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2VVO | 1.85 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 5.3.1.6 | A6P | ic50 = 6.3 mM | 260.136 |
4DDK | 1.75 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 6.3.2.1 | EOH, EDO, 0HN, GOL | Kd = 5.13 mM | 46.068, 62.068, 166.131, 92.094 |
4DDM | 1.83 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 6.3.2.1 | EDO, 0HO, GOL, EOH | Kd = 3.48 mM | 62.068, 180.184, 92.094, 46.068 |
4EFK | 1.7 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 6.3.2.1 | EOH, IMD, SO4, GOL, 0OC | Kd = 3.18 mM | 46.068, 69.085, 96.063, 92.094, 191.271 |
1RQ2 | 1.86 | MYCOBACTERIUM TUBERCULOSIS | NON-ENZYME CELL_CYCLE | CIT | ic50 = 3 mM | 192.124 |
4G46 | 1.52 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 1.14.-.- | TTY, SO4, HEM | Kd ~ 3 mM | 180.157, 96.063, 616.487 |
4G2G | 2.25 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 1.14.-.- | TDH, SO4, HEM, DMS | Kd ~ 2.8 mM | 253.256, 96.063, 616.487, 78.133 |
4KTJ | 1.35 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 1.14.-.- | SO4, HEM, KTJ | Kd = 1.9 mM | 96.063, 616.487, 175.187 |
2BET | 2.2 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 5.3.1.6 | DEZ | Ki = 1.7 mM | 216.083 |
4G47 | 1.34 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 1.14.-.- | TZF, SO4, HEM | Kd ~ 1.7 mM | 161.161, 96.063, 616.487 |
4G5Y | 1.8 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 6.3.2.1 | MG, 0OC, ATP, GOL, EOH | Kd = 1.69 mM | 24.305, 191.271, 507.181, 92.094, 46.068 |
4G44 | 1.24 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 1.14.-.- | TZM, SO4, HEM | Kd = 1.6 mM | 174.202, 96.063, 616.487 |
4IQ7 | 1.9 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 1.14.-.- | 1G9, HEM, SO4 | Kd = 1561 uM | 234.251, 616.487, 96.063 |
4EF6 | 1.94 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 6.3.2.1 | GOL, I2E, EOH, EDO | Kd = 1.18 mM | 92.094, 194.184, 46.068, 62.068 |
3IMC | 1.6 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 6.3.2.1 | SO4, GOL, EOH, BZ3 | Kd = 1100 uM | 96.063, 92.094, 46.068, 147.174 |
3IME | 2.39 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 6.3.2.1 | GOL, EOH, BZ2 | Kd = 1000 uM | 92.094, 46.068, 162.142 |
5OIC | 1.87 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 1.3.1.9 | NAD, ETX, 9VQ | ic50 < 1 mM | 663.425, 90.121, 188.226 |
4FZJ | 1.63 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 6.3.2.1 | EDO, 0W1, EOH, GOL | Kd = 0.74 mM | 62.068, 196.226, 46.068, 92.094 |
4G5F | 2.33 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 6.3.2.1 | EDO, 0JD, 15N, EOH, GOL | Kd = 0.7 mM, Kd = 0.88 mM | 62.068, 180.157, 180.157, 46.068, 92.094 |
5E5G | 1.95 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 2.5.1.54 | SO4, DTR, MN | Kd = 700 uM | 96.063, 204.225, 54.938 |
4DE5 | 2.25 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 6.3.2.1 | EDO, GOL, EOH, 0JD | Kd = 670 uM | 62.068, 92.094, 46.068, 180.157 |
4IPS | 1.2 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 1.14.-.- | SO4, HEM, GOL, 1G4 | Kd = 657 uM | 96.063, 616.487, 92.094, 312.363 |
6VS5 | 1.76 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 1.5.1.3 | CO, PO4, NDP, 9FH | Kd = 641 uM | 58.933, 94.971, 745.421, 202.209 |
4UNP | 2.3 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 2.7.4.9 | TXW | Kd = 590 uM | 202.252 |
