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3CKT | 1.65 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | YDP, CL | Ki = 0.48 uM | 603.753, 35.453 |
2ZGA | 1.65 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | YDP | Ki = 0.48 uM | 603.753 |
4CIE | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | Y7N, ACY, CL, SO4 | 422.474, 60.052, 35.453, 96.063 | |
1BV7 | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | XV6 | Ki = 0.5 nM | 758.908 |
1BV9 | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | XV6 | Ki = 1.1 nM | 758.908 |
1BWA | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | XV6 | Ki = 2.5 nM | 758.908 |
1QBR | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | XV6 | Ki = 0.027 nM | 758.908 |
1K6P | 2.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | XN3, ACT | Kd = 44 nM | 656.811, 59.044 |
1K6V | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | XN2, ACT | Kd = 120 nM | 670.837, 59.044 |
1K6T | 2.25 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | XN1, ACT | Kd = 24 nM | 627.816, 59.044 |
1HVR | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | XK2 | Ki = 0.31 nM | 606.752 |
4CIG | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | X0P, ACT, SO4 | Kd = 214 uM | 498.57, 59.044, 96.063 |
4CFA | 2.05 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | WOP, SO4 | 475.493, 96.063 | |
4CJQ | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | VXO, SO4, ACT | Kd = 256 uM | 436.5, 96.063, 59.044 |
4CER | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | VL4, CL, SO4 | 496.552, 35.453, 96.063 | |
1MT7 | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | VAL SER GLN ASN TYR PRO ILE VAL GLN ASN, ACT | 904.056, 59.044 | |
8HVP | 2.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | VAL SER GLN ASN LOV ILE VAL | Ki < 1 nM | 872.075 |
4PHV | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | VAC | ic50 = 0.67 nM | 618.761 |
1HPO | 2.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | UNI | Ki = 0.6 nM | 504.597 |
1S1T | 2.4 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.49 | UC1, PO4 | 335.848, 94.971 | |
4CHO | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | U2Z, EDO, ACT, GOL, SO4 | 217.267, 62.068, 59.044, 92.094, 96.063 | |
1A9M | 2.3 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | U0E | Ki = 119 nM | 596.762 |
1AXA | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | U0E | 596.762 | |
1GNM | 2.3 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | U0E | Ki = 560 nM | 596.762 |
1GNN | 2.3 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | U0E | Ki = 2100 nM | 596.762 |
1GNO | 2.3 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | U0E | Ki = 20 nM | 596.762 |
1RTH | 2.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.49 | U05 | ic50 = 0.4 uM | 298.297 |
1UPJ | 2.22 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | U01 | 373.24 | |
2NPH | 1.65 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | TYR VAL ASP GLY ALA, ALA GLU THR PHE | 522.535, 465.483 | |
1SP5 | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | TYR ASP GLN ILE LEU, DMS, CL, BME | 649.722, 78.133, 35.453, 78.133 | |
4FM6 | 1.4 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | TYR ASP GLN ILE ILE ILE, NA, GOL, CL | 485.582, 22.99, 92.094, 35.453 | |
4FL8 | 1.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | TYR ASP GLN ILE IL0 ILE GLU, GOL, GLN ILE IL0 ILE GLU ILE ALA, CL | 801.916, 92.094, 743.944, 35.453 | |
1HYZ | 2.3 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | TTO, SO4, CL | ic50 = 380 uM | 415.336, 96.063, 35.453 |
1HYV | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | TTA, SO4, CL | ic50 > 5 mM | 383.337, 96.063, 35.453 |
2RKI | 2.3 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.49 | TT1, SO4, MG, GOL, CL | 397.944, 96.063, 24.305, 92.094, 35.453 | |
6DIF | 1.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | TPV, GOL, CL, NA | Ki = 0.019 nM | 602.664, 92.094, 35.453, 22.99 |
2O4L | 1.33 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | TPV, GOL, CL | Kd = 608 pM | 602.664, 92.094, 35.453 |
2O4P | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | TPV, GOL | Kd = 19 pM | 602.664, 92.094 |
6DIL | 1.48 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | TPV, CL, GOL, ACT, NA | Ki = 7.6 nM | 602.664, 35.453, 92.094, 59.044, 22.99 |
1D4S | 2.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | TPV | Ki = 0.008 nM | 602.664 |
1D4Y | 1.97 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | TPV | Ki = 0.008 nM | 602.664 |
4NJU | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME HYDROLASES | TPV | 602.664 | |
3OUC | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | THR ILE MET MET GLN ARG GLY | 837.058 | |
1AID | 2.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | THK, CL | Ki = 15 uM | 452.048, 35.453 |
2AID | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | THK, CL | Ki = 15 uM | 452.048, 35.453 |
6VOE | 1.3 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | T2R, ACT, NA, CL | ic50 = 0.3 nM | 656.789, 59.044, 22.99, 35.453 |
2ZD1 | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.49 | T27, SO4, EDO | 366.419, 96.063, 62.068 | |
3BGR | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.49 | T27, EDO | 366.419, 62.068 | |
4CGF | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | SO4, UJ6, EDO, ACT | 96.063, 311.289, 62.068, 59.044 | |
2NMY | 1.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | SO4, ROC, NA, CL | 96.063, 670.841, 22.99, 35.453 |