5F6V | 1.49 | HOMO SAPIENS | ENZYME 6.3.2.- | 5VL | ic50 = 5.8 mM | 186.207 |
5F6W | 1.7 | HOMO SAPIENS | ENZYME 6.3.2.- | 5VL | ic50 = 5.8 mM | 186.207 |
5F6U | 1.55 | HOMO SAPIENS | ENZYME 6.3.2.- | 5VK | ic50 = 3 mM | 286.322 |
5C0K | 2.2 | HOMO SAPIENS | ENZYME 6.3.2.- | ZN, 4WK, EDO | ic50 = 1200 uM | 65.409, 188.247, 62.068 |
5H1T | 1.95 | HOMO SAPIENS | ENZYME 6.3.2.- | DMS, 7FF, ZN | Kd = 0.16 mM | 78.133, 206.241, 65.409 |
5AXI | 2.5 | MUS MUSCULUS | ENZYME 6.3.2.- | ASP GLY PTR MET PRO, CA, CL | ic50 = 120 uM | 658.602, 40.078, 35.453 |
5C3K | 2.02 | HOMO SAPIENS | ENZYME 6.3.2.- | 4XF, ZN | ic50 = 110 uM | 181.215, 65.409 |
5H1U | 1.9 | HOMO SAPIENS | ENZYME 6.3.2.- | DMS, ZN, 6KT | Kd = 63 uM | 78.133, 65.409, 193.226 |
5H1V | 2 | HOMO SAPIENS | ENZYME 6.3.2.- | ZN, DMS, 7FU | Kd = 34 uM | 65.409, 78.133, 223.255 |
5TDD | 1.55 | HOMO SAPIENS | ENZYME 6.3.2.- | EDO, HIS ILE PHE SER, ZN | Kd = 34 uM | 62.068, 471.582, 65.409 |
4P0A | 2.3 | HOMO SAPIENS | ENZYME 6.3.2.- | THR GLU ASP ASN ASP ASP ASP LEU TYR GLY | Kd = 30.3 uM | |
4IGK | 1.75 | HOMO SAPIENS | ENZYME 6.3.2.- | GOL, ALA CYS SEP PRO GLN PHE GLY | Kd = 28.2 uM | 92.094, 771.766 |
4J74 | 1.2 | XENOPUS LAEVIS | ENZYME 6.3.2.- | SO4, I18 | Kd = 26 uM | 96.063, 305.202 |
4J7D | 1.25 | XENOPUS LAEVIS | ENZYME 6.3.2.- | I31, SO4 | Kd = 20 uM | 495.483, 96.063 |
3NY3 | 1.6 | HOMO SAPIENS | ENZYME 6.3.2.- | ZN, ARG ILE PHE SER | Ka = 51900 M^-1 | 65.409, 507.636 |
4J7E | 1.63 | XENOPUS LAEVIS | ENZYME 6.3.2.- | SO4, I29 | Kd = 14 uM | 96.063, 565.555 |
5TDC | 1.61 | HOMO SAPIENS | ENZYME 6.3.2.- | SO4, NMM ILE PHE SER, ZN | Kd = 12.88 uM | 96.063, 433.577, 65.409 |
4J47 | 1.35 | HOMO SAPIENS | ENZYME 6.3.2.- | SER VAL PRO ILE, ZN | Ki = 12.02 uM | 414.503, 65.409 |
4YAT | 2.18 | HOMO SAPIENS | ENZYME 6.3.2.- | ZN, 4A8 | ic50 = 9.3 uM | 65.409, 347.389 |
4YAB | 1.9 | HOMO SAPIENS | ENZYME 6.3.2.- | SO4, 4CN, ZN | ic50 = 8.5 uM | 96.063, 244.312, 65.409 |
3ZVY | 1.95 | HOMO SAPIENS | ENZYME 6.3.2.- | ZN, TRS, ALA ARG THR LYS GLN THR ALA ARG, CL | Kd = 7.9 uM | 65.409, 122.143, 589.719, 35.453 |
5C7D | 2.25 | HOMO SAPIENS | ENZYME 6.3.2.- | 4YF, ZN | ic50 = 7.7 uM | 295.788, 65.409 |
3SOW | 1.95 | HOMO SAPIENS | ENZYME 6.3.2.- | ZN, ALA ARG THR M3L GLN THR ALA ARG LYS | Kd = 7.3 uM | 65.409, 675.853 |
5C7C | 2.32 | HOMO SAPIENS | ENZYME 6.3.2.- | ZN, 4YC | ic50 = 5.5 uM | 65.409, 322.853 |
4J46 | 1.42 | HOMO SAPIENS | ENZYME 6.3.2.- | ALA VAL PRO ILE, ZN | Ki = 5.24 uM | 398.504, 65.409 |
