1
|
3HNT
|
- |
AXR BXY BXY BXX
|
n/a
|
n/a
|
2
|
3HNV
|
- |
AXR BXY BXY BXX
|
n/a
|
n/a
|
3
|
3HNS
|
- |
AXR BXY BXY BXY BXX BXX
|
n/a
|
n/a
|
4
|
6N16
|
- |
ALA VAL GLY ILE GLY ALA VAL PHE
|
n/a
|
n/a
|
5
|
6MQR
|
- |
ALA VAL GLY ILE GLY ALA VAL PHE
|
n/a
|
n/a
|
6
|
3QG6
|
ic50
=
0.73
nM |
TYR SER THR CYS TYR PHE ILE MET
|
n/a
|
n/a
|
7
|
3IF1
|
- |
NGA
|
C8 H15 N O6
|
CC(=O)N[C@....
|
8
|
3IET
|
Kd
=
0.14
uM |
GLY THR LYS PRO PRO LEU GLU GLU LEU A2G
|
n/a
|
n/a
|
9
|
3PHQ
|
- |
KDO
|
C8 H14 O8
|
C1[C@H]([C....
|
10
|
2HRP
|
- |
MET SER LEU PRO GLY ARG TRP LYS PRO LYS
|
n/a
|
n/a
|
11
|
5NBW
|
- |
8SK
|
C20 H12 O
|
c1ccc2c(c1....
|
12
|
6MSY
|
- |
MAN MAN MAN MAN
|
n/a
|
n/a
|
13
|
3OAU
|
- |
MAN MAN
|
n/a
|
n/a
|
14
|
6N35
|
- |
MAN
|
C6 H12 O6
|
C([C@@H]1[....
|
15
|
6MUB
|
- |
BMA MAN MAN MAN MAN
|
n/a
|
n/a
|
16
|
6MU3
|
- |
BMA MAN MAN MAN
|
n/a
|
n/a
|
17
|
3OAZ
|
- |
2M5
|
C8 H16 O6
|
C[C@@H]([C....
|
18
|
4RBP
|
- |
KDO MAN MAN MAN MAN MAN
|
n/a
|
n/a
|
19
|
3OAY
|
- |
BDF
|
C6 H12 O6
|
C1[C@H]([C....
|
20
|
4OJF
|
- |
ASP ALA GLU PHE ARG HIS ASP SER
|
n/a
|
n/a
|
21
|
5D6C
|
- |
57S
|
C13 H26 N O13 P
|
CC(=O)N[C@....
|
22
|
6DWA
|
- |
HD4
|
C13 H26 N O13 P
|
CC(=O)N[C@....
|
23
|
2BMK
|
Kd
=
2.4
uM |
PDD
|
C11 H17 N2 O7 P
|
Cc1c(c(c(c....
|
24
|
1WC7
|
- |
PP3
|
C11 H17 N2 O7 P
|
Cc1c(c(c(c....
|
25
|
1WCB
|
Kd
=
26
nM |
PE1
|
C14 H24 N3 O7 P
|
Cc1c(c(c(c....
|
26
|
1MJ7
|
Kd
=
4.5
nM |
HAL
|
C23 H29 N2 O7 P
|
c1ccc(cc1)....
|
27
|
1MH5
|
Kd
=
0.61
nM |
HAL
|
C23 H29 N2 O7 P
|
c1ccc(cc1)....
|
28
|
1MFA
|
Kd
=
9.1
uM |
MMA GLA ABE
|
n/a
|
n/a
|
29
|
3I9G
|
Kd
=
1.1
nM |
S1P
|
C18 H38 N O5 P
|
CCCCCCCCCC....
|
30
|
1F4X
|
Kd
=
2.6
uM |
MGS
|
C12 H23 N O7
|
C[C@@H]1[C....
|
31
|
1AJ7
|
Kd
=
135
uM |
NPE
|
C11 H13 N O7 P
|
c1cc(ccc1[....
|
32
|
1GAF
|
Kd
=
10
nM |
NPE
|
C11 H13 N O7 P
|
c1cc(ccc1[....
