5F6V | 1.49 | HOMO SAPIENS | ENZYME 6.3.2.- | 5VL | ic50 = 5.8 mM | 186.207 |
5F6W | 1.7 | HOMO SAPIENS | ENZYME 6.3.2.- | 5VL | ic50 = 5.8 mM | 186.207 |
5F6U | 1.55 | HOMO SAPIENS | ENZYME 6.3.2.- | 5VK | ic50 = 3 mM | 286.322 |
5C0K | 2.2 | HOMO SAPIENS | ENZYME 6.3.2.- | EDO, ZN, 4WK | ic50 = 1200 uM | 62.068, 65.409, 188.247 |
5H1T | 1.95 | HOMO SAPIENS | ENZYME 6.3.2.- | ZN, DMS, 7FF | Kd = 0.16 mM | 65.409, 78.133, 206.241 |
5AXI | 2.5 | MUS MUSCULUS | ENZYME 6.3.2.- | ASP GLY PTR MET PRO, CA, CL | ic50 = 120 uM | 658.602, 40.078, 35.453 |
5C3K | 2.02 | HOMO SAPIENS | ENZYME 6.3.2.- | 4XF, ZN | ic50 = 110 uM | 181.215, 65.409 |
5H1U | 1.9 | HOMO SAPIENS | ENZYME 6.3.2.- | DMS, ZN, 6KT | Kd = 63 uM | 78.133, 65.409, 193.226 |
5H1V | 2 | HOMO SAPIENS | ENZYME 6.3.2.- | ZN, DMS, 7FU | Kd = 34 uM | 65.409, 78.133, 223.255 |
5TDD | 1.55 | HOMO SAPIENS | ENZYME 6.3.2.- | EDO, HIS ILE PHE SER, ZN | Kd = 34 uM | 62.068, 471.582, 65.409 |
4P0A | 2.3 | HOMO SAPIENS | ENZYME 6.3.2.- | THR GLU ASP ASN ASP ASP ASP LEU TYR GLY | Kd = 30.3 uM | |
4IGK | 1.75 | HOMO SAPIENS | ENZYME 6.3.2.- | GOL, ALA CYS SEP PRO GLN PHE GLY | Kd = 28.2 uM | 92.094, 771.766 |
4J74 | 1.2 | XENOPUS LAEVIS | ENZYME 6.3.2.- | SO4, I18 | Kd = 26 uM | 96.063, 305.202 |
4J7D | 1.25 | XENOPUS LAEVIS | ENZYME 6.3.2.- | I31, SO4 | Kd = 20 uM | 495.483, 96.063 |
3NY3 | 1.6 | HOMO SAPIENS | ENZYME 6.3.2.- | ZN, ARG ILE PHE SER | Ka = 51900 M^-1 | 65.409, 507.636 |
4J7E | 1.63 | XENOPUS LAEVIS | ENZYME 6.3.2.- | SO4, I29 | Kd = 14 uM | 96.063, 565.555 |
5TDC | 1.61 | HOMO SAPIENS | ENZYME 6.3.2.- | SO4, NMM ILE PHE SER, ZN | Kd = 12.88 uM | 96.063, 433.577, 65.409 |
4J47 | 1.35 | HOMO SAPIENS | ENZYME 6.3.2.- | SER VAL PRO ILE, ZN | Ki = 12.02 uM | 414.503, 65.409 |
4YAT | 2.18 | HOMO SAPIENS | ENZYME 6.3.2.- | ZN, 4A8 | ic50 = 9.3 uM | 65.409, 347.389 |
4YAB | 1.9 | HOMO SAPIENS | ENZYME 6.3.2.- | SO4, 4CN, ZN | ic50 = 8.5 uM | 96.063, 244.312, 65.409 |
3ZVY | 1.95 | HOMO SAPIENS | ENZYME 6.3.2.- | ZN, ALA ARG THR LYS GLN THR ALA ARG, TRS, CL | Kd = 7.9 uM | 65.409, 589.719, 122.143, 35.453 |
5C7D | 2.25 | HOMO SAPIENS | ENZYME 6.3.2.- | 4YF, ZN | ic50 = 7.7 uM | 295.788, 65.409 |
3SOW | 1.95 | HOMO SAPIENS | ENZYME 6.3.2.- | ZN, ALA ARG THR M3L GLN THR ALA ARG LYS | Kd = 7.3 uM | 65.409, 675.853 |