4WVT | 1.96 | HOMO SAPIENS | ENZYME 6.3.2.- | ZN, MAA PHE PRO PHE PHE 3V7 | ic50 = 4.87 uM | 65.409, 794.91 |
4LWT | 1.6 | XENOPUS LAEVIS | ENZYME 6.3.2.- | SO4, 20Q | ic50 = 3.9 uM | 96.063, 417.328 |
4IFI | 2.2 | HOMO SAPIENS | ENZYME 6.3.2.- | ACT, ARG SEP PRO VAL PHE SER | Kd = 3.34 uM | 59.044, 755.767 |
4ZGK | 2 | HOMO SAPIENS | ENZYME 6.3.2.- | 4NX | Kd = 3.1 uM | 498.785 |
3SOU | 1.8 | HOMO SAPIENS | ENZYME 6.3.2.- | ZN, ALA ARG THR LYS GLN THR ALA ARG LYS | Kd = 2.5 uM | 65.409, 919.1 |
4YAD | 1.73 | HOMO SAPIENS | ENZYME 6.3.2.- | 4A7, CL, ZN, GOL | ic50 = 2.5 uM | 376.427, 35.453, 65.409, 92.094 |
4J48 | 2.1 | HOMO SAPIENS | ENZYME 6.3.2.- | GOL, SO4, ALA MET ARG VAL, ZN | Ki = 2.41 uM | 92.094, 96.063, 461.632, 65.409 |
4WVU | 2.02 | HOMO SAPIENS | ENZYME 6.3.2.- | MAA VAL 3V8 PHE HOX, ZN, SO4, GOL | ic50 = 1.97 uM | 729.839, 65.409, 96.063, 92.094 |
4J44 | 1.3 | HOMO SAPIENS | ENZYME 6.3.2.- | ALA ILE ALA VAL, ZN | Ki = 1.87 uM | 372.466, 65.409 |
4JV9 | 2.5 | HOMO SAPIENS | ENZYME 6.3.2.- | SO4, 1MO | ic50 = 1.8 uM | 96.063, 426.335 |
4J45 | 1.48 | HOMO SAPIENS | ENZYME 6.3.2.- | ALA THR ALA ALA, ZN | Ki = 1.7 uM | 332.357, 65.409 |
4YAX | 2.25 | HOMO SAPIENS | ENZYME 6.3.2.- | 4AE, SO4, ZN, GOL | ic50 = 1.5 uM | 439.484, 96.063, 65.409, 92.094 |
5TDB | 1.1 | HOMO SAPIENS | ENZYME 6.3.2.- | EDO, DA2 ILE PHE SER, ZN | Kd = 1.45 uM | 62.068, 300.427, 65.409 |
3JZK | 2.1 | HOMO SAPIENS | ENZYME 6.3.2.- | YIN | ic50 = 1.23 uM | 536.218 |
4MDQ | 2.12 | HOMO SAPIENS | ENZYME 6.3.2.- | 28W | Ki = 1.2 uM | 501.963 |
4JV7 | 2.2 | HOMO SAPIENS | ENZYME 6.3.2.- | SO4, 1MN | ic50 = 1 uM | 96.063, 515.237 |
5C84 | 2.36 | HOMO SAPIENS | ENZYME 6.3.2.- | ZN, 4YL | ic50 = 0.64 uM | 65.409, 367.894 |
4JWR | 2.35 | HOMO SAPIENS | ENZYME 6.3.2.- | 1MY | ic50 = 0.61 uM | 452.328 |
4MDN | 1.91 | HOMO SAPIENS | ENZYME 6.3.2.- | SO4, Y30 | Ki = 0.6 uM | 96.063, 582.474 |
4WVS | 2.09 | HOMO SAPIENS | ENZYME 6.3.2.- | GOL, MAA LPH PRO PHE 4LZ, ZN, SO4 | ic50 = 0.54 uM | 92.094, 674.759, 65.409, 96.063 |
4ZFI | 2 | HOMO SAPIENS | ENZYME 6.3.2.- | 4NJ | Kd = 0.5 uM | 511.827 |
4ZYC | 1.95 | HOMO SAPIENS | ENZYME 6.3.2.- | SO4, 4SS | ic50 = 0.38 uM | 96.063, 534.006 |
3V3L | 1.65 | HOMO SAPIENS | ENZYME 6.3.2.- | V3L | Kd ~ 370 nM | 559.316 |
3CM2 | 2.5 | HOMO SAPIENS | ENZYME 6.3.2.- | ZN, X23 | Ki = 340 nM | 65.409, 491.625 |
3TU1 | 1.6 | HOMO SAPIENS | ENZYME 6.3.2.- | 07G | Ki = 0.25 uM | 476.88 |