|
33
|
3CFD
|
- |
SPB
|
C19 H19 N O3
|
c1ccc(cc1)....
|
34
|
4JN2
|
- |
4CC
|
C25 H25 N7 O3
|
[H]/N=C(c1....
|
35
|
1U8M
|
- |
GLU LEU ASP LYS TYR ALA SER
|
n/a
|
n/a
|
36
|
3IDG
|
- |
ALA LEU ASP LYS TRP ASP
|
n/a
|
n/a
|
37
|
1TJG
|
- |
GLU LEU ASP LYS TRP ALA SER
|
n/a
|
n/a
|
38
|
1U93
|
- |
GLU GLN ASP LYS TRP ALA SER
|
n/a
|
n/a
|
39
|
1U8H
|
- |
ALA LEU ASP LYS TRP ALA SER
|
n/a
|
n/a
|
40
|
1U8Q
|
- |
GLU LEU GLU LYS TRP ALA SER
|
n/a
|
n/a
|
41
|
3IDJ
|
- |
GLU LEU ASP ORN TRP ALA SER
|
n/a
|
n/a
|
42
|
2F5B
|
- |
GLU LEU ASP LYS TRP ALA SER
|
n/a
|
n/a
|
43
|
1U92
|
- |
GLU ALA ASP LYS TRP GLN SER
|
n/a
|
n/a
|
44
|
1U8I
|
- |
GLU LEU ASP LYS TRP ALA ASN
|
n/a
|
n/a
|
45
|
1U95
|
- |
GLU LEU ASP HIS TRP ALA SER
|
n/a
|
n/a
|
46
|
1U8J
|
- |
GLU LEU ASP LYS TRP ALA GLY
|
n/a
|
n/a
|
47
|
3IDI
|
- |
ALA LEU ASP LYS TRP GLN ASN
|
n/a
|
n/a
|
48
|
3IDN
|
- |
GLU LEU ASP HOX TRP ALA SER
|
n/a
|
n/a
|
49
|
1U91
|
- |
GLU ASN ASP LYS TRP ALA SER
|
n/a
|
n/a
|
50
|
3IDM
|
- |
GLU LEU ASP NRG TRP ALA SER
|
n/a
|
n/a
|
51
|
1U8K
|
- |
LEU GLU LEU ASP LYS TRP ALA SER LEU
|
n/a
|
n/a
|
52
|
2C1P
|
- |
FNZ
|
C18 H15 F N4 O
|
c1cc(ccc1C....
|
53
|
2R2E
|
- |
KDE
|
C11 H18 O8
|
C=CCO[C@@]....
|
54
|
3SY0
|
- |
KDA KDO KDO
|
n/a
|
n/a
|
55
|
3OKL
|
- |
KDA KDO
|
n/a
|
n/a
|
56
|
2R1Y
|
Kd
=
31
uM |
KDR KDO
|
n/a
|
n/a
|
57
|
2R2B
|
- |
KDA KDO KDO
|
n/a
|
n/a
|
58
|
2G5B
|
- |
PRO THR SER SER GLU GLN ILE
|
n/a
|
n/a
|
59
|
2R1X
|
Kd
=
16
uM |
KDA KDD
|
n/a
|
n/a
|
60
|
3OKK
|
- |
KDA KDO
|
n/a
|
n/a
|
61
|
3OKE
|
- |
KO2
|
C11 H18 O9
|
C=CCO[C@@]....
|
62
|
3OKN
|
- |
KDA KDO KDO
|
n/a
|
n/a
|
63
|
3HZM
|
Kd
=
0.000000064
M |
KDO
|
C8 H14 O8
|
C1[C@H]([C....
|
64
|
2R23
|
Kd
=
190
uM |
KDA KO1
|
n/a
|
n/a
|
65
|
1Q9W
|
- |
GP1 GP4 KDO KDO KDO
|
n/a
|
n/a
|
66
|
3T65
|
- |
KDA KDO
|
n/a
|
n/a
|
67
|
2R1W
|
Kd
=
25
uM |
KDA KDB
|
n/a
|
n/a
|
68
|
3OKO
|
- |
KDA KDO KDO
|
n/a
|
n/a
|
69
|
3HZV
|
- |
KDA KDO KDO
|
n/a
|
n/a
|
70
|
3T4Y
|
- |
KDO
|
C8 H14 O8
|
C1[C@H]([C....
