2HS1 | 0.84 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | DMS, CL, 017 | Ki = 3.3 nM | 78.133, 35.453, 547.664 |
5YOK | 0.85 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 8Z0, GOL | | 756.907, 92.094 |
3A2O | 0.88 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | KNJ, GOL | Ki = 0.83 nM | 568.727, 92.094 |
3FX5 | 0.93 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | KNI, GOL | Ki < 1 nM | 667.839, 92.094 |
2NMZ | 0.97 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | SO4, ROC | | 96.063, 670.841 |
6IXD | 1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | CL, GOL, B0F, SO4 | Ki = 0.16 nM | 35.453, 92.094, 873.092, 96.063 |
3NU3 | 1.02 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, GOL, CL, 478 | Ki = 0.15 nM | 22.99, 92.094, 35.453, 505.627 |
1NH0 | 1.03 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | SO4, KI2 PHE GLU GLU NH2, BME | Ki = 0.18 nM | 96.063, 732.767, 78.133 |
2J9J | 1.04 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | SO4, GOL, ACT, ACE SER LEU ASN JG3 ILE VME | | 96.063, 92.094, 59.044, 818.006 |
3BVA | 1.05 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, 2NC | Ka = 3300000 M^-1 | 92.094, 770.983 |
2JE4 | 1.07 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | SO4, GOL, ACT, ACE SER LEU ASN JG3 ILE VME | | 96.063, 92.094, 59.044, 818.006 |
3MWS | 1.09 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | CL, 017 | | 35.453, 547.664 |
2AVM | 1.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, ACY, 2NC | Ki = 2 uM | 92.094, 60.052, 770.983 |
2AVO | 1.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | SO4, MK1, GOL, DMS, ACY | Ki = 1.4 nM | 96.063, 613.789, 92.094, 78.133, 60.052 |
2AVS | 1.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | SO4, PO4, MK1, DMS, ACY | Ki = 27 nM | 96.063, 94.971, 613.789, 78.133, 60.052 |
2IDW | 1.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, GOL, DMS, CL, ACY, 017 | Ki = 1.3 nM | 94.971, 92.094, 78.133, 35.453, 60.052, 547.664 |
2NMY | 1.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | SO4, ROC, NA, CL | | 96.063, 670.841, 22.99, 35.453 |
4EJD | 1.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 1F1, IVA VAL VAL STA ALA STA, GOL, BME | Kd = 14.5 uM | 161.157, 696.992, 92.094, 78.133 |
2QD7 | 1.11 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, GOL, DMS, 065 | Ki = 0.8 nM | 94.971, 92.094, 78.133, 576.658 |
6BRA | 1.11 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | SER GLY ILE PHE LEU GLU THR SER, CL | | 854.956, 35.453 |
6CDJ | 1.13 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, GR8, CL, GOL, ACT | Ki = 2 pM | 22.99, 720.847, 35.453, 92.094, 59.044 |
6U7P | 1.13 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, FMT, B4R, CL, GOL | | 22.99, 46.025, 590.493, 35.453, 92.094 |
6DV4 | 1.14 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, ACT, GA5, CL, NA | Ki = 1.6 nM | 92.094, 59.044, 695.865, 35.453, 22.99 |
5IVT | 1.15 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | ACT, CL, 6EE | ic50 = 0.8 nM | 59.044, 35.453, 674.034 |
3NU6 | 1.16 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, CL, ACT, 478 | Ki = 0.5 nM | 22.99, 35.453, 59.044, 505.627 |
3OXC | 1.16 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | SO4, ROC, FMT | Ki = 3.9 nM | 96.063, 670.841, 46.025 |
5JG1 | 1.16 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 6KR, GOL, NA, CL | Ki = 1.9 nM | 634.824, 92.094, 22.99, 35.453 |
6VCE | 1.18 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, G6R, NA, CL | ic50 = 79 pM | 92.094, 704.847, 22.99, 35.453 |
1K1T | 1.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | SO4, 0Q4 | | 96.063, 833.053 |
1T3R | 1.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, 017 | Ki = 14 pM | 94.971, 547.664 |
2J9K | 1.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | SO4, GOL, ACT, 2NC | | 96.063, 92.094, 59.044, 770.983 |
2NNP | 1.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | SO4, ROC, GOL, ACY | | 96.063, 670.841, 92.094, 60.052 |
2QCI | 1.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | ACT, NA, 065, CL | Ki = 4.6 nM | 59.044, 22.99, 576.658, 35.453 |
