1AQ1 | 2 | HOMO SAPIENS | ENZYME 2.7.11.22 | STU | 466.531 | |
1B38 | 2 | HOMO SAPIENS | ENZYME 2.7.11.22 | MG, ATP | Kd = 0.254 uM | 24.305, 507.181 |
1B39 | 2.1 | HOMO SAPIENS | ENZYME 2.7.11.22 | MG, ATP | Kd = 0.12 uM | 24.305, 507.181 |
1CKP | 2.05 | HOMO SAPIENS | ENZYME 2.7.11.22 | PVB, EDO | 432.904, 62.068 | |
1DI8 | 2.2 | HOMO SAPIENS | ENZYME 2.7.11.22 | DTQ | ic50 = 1 uM | 297.309 |
1DM2 | 2.1 | HOMO SAPIENS | ENZYME 2.7.11.22 | HMD, EDO | 324.133, 62.068 | |
1E1V | 1.95 | HOMO SAPIENS | ENZYME 2.7.11.22 | CMG | Ki = 12 uM | 247.296 |
1E1X | 1.85 | HOMO SAPIENS | ENZYME 2.7.11.22 | NW1 | Ki = 1.3 uM | 251.285 |
1E9H | 2.5 | HOMO SAPIENS | ENZYME 2.7.11.22 | INR | ic50 = 35 nM | 342.326 |
1FIN | 2.3 | HOMO SAPIENS | ENZYME 2.7.11.22 | ATP | 507.181 | |
1FVT | 2.2 | HOMO SAPIENS | ENZYME 2.7.11.22 | 106 | 395.231 | |
1GII | 2 | HOMO SAPIENS | ENZYME 2.7.11.22 | 1PU | 308.335 | |
1GIJ | 2.2 | HOMO SAPIENS | ENZYME 2.7.11.22 | 2PU | 366.417 | |
1GZ8 | 1.3 | HOMO SAPIENS | ENZYME 2.7.11.22 | MBP | 235.243 | |
1H00 | 1.6 | HOMO SAPIENS | ENZYME 2.7.11.22 | FCP, FAP | ic50 = 38 uM, ic50 = 38 uM | 415.436, 415.436 |
1H01 | 1.79 | HOMO SAPIENS | ENZYME 2.7.11.22 | GOL, FBL, FAL | ic50 = 22 uM, ic50 = 22 uM | 92.094, 448.346, 448.346 |
1H07 | 1.85 | HOMO SAPIENS | ENZYME 2.7.11.22 | MFQ, MFP | ic50 = 3 uM, ic50 = 3 uM | 511.414, 511.414 |
1H08 | 1.8 | HOMO SAPIENS | ENZYME 2.7.11.22 | GOL, BYP BWP | 92.094 | |
1H0V | 1.9 | HOMO SAPIENS | ENZYME 2.7.11.22 | UN4 | 248.241 | |
1H1P | 2.1 | HOMO SAPIENS | ENZYME 2.7.11.22 | CMG | Ki = 12 uM | 247.296 |
1H1Q | 2.5 | HOMO SAPIENS | ENZYME 2.7.11.22 | 2A6 | ic50 = 1 uM | 323.392 |
1H1R | 2 | HOMO SAPIENS | ENZYME 2.7.11.22 | 6CP | ic50 = 2.3 uM | 357.837 |
1H1S | 2 | HOMO SAPIENS | ENZYME 2.7.11.22 | 4SP | Ki = 6 nM | 402.471 |
1H24 | 2.5 | HOMO SAPIENS | ENZYME 2.7.11.22 | PRO VAL LYS ARG ARG LEU ASP LEU GLU | Kd = 0.5 uM | 1111.36 |
1HCK | 1.9 | HOMO SAPIENS | ENZYME 2.7.11.22 | MG, ATP | 24.305, 507.181 | |
1JSV | 1.96 | HOMO SAPIENS | ENZYME 2.7.11.22 | U55 | 265.292 | |
1JVP | 1.53 | HOMO SAPIENS | ENZYME 2.7.11.22 | LIG | ic50 = 1.6 uM | 233.268 |
1KE5 | 2.2 | HOMO SAPIENS | ENZYME 2.7.11.22 | LS1 | ic50 = 560 nM | 329.374 |
1KE6 | 2 | HOMO SAPIENS | ENZYME 2.7.11.22 | LS2 | ic50 = 5.7 nM | 401.463 |
1KE7 | 2 | HOMO SAPIENS | ENZYME 2.7.11.22 | LS3 | ic50 = 8.9 nM | 393.416 |
1KE8 | 2 | HOMO SAPIENS | ENZYME 2.7.11.22 | LS4 | ic50 = 1000 nM | 398.459 |
1KE9 | 2 | HOMO SAPIENS | ENZYME 2.7.11.22 | LS5 | ic50 = 660 nM | 357.387 |
1OI9 | 2.1 | HOMO SAPIENS | ENZYME 2.7.11.22 | MG, SGM, N20 | ic50 = 69 nM | 24.305, 108.159, 339.392 |
1OIQ | 2.31 | HOMO SAPIENS | ENZYME 2.7.11.22 | HDU | ic50 = 2.9 uM | 267.286 |
1OIR | 1.91 | HOMO SAPIENS | ENZYME 2.7.11.22 | HDY | ic50 = 0.032 uM | 418.492 |
1OIT | 1.6 | HOMO SAPIENS | ENZYME 2.7.11.22 | HDT | ic50 < 0.003 uM | 366.397 |
1OIU | 2 | HOMO SAPIENS | ENZYME 2.7.11.22 | SGM, N76, MG | ic50 = 0.21 uM | 108.159, 402.471, 24.305 |
1OIY | 2.4 | HOMO SAPIENS | ENZYME 2.7.11.22 | SGM, N41, MG | ic50 = 64 nM | 108.159, 366.417, 24.305 |
1OKV | 2.4 | HOMO SAPIENS | ENZYME 2.7.11.22 | ARG ARG LEU ILE PHE NH2 | ic50 = 0.68 uM | 706.938 |
1OKW | 2.5 | HOMO SAPIENS | ENZYME 2.7.11.22 | ACE ARG ARG LEU ASN FCL NH2 | ic50 = 5.6 uM | 782.348 |
1P2A | 2.5 | HOMO SAPIENS | ENZYME 2.7.11.22 | 5BN | ic50 = 12 nM | 310.326 |
1P5E | 2.22 | HOMO SAPIENS | ENZYME 2.7.11.22 | TBS | 434.708 | |
1PKD | 2.3 | HOMO SAPIENS | ENZYME 2.7.11.22 | UCN | 482.53 | |
1PXI | 1.95 | HOMO SAPIENS | ENZYME 2.7.11.22 | CK1 | 246.116 | |
1PXJ | 2.3 | HOMO SAPIENS | ENZYME 2.7.11.22 | CK2 | 206.267 | |
1PXL | 2.5 | HOMO SAPIENS | ENZYME 2.7.11.22 | CK4 | 350.361 | |
1PXN | 2.5 | HOMO SAPIENS | ENZYME 2.7.11.22 | CK6 | Ki = 0.07 uM | 313.378 |
1PXO | 1.96 | HOMO SAPIENS | ENZYME 2.7.11.22 | CK7 | Ki = 2 nM | 328.349 |
1PXP | 2.3 | HOMO SAPIENS | ENZYME 2.7.11.22 | CK8 | Ki = 0.22 uM | 325.431 |
1PYE | 2 | HOMO SAPIENS | ENZYME 2.7.11.22 | PM1 | Ki = 386 nM | 377.344 |