1
|
1YPE
|
Ki
=
8
nM |
UIP
|
C26 H30 N4 O3
|
CC[C@@H]1[....
|
2
|
1YPM
|
Ki
=
1.9
uM |
RA4
|
C23 H35 N7 O5
|
[H]/N=C(N)....
|
3
|
1YPJ
|
Ki
=
95
nM |
UIB
|
C26 H32 N4 O3
|
CC[C@@H]1[....
|
4
|
1YPG
|
Ki
=
10
nM |
UIR
|
C27 H30 N4 O3
|
c1cc(ccc1[....
|
5
|
1H8D
|
- |
PHW
|
C45 H48 N3 O9 P
|
CO/C=C/C[C....
|
6
|
1H8I
|
- |
ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU
|
n/a
|
n/a
|
7
|
1YPL
|
Ki
=
10.6
uM |
RA8
|
C23 H38 N6 O4 S
|
[H]/N=C(/N....
|
8
|
3U8T
|
Ki
=
16.5
uM |
DPN PRO DAR CYS NH2
|
n/a
|
n/a
|
9
|
1EB1
|
Ki
=
37
pM |
ZAL PRO MMO
|
n/a
|
n/a
|
10
|
1YPK
|
- |
CCR
|
C29 H39 N5 O7 S
|
Cc1cc(c(c(....
|
11
|
1SB1
|
Ki
=
128
nM |
165
|
C28 H35 N5 O4 S2
|
c1ccc(cc1)....
|
12
|
4LOY
|
- |
ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU
|
n/a
|
n/a
|
13
|
4HFP
|
Kd
=
42
nM |
15U
|
C23 H36 N6 O5 S
|
[H]/N=C(N)....
|
14
|
1TWX
|
- |
ASP PHE GLU GLU ILE PRO GLY GLU TYS LEU
|
n/a
|
n/a
|
15
|
1VR1
|
- |
ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU
|
n/a
|
n/a
|
16
|
3BV9
|
Ki
=
4.4
uM |
DAR OIC PRO DAL 4PH NH2
|
n/a
|
n/a
|
17
|
3U8R
|
Ki
=
7.7
uM |
DPN PRO DAR ILE NH2
|
n/a
|
n/a
|
18
|
3U8O
|
Ki
=
0.92
uM |
DPN PRO DAR DTH NH2
|
n/a
|
n/a
|
19
|
1UVT
|
Ki
=
0.023
uM |
I48
|
C20 H22 N3 O3 S
|
Cc1cc(cc(c....
|
20
|
1ETT
|
Ki
=
1.3
uM |
4QQ
|
C22 H28 N4 O3 S
|
[H]/N=C(c1....
|
21
|
1ETR
|
- |
MIT
|
C23 H37 N6 O5 S
|
C[C@@H]1CC....
|
22
|
1ETS
|
Ki
=
6
nM |
MID
|
C27 H31 N5 O4 S
|
[H]/N=C(/c....
|
23
|
1HXF
|
- |
ASP PHE GLU GLU ILE PRO GLY GLU TYR LEU
|
n/a
|
n/a
|
24
|
1C5N
|
Ki
=
20
uM |
ESI
|
C9 H8 I N2 S
|
c1cc2c(cc(....
|
25
|
2JH0
|
Ki
=
2
nM |
701
|
C18 H24 Cl N3 O5 S2
|
C[C@@H](C(....
|
26
|
1WBG
|
ic50
=
1
mM |
L03
|
C9 H8 Cl N3 S
|
CSc1[nH]c(....
|
27
|
1AFE
|
- |
ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU
|
n/a
|
n/a
|
28
|
3DA9
|
Kd
=
3.1
uM |
44U
|
C23 H29 N3 O2
|
CCCNC(=O)[....
|
29
|
2UUJ
|
- |
ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU
|
n/a
|
n/a
|
30
|
1QHR
|
- |
ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU
|
n/a
|
n/a
|
31
|
1QJ1
|
ic50
=
9
nM |
ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU
|
n/a
|
n/a
|
32
|
1AE8
|
- |
AZL
|
C21 H33 N5 O4
|
CCOC(=O)N[....
|
33
|
1C5L
|
- |
ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU
|
n/a
|
n/a
|
34
|
4BAO
|
Ki
=
4.29
nM |
MVF
|
C22 H32 N6 O3
|
[H]/N=C(/c....
|
35
|
2JH5
|
Ki
=
367
nM |
895
|
C17 H22 Cl N3 O5 S2
|
C[C@@H](C(....
|
36
|
1HXE
|
- |
ASP PHE GLU GLU ILE PRO GLY GLU TYR LEU
|
n/a
|
n/a
|
37
|
1QJ6
|
ic50
=
18
nM |
ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU
|
n/a
|
n/a
|
38
|
1AWF
|
Ki
=
0.97
uM |
ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU
|
n/a
|
n/a
|
39
|
2GDE
|
ic50
=
5.7
nM |
SN3
|
C26 H43 Cl N6 O10 S
|
[H]/N=C(N)....
|
40
|
8KME
|
Ki
=
8
uM |
ACE 0BN CHG MLY LEU PRO NH2
|
n/a
|
n/a
|
41
|
1NY2
|
- |
ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU
|
n/a
|
n/a
|
42
|
2H9T
|
- |
SVR
|
C51 H40 N6 O23 S6
|
Cc1ccc(cc1....
|
43
|
1QJ7
|
ic50
=
18
nM |
ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU
|
n/a
|
n/a
|
44
|
1UMA
|
- |
IN2
|
C8 H18 N4 O3
|
CN(C)C(=O)....
|
45
|
2UUK
|
- |
ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU
|
n/a
|
n/a
|
46
|
1AD8
|
Ki
=
247
nM |
ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU
|
n/a
|
n/a
|
47
|
2UUF
|
- |
ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU
|
n/a
|
n/a
|
48
|
1XMN
|
- |
SGN IDS SGN IDS SGN
|
n/a
|
n/a
|
49
|
2JH6
|
Ki
=
17
nM |
894
|
C17 H24 Cl N3 O5 S2
|
C[C@@H](C(....
|
50
|
2ANM
|
ic50
=
1.8
nM |
CDO
|
C23 H32 N6 O4
|
[H]/N=C(/c....
|
51
|
1HAH
|
- |
ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU
|
n/a
|
n/a
|
52
|
3BF6
|
ic50
=
40
uM |
SVR
|
C51 H40 N6 O23 S6
|
Cc1ccc(cc1....
|
53
|
1WAY
|
ic50
=
400
uM |
L02
|
C14 H16 Cl N3
|
c1cc(ccc1c....
|
54
|
7KME
|
Ki
=
40
uM |
ASP PHE GLU GLU ILE PRO GLU GLU TYS LEU
|
n/a
|
n/a
|
55
|
3PMA
|
- |
GU4 YYJ
|
n/a
|
n/a
|
56
|
3BEF
|
- |
ASN ASP LYS TYR GLU PRO PHE TRP GLU
|
n/a
|
n/a
|