3CYX | 1.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | ROC, PO4, NA, GOL, ACY | Ki = 10 nM | 670.841, 94.971, 22.99, 92.094, 60.052 |
3NU4 | 1.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, CL, 478 | Ki = 1.5 nM | 22.99, 35.453, 505.627 |
4FL8 | 1.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | TYR ASP GLN ILE IL0 ILE GLU, GOL, GLN ILE IL0 ILE GLU ILE ALA, CL | | 801.916, 92.094, 743.944, 35.453 |
6DIF | 1.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | TPV, GOL, CL, NA | Ki = 0.019 nM | 602.664, 92.094, 35.453, 22.99 |
6DV0 | 1.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, GA8, CL, NA | Ki = 0.38 nM | 92.094, 697.904, 35.453, 22.99 |
6OGT | 1.21 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME HYDROLASES | JDY, EDO, GOL | ic50 = 31 nM | 688.83, 62.068, 92.094 |
2F8G | 1.22 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, GOL, CL, ACY, 017 | Ki = 2 nM | 22.99, 92.094, 35.453, 60.052, 547.664 |
2HS2 | 1.22 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | DMS, CL, 017 | Ki = 4.9 nM | 78.133, 35.453, 547.664 |
5DGU | 1.22 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | ACT, 5B7, NA, CL | Ki = 0.0045 nM | 59.044, 606.727, 22.99, 35.453 |
6E9A | 1.22 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | FMT, CL, J0S, NA | Ki = 0.0012 nM | 46.025, 35.453, 575.674, 22.99 |
1SDU | 1.25 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | ACT, SO4, MK1 | Ki = 86 pM | 59.044, 96.063, 613.789 |
2F81 | 1.25 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, GOL, CL, 017 | Ki = 0.03 nM | 22.99, 92.094, 35.453, 547.664 |
2NNK | 1.25 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | ROC, NA, GOL, CL, ACY | | 670.841, 22.99, 92.094, 35.453, 60.052 |
6CDL | 1.25 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | ACT, GOL, GR5, CL, NA | Ki = 0.012 nM | 59.044, 92.094, 720.847, 35.453, 22.99 |
6VOD | 1.25 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, T1R, CL, GOL, FMT | ic50 = 38 nM | 22.99, 588.712, 35.453, 92.094, 46.025 |
3S43 | 1.26 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | IOD, GOL, 478 | Ki = 2.53 nM | 126.904, 92.094, 505.627 |
6DJ1 | 1.26 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | AB1, CL, NA | Ki = 0.031 nM | 628.801, 35.453, 22.99 |
3OK9 | 1.27 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, GOL, G52, CL | Ki = 5.9 pM | 22.99, 92.094, 604.712, 35.453 |
5UPZ | 1.27 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, CL, 8HD, NA | Ki = 0.63 nM | 92.094, 35.453, 662.796, 22.99 |
5WLO | 1.27 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | ACT, GR7, GOL, CL, NA | Ki = 0.015 nM | 59.044, 630.749, 92.094, 35.453, 22.99 |
2QD6 | 1.28 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, CL, ACT, 065 | Ki = 2.1 nM | 22.99, 35.453, 59.044, 576.658 |
3NU5 | 1.29 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, CL, ACT, 478 | Ki = 4.5 nM | 22.99, 35.453, 59.044, 505.627 |
4KB9 | 1.29 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | G79, GOL, NA, CL, ACT | Ki = 0.01 nM | 616.765, 92.094, 22.99, 35.453, 59.044 |
1SDT | 1.3 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | MK1, CL | Ki = 540 pM | 613.789, 35.453 |
2A1E | 1.3 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, IPF, GOL, DMS, CL, ACT | | 22.99, 905.092, 92.094, 78.133, 35.453, 59.044 |
2IEN | 1.3 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, GOL, CL, ACY, 017 | Ki = 1 nM | 22.99, 92.094, 35.453, 60.052, 547.664 |
3BVB | 1.3 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | CL, 017, NA, GOL | Ka = 3170000 M^-1 | 35.453, 547.664, 22.99, 92.094 |
3KFR | 1.3 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | BME, 3TL, 1F1 | | 78.133, 909.077, 161.157 |
4DQE | 1.3 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | ACT, 017 | | 59.044, 547.664 |
6B4N | 1.3 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, G53, CL | Ki = 27.9 pM | 22.99, 657.731, 35.453 |
6E7J | 1.3 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | HWY, NA, CL | Ki = 0.33 nM | 651.77, 22.99, 35.453 |
6VOE | 1.3 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | T2R, ACT, NA, CL | ic50 = 0.3 nM | 656.789, 59.044, 22.99, 35.453 |
