50 = 2 nM | 625.711 |
1F7A | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | LYS ALA ARG VAL LEU ALA GLU ALA MET SER, ACT | 916.136, 59.044 | |
1MT8 | 2.15 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | LYS ALA ARG VAL LEU ALA GLU ALA MET SER, ACT | 916.136, 59.044 | |
3OU1 | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME HYDROLASES | LYS VAL LEU PHE LEU ASP GLY | 790.96 | |
3ZPU | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | M8B, CL | Ki = 4.2 nM | 742.743, 35.453 |
3ZPT | 1.54 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | M8Y, CL | Ki = 3.1 nM | 728.716, 35.453 |
1QS4 | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | MG, 100 | ic50 = 2.3 uM | 24.305, 289.677 |
5OI5 | 2.4 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | MG, 9VK | ic50 = 0.19 uM | 24.305, 413.573 |
4LH5 | 2.19 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | MG, LF0 | ic50 = 0.23 uM | 24.305, 405.486 |
1C6Y | 2.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | MK1 | Ki = 0.31 nM | 613.789 |
1HSG | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | MK1 | Ki = 0.38 nM | 613.789 |
1HSH | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | MK1 | Ki = 2.45 nM | 613.789 |
1SGU | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | MK1 | Ki = 4235 nM | 613.789 |
1K6C | 2.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | MK1, ACT | Kd = 33 nM | 613.789, 59.044 |
1SDT | 1.3 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | MK1, CL | Ki = 540 pM | 613.789, 35.453 |
1SDV | 1.4 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | MK1, CL | Ki = 1810 pM | 613.789, 35.453 |
1EC3 | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | MS3 | Ki = 0.92 nM | 768.898 |
2Q54 | 1.85 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | MU1, ACT, PO4 | Ki = 0.98 nM | 656.768, 59.044, 94.971 |
6ONE | 2.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | NON-ENZYME OTHER | MVY, EPE, NAG | 314.74, 238.305, 221.208 | |
4INB | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | NON-ENZYME OTHER | NA, 1F6 | ic50 = 0.89 uM | 22.99, 419.397 |
6DJ1 | 1.26 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, AB1, CL | Ki = 0.031 nM | 22.99, 628.801, 35.453 |
2IEO | 1.53 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, CL, 017 | Ki = 3.2 nM | 22.99, 35.453, 547.664 |
3NU4 | 1.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, CL, 478 | Ki = 1.5 nM | 22.99, 35.453, 505.627 |
3PWM | 1.46 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, CL, ACT, 017 | 22.99, 35.453, 59.044, 547.664 | |
2QD6 | 1.28 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, CL, ACT, 065 | Ki = 2.1 nM | 22.99, 35.453, 59.044, 576.658 |
2QD8 | 1.35 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, CL, ACT, 065 | Ki = 0.85 nM | 22.99, 35.453, 59.044, 576.658 |
2Z4O | 1.6 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, CL, ACT, 065 | Ki = 0.27 nM | 22.99, 35.453, 59.044, 576.658 |
3NU5 | 1.29 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, CL, ACT, 478 | Ki = 4.5 nM | 22.99, 35.453, 59.044, 505.627 |
3NU6 | 1.16 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, CL, ACT, 478 | Ki = 0.5 nM | 22.99, 35.453, 59.044, 505.627 |
5DGU | 1.22 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, CL, ACT, 5B7 | Ki = 0.0045 nM | 22.99, 35.453, 59.044, 606.727 |
6U7P | 1.13 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, FMT, B4R, CL, GOL | 22.99, 46.025, 590.493, 35.453, 92.094 | |
6B4N | 1.3 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, G53, CL | Ki = 27.9 pM | 22.99, 657.731, 35.453 |
2F81 | 1.25 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, GOL, CL, 017 | Ki = 0.03 nM | 22.99, 92.094, 35.453, 547.664 |
3BVB | 1.3 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, GOL, CL, 017 | Ka = 3170000 M^-1 | 22.99, 92.094, 35.453, 547.664 |
3NU3 | 1.02 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, GOL, CL, 478 | Ki = 0.15 nM | 22.99, 92.094, 35.453, 505.627 |
3S54 | 1.42 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, GOL, CL, ACT, 017 | Ki = 0.23 nM | 22.99, 92.094, 35.453, 59.044, 547.664 |
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