5C7C | 2.32 | HOMO SAPIENS | ENZYME 6.3.2.- | ZN, 4YC | ic50 = 5.5 uM | 65.409, 322.853 |
4J46 | 1.42 | HOMO SAPIENS | ENZYME 6.3.2.- | ALA VAL PRO ILE, ZN | Ki = 5.24 uM | 398.504, 65.409 |
4WVT | 1.96 | HOMO SAPIENS | ENZYME 6.3.2.- | ZN, MAA PHE PRO PHE PHE 3V7 | ic50 = 4.87 uM | 65.409, 794.91 |
4LWT | 1.6 | XENOPUS LAEVIS | ENZYME 6.3.2.- | SO4, 20Q | ic50 = 3.9 uM | 96.063, 417.328 |
4IFI | 2.2 | HOMO SAPIENS | ENZYME 6.3.2.- | ACT, ARG SEP PRO VAL PHE SER | Kd = 3.34 uM | 59.044, 755.767 |
4ZGK | 2 | HOMO SAPIENS | ENZYME 6.3.2.- | 4NX | Kd = 3.1 uM | 498.785 |
3SOU | 1.8 | HOMO SAPIENS | ENZYME 6.3.2.- | ZN, ALA ARG THR LYS GLN THR ALA ARG LYS | Kd = 2.5 uM | 65.409, 919.1 |
4YAD | 1.73 | HOMO SAPIENS | ENZYME 6.3.2.- | 4A7, CL, ZN, GOL | ic50 = 2.5 uM | 376.427, 35.453, 65.409, 92.094 |
4J48 | 2.1 | HOMO SAPIENS | ENZYME 6.3.2.- | GOL, SO4, ALA MET ARG VAL, ZN | Ki = 2.41 uM | 92.094, 96.063, 461.632, 65.409 |
4WVU | 2.02 | HOMO SAPIENS | ENZYME 6.3.2.- | MAA VAL 3V8 PHE HOX, ZN, SO4, GOL | ic50 = 1.97 uM | 729.839, 65.409, 96.063, 92.094 |
4J44 | 1.3 | HOMO SAPIENS | ENZYME 6.3.2.- | ALA ILE ALA VAL, ZN | Ki = 1.87 uM | 372.466, 65.409 |
4JV9 | 2.5 | HOMO SAPIENS | ENZYME 6.3.2.- | SO4, 1MO | ic50 = 1.8 uM | 96.063, 426.335 |
4J45 | 1.48 | HOMO SAPIENS | ENZYME 6.3.2.- | ALA THR ALA ALA, ZN | Ki = 1.7 uM | 332.357, 65.409 |
4YAX | 2.25 | HOMO SAPIENS | ENZYME 6.3.2.- | GOL, 4AE, SO4, ZN | ic50 = 1.5 uM | 92.094, 439.484, 96.063, 65.409 |
5TDB | 1.1 | HOMO SAPIENS | ENZYME 6.3.2.- | EDO, DA2 ILE PHE SER, ZN | Kd = 1.45 uM | 62.068, 300.427, 65.409 |
3JZK | 2.1 | HOMO SAPIENS | ENZYME 6.3.2.- | YIN | ic50 = 1.23 uM | 536.218 |
4MDQ | 2.12 | HOMO SAPIENS | ENZYME 6.3.2.- | 28W | Ki = 1.2 uM | 501.963 |
4JV7 | 2.2 | HOMO SAPIENS | ENZYME 6.3.2.- | SO4, 1MN | ic50 = 1 uM | 96.063, 515.237 |
5C84 | 2.36 | HOMO SAPIENS | ENZYME 6.3.2.- | ZN, 4YL | ic50 = 0.64 uM | 65.409, 367.894 |
4JWR | 2.35 | HOMO SAPIENS | ENZYME 6.3.2.- | 1MY | ic50 = 0.61 uM | 452.328 |
4MDN | 1.91 | HOMO SAPIENS | ENZYME 6.3.2.- | SO4, Y30 | Ki = 0.6 uM | 96.063, 582.474 |
4WVS | 2.09 | HOMO SAPIENS | ENZYME 6.3.2.- | GOL, MAA LPH PRO PHE 4LZ, ZN, SO4 | ic50 = 0.54 uM | 92.094, 674.759, 65.409, 96.063 |
4ZFI | 2 | HOMO SAPIENS | ENZYME 6.3.2.- | 4NJ | Kd = 0.5 uM | 511.827 |
4ZYC | 1.95 | HOMO SAPIENS | ENZYME 6.3.2.- | SO4, 4SS | ic50 = 0.38 uM | 96.063, 534.006 |