4FLG | 1.31 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, ILE GLU ILE, GOL, GLN ILE ILE, CL, ASP GLN ILE ILE | | 22.99, 315.37, 92.094, 315.414, 35.453, 386.493 |
4J55 | 1.31 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 031 | | 601.711 |
6DJ7 | 1.31 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, G10, ACT, CL, NA | Ki = 1.9 nM | 92.094, 583.645, 59.044, 35.453, 22.99 |
6KMP | 1.31 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | KVS | | 800.986 |
2O4L | 1.33 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | TPV, GOL, CL | Kd = 608 pM | 602.664, 92.094, 35.453 |
5UOV | 1.33 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 8FP, NA, GOL, CL, ACT | Ki = 0.025 nM | 704.898, 22.99, 92.094, 35.453, 59.044 |
6U7O | 1.33 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | Q1D, NA, FMT, CL, GOL | Ki = 15.5 uM | 602.504, 22.99, 46.025, 35.453, 92.094 |
1T7I | 1.35 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, ACT, 017 | | 94.971, 59.044, 547.664 |
2BB9 | 1.35 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | AKC | ic50 = 0.44 nM | 625.711 |
2HB3 | 1.35 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, GRL, GOL, CL | Ki = 0.0045 nM | 22.99, 560.702, 92.094, 35.453 |
2QD8 | 1.35 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, CL, ACT, 065 | Ki = 0.85 nM | 22.99, 35.453, 59.044, 576.658 |
3NUO | 1.35 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | IOD, 478 | Ki = 0.16 nM | 126.904, 505.627 |
6DJ2 | 1.36 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | AB1, CL, NA | Ki = 4.5 nM | 628.801, 35.453, 22.99 |
3UCB | 1.38 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 017 | Kd = 41 nM | 547.664 |
4U7V | 1.38 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | BME, 3EN | Ki = 3.2 uM | 78.133, 524.675 |
1SDV | 1.4 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | MK1, CL | Ki = 1810 pM | 613.789, 35.453 |
2XDE | 1.4 | HUMAN IMMUNODEFICIENCY VIRUS 1 | NON-ENZYME OTHER | 1B0 | Kd = 3.42 uM | 425.522 |
4DJP | 1.4 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, M73 | Ki = 0.028 nM | 94.971, 564.691 |
4DJQ | 1.4 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, M86 | Ki = 0.048 nM | 94.971, 576.705 |
4FM6 | 1.4 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | TYR ASP GLN ILE ILE ILE, NA, GOL, CL | | 485.582, 22.99, 92.094, 35.453 |
2QNP | 1.41 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | QN2, CL | Ki = 0.39 uM | 813.508, 35.453 |
6OGQ | 1.41 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME HYDROLASES | PEG, GOL, JDV, SO4 | ic50 = 26 nM | 106.12, 92.094, 688.83, 96.063 |
3S54 | 1.42 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, GOL, CL, ACT, 017 | Ki = 0.23 nM | 22.99, 92.094, 35.453, 59.044, 547.664 |
2FNT | 1.44 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, ARG GLN VAL ASN PHE LEU GLY LYS ILE ASN, ACT | | 94.971, 675.808, 59.044 |
2F80 | 1.45 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | SO4, CL, 017 | Ki = 6.6 nM | 96.063, 35.453, 547.664 |
2PK6 | 1.45 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | O33, GOL | Kd = 13 pM | 771.945, 92.094 |
3PWR | 1.45 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | ROC, GOL, CL | | 670.841, 92.094, 35.453 |
3PWM | 1.46 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, CL, ACT, 017 | | 22.99, 35.453, 59.044, 547.664 |
5IVS | 1.46 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 6EF, CL | ic50 = 6.1 nM | 650.763, 35.453 |
6B3F | 1.46 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | CKV, CL | | 621.712, 35.453 |
6O48 | 1.46 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | FMT, GOL, 0Q4, NA, CL | Ki = 75 nM | 46.025, 92.094, 833.053, 22.99, 35.453 |
6OYD | 1.46 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NKA | ic50 = 0.12 nM | 674.78 |
2QNN | 1.48 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | QN1, GOL, CL | Ki = 0.07 uM | 783.76, 92.094, 35.453 |
6B38 | 1.48 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | CKM, CL | | 621.712, 35.453 |
6DIL | 1.48 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | TPV, CL, GOL, ACT, NA | Ki = 7.6 nM | 602.664, 35.453, 92.094, 59.044, 22.99 |