|
71
|
3OKD
|
- |
KDO
|
C8 H14 O8
|
C1[C@H]([C....
|
72
|
3T77
|
- |
KDA KDO
|
n/a
|
n/a
|
73
|
3HZY
|
Kd
=
0.000000064
M |
KDA KDO KDO
|
n/a
|
n/a
|
74
|
3HZK
|
Kd
=
0.3
M |
KDA KDO
|
n/a
|
n/a
|
75
|
2R2H
|
- |
KO2
|
C11 H18 O9
|
C=CCO[C@@]....
|
76
|
3BPC
|
Kd
=
16
uM |
KDA KDB
|
n/a
|
n/a
|
77
|
4HGW
|
Kd
=
0.000000064
M |
KTU KDO
|
n/a
|
n/a
|
78
|
5XQW
|
Kd
=
1.6
nM |
8EU
|
C9 H12 N O5 P
|
CCP(=O)(O)....
|
79
|
5TKJ
|
- |
ALA VAL GLY ILE GLY ALA VAL PHE
|
n/a
|
n/a
|
80
|
6CDP
|
- |
ALA VAL GLY ILE GLY ALA VAL PHE
|
n/a
|
n/a
|
81
|
6CDM
|
- |
ALA VAL GLY ILE GLY ALA VAL PHE
|
n/a
|
n/a
|
82
|
1Y0L
|
Kd
~
1
nM |
HAN
|
C14 H19 N3 O2
|
Cc1cc2c(cc....
|
83
|
1E4W
|
Kd
=
25
nM |
SER HIS PHE ASN GLU TYR GLU
|
n/a
|
n/a
|
84
|
3V52
|
- |
GLU PRO GLN ALA PRO TRP MET GLU
|
n/a
|
n/a
|
85
|
3UYR
|
- |
GLU PRO GLN ALA PRO TRP MET GLU
|
n/a
|
n/a
|
86
|
3V4U
|
- |
GLU PRO GLN ALA PRO TRP MET GLU GLN
|
n/a
|
n/a
|
87
|
3UO1
|
- |
GLU PRO GLN ALA PRO TRP MET GLU GLN
|
n/a
|
n/a
|
88
|
1F3D
|
- |
TPM
|
C12 H18 N3
|
c1cc(ccc1C....
|
89
|
2OK0
|
Kd
=
0.2
nM |
DT DC
|
n/a
|
n/a
|
90
|
1MRF
|
- |
DI
|
C10 H13 N4 O7 P
|
c1nc2c(n1[....
|
91
|
1MRD
|
- |
IDP
|
C10 H14 N4 O11 P2
|
c1nc2c(n1[....
|
92
|
1MRE
|
- |
GDP
|
C10 H15 N5 O11 P2
|
c1nc2c(n1[....
|
93
|
6UG7
|
- |
BGC GAL GLA NGA GAL SIA
|
n/a
|
n/a
|
94
|
6UG8
|
- |
BGC GAL GLA NGA GAL SIA
|
n/a
|
n/a
|
95
|
5MY4
|
- |
PCA PHE ARG HIS ASP SER GLY TYR GLU VAL
|
n/a
|
n/a
|
96
|
3FO0
|
- |
BZH
|
C12 H14 N4 O3
|
c1cc2c(cc1....
|
97
|
3FO2
|
- |
BZH
|
C12 H14 N4 O3
|
c1cc2c(cc1....
|
98
|
3FO1
|
- |
BZH
|
C12 H14 N4 O3
|
c1cc2c(cc1....
|
99
|
5DTF
|
- |
5CT
|
C10 H23 N3 O3
|
C(CCNC[C@H....