3V3L | 1.65 | HOMO SAPIENS | ENZYME 6.3.2.- | V3L | Kd ~ 370 nM | 559.316 |
3CM2 | 2.5 | HOMO SAPIENS | ENZYME 6.3.2.- | ZN, X23 | Ki = 340 nM | 65.409, 491.625 |
3TU1 | 1.6 | HOMO SAPIENS | ENZYME 6.3.2.- | 07G | Ki = 0.25 uM | 476.88 |
4JRG | 1.9 | XENOPUS LAEVIS | ENZYME 6.3.2.- | I09 | ic50 = 196 nM | 518.475 |
5C83 | 2.33 | HOMO SAPIENS | ENZYME 6.3.2.- | 4YN, ZN | ic50 = 0.16 uM | 423.571, 65.409 |
1RV1 | 2.3 | HOMO SAPIENS | ENZYME 6.3.2.- | IMZ | ic50 = 0.14 uM | 686.434 |
2AXI | 1.4 | HOMO SAPIENS | ENZYME 6.3.2.- | PRO PHE GLU 6CW LEU ASP TRP GLU PHE DPR, MPO, SO4 | ic50 = 140 nM | 1379.92, 209.263, 96.063 |
4YBM | 1.46 | HOMO SAPIENS | ENZYME 6.3.2.- | GOL, 4BJ, SO4, ZN | ic50 = 0.14 uM | 92.094, 575.632, 96.063, 65.409 |
4YBT | 1.82 | HOMO SAPIENS | ENZYME 6.3.2.- | DMS, ZN, 4BV | ic50 = 0.1 uM | 78.133, 65.409, 513.566 |
5OAI | 2 | HOMO SAPIENS | ENZYME 6.3.2.- | B5K | Ki = 0.1 uM | 495.879 |
5EPL | 1.81 | HOMO SAPIENS | ENZYME 6.3.2.- | UNX, 5R0 PHE ALA LEU ELY 5R5 | Kd = 0.094 uM | 796.043 |
4HG7 | 1.6 | HOMO SAPIENS | ENZYME 6.3.2.- | NUT, SO4 | ic50 = 90 nM | 581.49, 96.063 |
4J3E | 1.91 | XENOPUS LAEVIS | ENZYME 6.3.2.- | NUT, SO4 | ic50 = 0.088 uM | 581.49, 96.063 |
4JVE | 2.3 | HOMO SAPIENS | ENZYME 6.3.2.- | 1MQ | ic50 = 0.086 uM | 528.399 |
4JSC | 2.5 | XENOPUS LAEVIS | ENZYME 6.3.2.- | 1OY | ic50 = 74 nM | 554.456 |
3W69 | 1.9 | HOMO SAPIENS | ENZYME 6.3.2.- | LTZ, SO4 | ic50 = 0.058 uM | 696.729, 96.063 |
4YBS | 1.83 | HOMO SAPIENS | ENZYME 6.3.2.- | ZN, 4BK, DMS | ic50 = 0.057 uM | 65.409, 499.583, 78.133 |
5HMK | 2.17 | HOMO SAPIENS | ENZYME 6.3.2.- | 62Q | ic50 = 0.04 uM | 708.69 |
4QPL | 1.9 | MUS MUSCULUS | ENZYME 6.3.2.- | V3L, ZN | Kd = 39 nM | 559.316, 65.409 |
3LBL | 1.6 | HOMO SAPIENS | ENZYME 6.3.2.- | MI6 | Ki = 36 nM | 577.518 |
4DIJ | 1.9 | HOMO SAPIENS | ENZYME 6.3.2.- | BLF | ic50 = 0.03 uM | 574.5 |
4IPF | 1.7 | XENOPUS LAEVIS | ENZYME 6.3.2.- | SO4, 1F0 | ic50 = 18 nM | 96.063, 727.783 |
4KJV | 1.7 | HOMO SAPIENS | ENZYME 6.3.2.- | 1RK, ZN | ic50 = 0.018 uM | 547.599, 65.409 |
5HMI | 1.74 | HOMO SAPIENS | ENZYME 6.3.2.- | SO4, 62T | ic50 = 0.015 uM | 96.063, 714.718 |
4HBM | 1.9 | HOMO SAPIENS | ENZYME 6.3.2.- | 0Y7 | Kd = 12 nM | 450.355 |
4JVR | 1.7 | HOMO SAPIENS | ENZYME 6.3.2.- | 1MT | ic50 = 9.4 nM | 507.428 |
4OGV | 2.2 | HOMO SAPIENS | ENZYME 6.3.2.- | 2U7 | ic50 = 9 nM | 556.498 |
