1Y63 | 1.7 | LEISHMANIA MAJOR | NON-ENZYME OTHER | NA, MN, BR, ADP | | 22.99, 54.938, 79.904, 427.201 |
2X77 | 2.1 | LEISHMANIA MAJOR | NON-ENZYME OTHER | MG, GDP | | 24.305, 443.201 |
1XTP | 1.94 | LEISHMANIA MAJOR | ENZYME TRANSFERASES | SAI | | 431.306 |
3KFL | 2 | LEISHMANIA MAJOR | ENZYME 6.1.1.10 | ZN, POP, MG, ME8, FMT, EDO | | 65.409, 175.959, 24.305, 478.417, 46.025, 62.068 |
6SWX | 1.95 | LEISHMANIA MAJOR | ENZYME 6.1.1.10 | LWN | ic50 = 2.06 uM | 348.307 |
5L2R | 2.05 | LEISHMANIA MAJOR | ENZYME 4.2.1.2 | PEG, SF4, GOL, MLA, LMR | ic50 = 9.8 mM | 106.12, 351.64, 92.094, 104.061, 134.087 |
6MSN | 1.59 | LEISHMANIA MAJOR | ENZYME 4.2.1.2 | JYD, SF4 | Ki = 8.9 uM | 150.153, 351.64 |
6MSO | 2.05 | LEISHMANIA MAJOR | ENZYME 4.2.1.2 | JYD, SF4, 1PE, GOL | Ki = 3 uM | 150.153, 351.64, 238.278, 92.094 |
2CJE | 2.34 | LEISHMANIA MAJOR | ENZYME 3.6.1.23 | DUN, MG | | 387.177, 24.305 |
2YAY | 1.86 | LEISHMANIA MAJOR | ENZYME 3.6.1.23 | DUP, CA | Kd = 0.8 uM | 467.157, 40.078 |
2YAZ | 2.4 | LEISHMANIA MAJOR | ENZYME 3.6.1.23 | UMP, SO4, MG | Kd = 7.3 uM | 308.182, 96.063, 24.305 |
2YB0 | 2.28 | LEISHMANIA MAJOR | ENZYME 3.6.1.23 | SO4, DUR | Kd = 140 uM | 96.063, 228.202 |
5NTH | 2.5 | LEISHMANIA MAJOR | ENZYME 3.4.11.- | BB2, BCT, MN | | 385.498, 61.017, 54.938 |
2R8Q | 1.5 | LEISHMANIA MAJOR | ENZYME 3.1.4.17 | ZN, MG, IBM | ic50 = 580 uM | 65.409, 24.305, 222.244 |
2OEG | 2.3 | LEISHMANIA MAJOR | ENZYME 2.7.7.9 | UPG | | 566.302 |
3OH0 | 2.15 | LEISHMANIA MAJOR | ENZYME 2.7.7.64 | GOL, UTP | | 92.094, 484.141 |
3OH1 | 2.18 | LEISHMANIA MAJOR | ENZYME 2.7.7.64 | UGB, GOL | | 580.285, 92.094 |
3OH2 | 2.14 | LEISHMANIA MAJOR | ENZYME 2.7.7.64 | GOL, GDU | | 92.094, 566.302 |
3OH3 | 2.03 | LEISHMANIA MAJOR | ENZYME 2.7.7.64 | UAD, GOL | | 536.276, 92.094 |
3OH4 | 2.21 | LEISHMANIA MAJOR | ENZYME 2.7.7.64 | UPG, GOL | | 566.302, 92.094 |
3NGU | 2.29 | LEISHMANIA MAJOR | ENZYME 2.7.4.6 | ADP | | 427.201 |
2HFU | 2 | LEISHMANIA MAJOR | ENZYME 2.7.1.36 | MEV | | 147.149 |
4UXH | 2.4 | LEISHMANIA MAJOR | ENZYME 2.7.1.21 | T5A, ZN | ic50 = 1.1 uM | 891.354, 65.409 |
4JZB | 1.9 | LEISHMANIA MAJOR | ENZYME 2.5.1.1 | IPE, NA, CA, P2H | Kd = 342.5 nM | 246.092, 22.99, 40.078, 360.216 |
4JZX | 1.8 | LEISHMANIA MAJOR | ENZYME 2.5.1.1 | 476, IPE, CA | Kd = 198.6 nM | 324.227, 246.092, 40.078 |