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6MCR | 1.48 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | JDY, EDO | 688.83, 62.068 | |
5JFP | 1.49 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 6KK, CL, NA | Ki = 0.48 nM | 620.797, 35.453, 22.99 |
1XL2 | 1.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, CL, 189 | Ki = 1.5 uM | 92.094, 35.453, 577.777 |
2AVV | 1.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | MK1, CL, ACY | Ki = 0.55 nM | 613.789, 35.453, 60.052 |
2FGV | 1.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | QNC ASN HPH DIQ NTB, PO4 | Kd = 760 nM | 670.855, 94.971 |
2I4D | 1.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | QFI | Ki = 2.1 pM | 672.681 |
2I4U | 1.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | DJR | Ki = 2.7 pM | 562.675 |
2I4V | 1.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | DJR | Ki = 6.3 pM | 562.675 |
2PWR | 1.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, G4G, CL | Ki = 0.26 uM | 92.094, 647.764, 35.453 |
3NUJ | 1.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | IOD, 478 | Ki = 0.41 nM | 126.904, 505.627 |
3S53 | 1.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, IOD, 017 | Ki = 0.23 nM | 94.971, 126.904, 547.664 |
4DQB | 1.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | PO4, EDO, DMS, 017 | 94.971, 62.068, 78.133, 547.664 | |
4Q1Y | 1.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | ACT, 017, PO4 | Ki = 45 pM | 59.044, 547.664, 94.971 |
5IVR | 1.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 6EG, CL | 566.69, 35.453 | |
5T2Z | 1.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME HYDROLASES | 017 | 547.664 | |
5YOJ | 1.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 8Z0, GOL | 756.907, 92.094 | |
6B3G | 1.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | CL, CKY | 35.453, 621.712 | |
6OTG | 1.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, FMT, 4UY | Ki = 31.4 nM | 92.094, 46.025, 591.716 |
6MCS | 1.52 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | JDV | 688.83 | |
2IEO | 1.53 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, CL, 017 | Ki = 3.2 nM | 22.99, 35.453, 547.664 |
5ULT | 1.53 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | CL, NA, 8FM | Ki = 0.014 nM | 35.453, 22.99, 588.712 |
6OGP | 1.53 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | EDO, MJD | ic50 = 0.055 uM | 62.068, 692.77 |
2O4S | 1.54 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, CL, AB1 | Kd = 31 pM | 92.094, 35.453, 628.801 |
3ZPT | 1.54 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | M8Y, CL | Ki = 3.1 nM | 728.716, 35.453 |
4E43 | 1.54 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, DMS, BME, ASN LEU LEU GLN LYS LYS, ACT | 92.094, 78.133, 78.133, 729.945, 59.044 | |
6OYR | 1.54 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NJY | ic50 = 0.29 nM | 674.78 |
1DAZ | 1.55 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 0Q4 | 833.053 | |
1K1U | 1.55 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 0Q4 | 833.053 | |
2I4W | 1.55 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | KGQ | Ki = 2.6 pM | 728.787 |
2I4X | 1.55 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | KGQ | Ki = 1.9 pM | 728.787 |
2PQZ | 1.55 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | G0G, CL | Ki = 2.15 uM | 561.715, 35.453 |
3ZPS | 1.55 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | EQM, CL | 730.732, 35.453 | |
4DJR | 1.55 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 0KJ, PO4 | Ki = 0.003 nM | 588.739, 94.971 |
4J54 | 1.55 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | ACT, G52, IOD | 59.044, 604.712, 126.904 | |
5TKK | 1.55 | HUMAN IMMUNODEFICIENCY VIRUS 1 | NON-ENZYME OTHER | ALA VAL GLY ILE GLY ALA VAL PHE | 471.579 | |
5IVQ | 1.57 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 6EH, CL | 425.521, 35.453 | |
2FDD | 1.58 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 385 | ic50 = 4.8 nM | 703.823 |
2R43 | 1.58 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GOL, G3G, CL | Ki = 1 uM | 92.094, 591.744, 35.453 |
6BXQ | 1.58 | HUMAN IMMUNODEFICIENCY VIRUS 1 | NON-ENZYME IMMUNE | ARG VAL LYS GLU LYS TYR GLN HIS LEU TRP | 1098.3 | |
2F3K | 1.6 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | RO1, PO4 | Kd = 0.95 nM | 711.911, 94.971 |
2FXD | 1.6 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | SO4, DR7, ACT | ic50 = 12 nM | 96.063, 704.855, 59.044 |
2O4K | 1.6 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | DR7, CL | Kd = 35 pM | 704.855, 35.453 |
2Z4O | 1.6 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | NA, CL, ACT, 065 | Ki = 0.27 nM | 22.99, 35.453, 59.044, 576.658 |
3OU4 | 1.6 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME HYDROLASES | PHE ASN PHE PRO GLN ILE THR | 865.986 | |
3OUB | 1.6 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | GLN VAL ASN PHE LEU GLY LYS | 789.932 | |
3VQ8 | 1.6 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | CD, BCU, CL, SO4 | 112.411, 164.201, 35.453, 96.063 | |
5KR1 | 1.6 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 017 | Ki = 0.32 nM | 547.664 |
6B3C | 1.6 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | CKS, CL | 621.712, 35.453 | |
6C8X | 1.61 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | BVR, GOL, CL | Ki = 0.5 pM | 575.459, 92.094, 35.453 |
5DGW | 1.62 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 5B5, NA, CL | Ki = 0.009 nM | 619.769, 22.99, 35.453 |
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