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1C70 | 2.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | L75 | Ki = 0.05 nM | 652.822 |
1HVS | 2.25 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | A77 | Ki = 50 pM | 794.981 |
4DJQ | 1.4 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, M86 | Ki = 0.048 nM | 94.971, 576.705 |
4Q1Y | 1.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | ACT, 017, PO4 | Ki = 45 pM | 59.044, 547.664, 94.971 |
2QI4 | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, MZ6, ACT | Ki = 0.036 nM | 94.971, 567.719, 59.044 |
2O4K | 1.6 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | DR7, CL | Kd = 35 pM | 704.855, 35.453 |
1MSM | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | JE2 | Kd = 33 pM | 575.718 |
2O4S | 1.54 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, CL, AB1 | Kd = 31 pM | 92.094, 35.453, 628.801 |
6DJ1 | 1.26 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | AB1, CL, NA | Ki = 0.031 nM | 628.801, 35.453, 22.99 |
2F81 | 1.25 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, GOL, CL, 017 | Ki = 0.03 nM | 22.99, 92.094, 35.453, 547.664 |
4DJP | 1.4 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, M73 | Ki = 0.028 nM | 94.971, 564.691 |
6B4N | 1.3 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, G53, CL | Ki = 27.9 pM | 22.99, 657.731, 35.453 |
1QBR | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | XV6 | Ki = 0.027 nM | 758.908 |
2QI6 | 1.85 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, MZ8 | Ki = 0.027 nM | 94.971, 553.693 |
6PJL | 1.99 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | SO4, OQA | Ki = 0.027 nM | 96.063, 611.726 |
6DH1 | 1.97 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | SO4, K13 | Ki = 26.1 pM | 96.063, 561.69 |
6DH0 | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 017 | Ki = 25.6 pM | 547.664 |
5UOV | 1.33 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 8FP, NA, GOL, CL, ACT | Ki = 0.025 nM | 704.898, 22.99, 92.094, 35.453, 59.044 |
1QBT | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 146 | Ki = 0.024 nM | 824.924 |
1DIF | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | BME, A85 | Ki = 22 pM | 78.133, 830.962 |
2PK5 | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, 075 | Kd = 20 pM | 92.094, 803.943 |
2O4P | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | TPV, GOL | Kd = 19 pM | 602.664, 92.094 |
5TYS | 2.01 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 7OA | ic50 = 0.019 nM | 706.82 |
6DIF | 1.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | TPV, GOL, CL, NA | Ki = 0.019 nM | 602.664, 92.094, 35.453, 22.99 |
6PJG | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | ORV | Ki = 0.019 nM | 569.646 |
6PJD | 1.89 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | SO4, OQY | Ki = 0.018 nM | 96.063, 611.726 |
6PJC | 1.97 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | SO4, OR1 | Ki = 0.017 nM | 96.063, 602.717 |
3GI4 | 1.85 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, K60, ACT | Ki = 0.016 nM | 94.971, 677.688, 59.044 |
1HXW | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | RIT | Ki = 15 pM | 720.944 |
5WLO | 1.27 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | ACT, GR7, GOL, CL, NA | Ki = 0.015 nM | 59.044, 630.749, 92.094, 35.453, 22.99 |
1T3R | 1.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, 017 | Ki = 14 pM | 94.971, 547.664 |
2QI5 | 1.85 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, MZ7 | Ki = 0.014 nM | 94.971, 588.782 |
3I7E | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | DJR | Ki = 14 pM | 562.675 |
5ULT | 1.53 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | CL, NA, 8FM | Ki = 0.014 nM | 35.453, 22.99, 588.712 |
6BZ2 | 1.67 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | ACT, CL, 7OA, NA | Ki = 14 pM | 59.044, 35.453, 706.82, 22.99 |
2PK6 | 1.45 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | O33, GOL | Kd = 13 pM | 771.945, 92.094 |
6PJM | 1.93 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | OQV, SO4 | Ki = 0.013 nM | 611.726, 96.063 |
6DH2 | 1.98 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | SO4, A60 | Ki = 12.8 pM | 96.063, 575.717 |
6CDL | 1.25 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GR5, CL, NA, ACT, GOL | Ki = 0.012 nM | 720.847, 35.453, 22.99, 59.044, 92.094 |
3LZS | 1.95 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | ACT, 017 | Kd = 0.0109 nM | 59.044, 547.664 |
4KB9 | 1.29 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | G79, GOL, NA, CL, ACT | Ki = 0.01 nM | 616.765, 92.094, 22.99, 35.453, 59.044 |
5DGW | 1.62 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 5B5, NA, CL | Ki = 0.009 nM | 619.769, 22.99, 35.453 |
1D4S | 2.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | TPV | Ki = 0.008 nM | 602.664 |
1D4Y | 1.97 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | TPV | Ki = 0.008 nM | 602.664 |
3M9F | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | CL, 595 | ic50 = 0.007 nM | 35.453, 650.828 |
4Q1X | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, 017, GOL | Ki = 7 pM | 94.971, 547.664, 92.094 |
2I4V | 1.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | DJR | Ki = 6.3 pM | 562.675 |
3GI5 | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, K62 | Ki = 0.006 nM | 94.971, 651.727 |
3GI6 | 1.84 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, D78 | Ki = 0.006 nM | 94.971, 663.704 |
3OK9 | 1.27 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, GOL, G52, CL | Ki = 5.9 pM | 22.99, 92.094, 604.712, 35.453 |
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