4OQ3 | 2.3 | HOMO SAPIENS | ENZYME 6.3.2.- | 2V8 | ic50 = 0.008 uM | 437.318 |
4ZYI | 1.67 | HOMO SAPIENS | ENZYME 6.3.2.- | CL, 4TH | ic50 = 0.008 uM | 35.453, 556.094 |
6Q9H | 2 | HOMO SAPIENS | ENZYME 6.3.2.- | HRH | ic50 = 7.8 nM | 418.292 |
4LWV | 2.32 | XENOPUS LAEVIS | ENZYME 6.3.2.- | SO4, 20W | ic50 = 7 nM | 96.063, 619.534 |
5HMH | 1.79 | HOMO SAPIENS | ENZYME 6.3.2.- | SO4, 62R | ic50 = 0.007 uM | 96.063, 756.755 |
4KJU | 1.6 | HOMO SAPIENS | ENZYME 6.3.2.- | 1RH, ZN | ic50 = 0.006 uM | 551.636, 65.409 |
2GV2 | 1.8 | HOMO SAPIENS | ENZYME 6.3.2.- | ACE PHE MET AIB PM3 6CW GLU 1AC LEU | ic50 = 5 nM | 1206.71 |
4LWU | 1.14 | XENOPUS LAEVIS | ENZYME 6.3.2.- | SO4, 20U | ic50 = 0.005 uM | 96.063, 583.481 |
4QO4 | 1.7 | HOMO SAPIENS | ENZYME 6.3.2.- | 35S | ic50 = 0.005 uM | 551.503 |
4ERE | 1.8 | HOMO SAPIENS | ENZYME 6.3.2.- | 0R2, SO4 | ic50 = 4.2 nM | 520.445, 96.063 |
2VSL | 2.1 | HOMO SAPIENS | ENZYME 6.3.2.- | ZN, MAA LYS PRO PHE, 15P | Ki = 4 nM | 65.409, 461.607, 1529.83 |
6Q9L | 1.13 | HOMO SAPIENS | ENZYME 6.3.2.- | HTZ, CL | ic50 = 3.9 nM | 659.648, 35.453 |
4LGE | 1.55 | HOMO SAPIENS | ENZYME 6.3.2.- | ZN, 1Y0 | ic50 = 3.5 nM | 65.409, 537.694 |
6Q9O | 1.21 | HOMO SAPIENS | ENZYME 6.3.2.- | HU8 | ic50 = 3.4 nM | 570.489 |
4HY4 | 1.25 | HOMO SAPIENS | ENZYME 6.3.2.- | 1BG, ZN | ic50 = 2.7 nM | 523.71, 65.409 |
4ZYF | 1.8 | HOMO SAPIENS | ENZYME 6.3.2.- | 4T4, CL | Kd = 2.3 nM | 659.257, 35.453 |
4LGU | 2 | HOMO SAPIENS | ENZYME 6.3.2.- | 1YH, ZN | ic50 = 2.1 nM | 525.683, 65.409 |
4OCC | 1.8 | HOMO SAPIENS | ENZYME 6.3.2.- | 2TZ | ic50 = 2 nM | 556.498 |
4MU7 | 1.79 | HOMO SAPIENS | ENZYME 6.3.2.- | ZN, 2DY | ic50 = 1.4 nM | 65.409, 587.752 |
4HY5 | 1.75 | HOMO SAPIENS | ENZYME 6.3.2.- | 1AQ, ZN | ic50 = 1.3 nM | 605.716, 65.409 |
4YC9 | 1.82 | HOMO SAPIENS | ENZYME 6.3.2.- | 4C1, GOL, ZN | Kd = 1.3 nM | 642.763, 92.094, 65.409 |
4MTI | 2.15 | HOMO SAPIENS | ENZYME 6.3.2.- | 2DX, ZN | ic50 = 1.2 nM | 539.709, 65.409 |
5TRF | 2.1 | HOMO SAPIENS | ENZYME 6.3.2.- | 7HC, SO4, GOL | Ki = 0.88 nM | 562.503, 96.063, 92.094 |
4ERF | 2 | HOMO SAPIENS | ENZYME 6.3.2.- | 0R3 | Kd = 0.4 nM | 478.408 |
4OBA | 1.6 | HOMO SAPIENS | ENZYME 6.3.2.- | 2TW | ic50 = 0.4 nM | 568.509 |
5LN2 | 1.58 | HOMO SAPIENS | ENZYME 6.3.2.- | 6ZT, SO4, CL | ic50 = 0.13 nM | 593.543, 96.063, 35.453 |