3IOE | 1.95 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 6.3.2.1 | SO4, GOL, EOH, A7D | Kd = 540 uM | 96.063, 92.094, 46.068, 371.412 |
5JZS | 2.27 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 3.7.1.8 | FGZ | ic50 = 0.54 mM | 207.011 |
3CE6 | 1.6 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 3.3.1.1 | NAD, ADN | ic50 ~ 500 uM | 663.425, 267.241 |
4G48 | 1.5 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 1.14.-.- | HEM, SO4, PZB | Kd = 500 uM | 616.487, 96.063, 268.267 |
4DDH | 2.07 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 6.3.2.1 | EOH, GOL, MS0, EDO | Kd = 0.48 mM | 46.068, 92.094, 206.195, 62.068 |
4G45 | 1.53 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 1.14.-.- | SO4, MQN, HEM | Kd = 400 uM | 96.063, 158.2, 616.487 |
3IOB | 1.8 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 6.3.2.1 | SO4, GOL, EOH, A4D | Kd = 380 uM | 96.063, 92.094, 46.068, 283.307 |
4N8Q | 2.08 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 2.4.2.18 | FA0 | Ki = 380 uM | 155.126 |
4C6Z | 1.8 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 2.3.1.41 | K, TLE, M7U, EDO | Ki = 357 uM | 39.098, 224.319, 690.971, 62.068 |
5IBH | 2.02 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 1.14.-.- | SO4, HEM, 69R | Kd = 275 uM | 96.063, 616.487, 347.371 |
3ST6 | 1.75 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 4.1.3.- | RVE | Ki = 240 uM | 224.167 |
3IOC | 2.5 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 6.3.2.1 | GOL, A5D | Kd = 210 uM | 92.094, 405.494 |
3ISJ | 2.2 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 6.3.2.1 | SO4, GOL, EOH, A8D | Kd = 210 uM | 96.063, 92.094, 46.068, 268.289 |
1H0R | 2.1 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 4.2.1.10 | PO4, GOL, FA1, CL | Ki = 200 uM | 94.971, 92.094, 174.151, 35.453 |
3N7A | 2 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 4.2.1.10 | GOL, FA1 | Ki = 200 uM | 92.094, 174.151 |
2FF4 | 1.9 | MYCOBACTERIUM TUBERCULOSIS | NON-ENZYME OTHER | SER LEU GLU VAL TPO GLU ALA ASP THR | Kd = 185 uM | 823.727 |
4KTK | 1.4 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 1.14.-.- | SO4, HEM, KTK | Kd = 180 uM | 96.063, 616.487, 283.282 |
4QVB | 2.3 | MYCOBACTERIUM TUBERCULOSIS | ENZYME OXIDOREDUCTASES | PGO, NA, PDO, EDO, F42, FMT | Kd = 170 uM | 76.094, 22.99, 76.094, 62.068, 773.593, 46.025 |
5IBF | 1.7 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 1.14.-.- | HEM, SO4, 69W | Kd = 140 uM | 616.487, 96.063, 250.298 |
2YIM | 1.41 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 5.1.99.4 | PO4, MC4, GOL | Kd = 120 uM | 94.971, 864.626, 92.094 |
1MRS | 2 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 2.7.4.9 | SO4, MG, 5HU | Ki = 110 uM | 96.063, 24.305, 338.208 |
2VI5 | 2.3 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 2.5.1.9 | Y19, PO4, K | Ki = 110 uM | 332.31, 94.971, 39.098 |
1X8V | 1.55 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 1.14.13.70 | HEM, ESL | Kd = 100 uM | 616.487, 288.381 |
5E2L | 2.5 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 2.5.1.54 | CL, SO4, DPN, GOL, MN | Kd = 93 uM | 35.453, 96.063, 165.189, 92.094, 54.938 |
3N8K | 2.25 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 4.2.1.10 | D1X, CL | Kd = 90 uM | 155.108, 35.453 |
4X5E | 1.77 | MYCOBACTERIUM TUBERCULOSIS | ENZYME 2.4.2.18 | POP, MG, GOL, BE2 | Ki = 89 uM | 175.959, 24.305, 92.094, 137.136 |