|
100
|
5MYO
|
- |
PCA PHE ARG HIS ASP SER GLY TYR GLU VAL
|
n/a
|
n/a
|
101
|
1QYG
|
- |
BCG
|
C16 H19 N O4
|
C[N@]1[C@H....
|
102
|
1RIV
|
- |
OBE
|
C16 H19 N O5
|
C[N@H+]1[C....
|
103
|
1Q72
|
Kd
=
0.0000123
M |
COC
|
C17 H21 N O4
|
C[N@]1[C@H....
|
104
|
1RIU
|
- |
RBE
|
C15 H17 N O4
|
c1ccc(cc1)....
|
105
|
6OBD
|
- |
ASN ASP THR SER GLN THR SER SER PRO SER OPE
|
n/a
|
n/a
|
106
|
3FN0
|
Kd
~
40
uM |
TRP ASN TRP PHE ASP ILE THR ASN LYS
|
n/a
|
n/a
|
107
|
1S3K
|
Kd
=
0.24
uM |
NDG FUC GAL FUC
|
n/a
|
n/a
|
108
|
3EYV
|
- |
NDG FUC GAL FUC
|
n/a
|
n/a
|
109
|
5I8C
|
- |
ALA VAL GLY ILE GLY ALA VAL PHE LEU
|
n/a
|
n/a
|
110
|
6UCE
|
- |
ALA VAL GLY ILE GLY ALA VAL PHE
|
n/a
|
n/a
|
111
|
6UCF
|
- |
ALA VAL GLY ILE GLY ALA VAL PHE
|
n/a
|
n/a
|
112
|
2AJX
|
- |
TGN
|
C16 H22 N O5 P
|
C[N@]1[C@H....
|
113
|
2AJZ
|
- |
ECG
|
C10 H17 N O3
|
C[N@]1[C@H....
|
114
|
2AK1
|
- |
BEZ
|
C7 H6 O2
|
c1ccc(cc1)....
|
115
|
2AJV
|
- |
COC
|
C17 H21 N O4
|
C[N@]1[C@H....
|
116
|
2AJY
|
- |
ECG
|
C10 H17 N O3
|
C[N@]1[C@H....
|
117
|
5VH4
|
- |
NAD
|
C21 H27 N7 O14 P2
|
c1cc(c[n+]....
|
118
|
1A4K
|
Kd
=
0.01
uM |
FRA
|
C21 H23 N3 O7
|
CC(=O)Nc1c....
|
119
|
6DZN
|
- |
AE3
|
C6 H14 O3
|
CCOCCOCCO
|
120
|
3IJH
|
Kd
=
100
uM |
KO2
|
C11 H18 O9
|
C=CCO[C@@]....
|
121
|
1YEE
|
- |
PNB
|
C13 H17 N2 O8 P
|
c1cc(ccc1C....
|
122
|
1KN4
|
- |
PDE
|
C13 H17 N2 O8 P
|
C[C@@H](C(....
|
123
|
1YEG
|
- |
BPN
|
C7 H7 N O3
|
c1cc(ccc1C....
|
124
|
1YEK
|
- |
NPO
|
C6 H5 N O3
|
c1cc(ccc1[....
|
125
|
1YEI
|
Kd
=
35
nM |
PGG
|
C12 H15 N2 O8 P
|
c1cc(ccc1[....
|
126
|
1YEC
|
- |
PNB
|
C13 H17 N2 O8 P
|
c1cc(ccc1C....
|
127
|
1YEJ
|
Kd
=
35
nM |
PNF
|
C16 H23 N2 O8 P
|
c1cc(ccc1[....
|
128
|
1YEF
|
- |
PNC
|
C14 H17 N3 O6
|
c1cc(ccc1C....
|
129
|
1KN2
|
- |
PNE
|
C13 H17 N2 O8 P
|
CC(C(=O)O)....
|
130
|
4OCX
|
Kd
~
3.6
pM |
MT1
|
C20 H23 N8 O5
|
CN(Cc1cnc2....
|
131
|
4S1D
|
- |
41M
|
C16 H29 N5 O3 S
|
C1[C@H]2[C....
|
132
|
1FLR
|
Kd
=
0.1
nM |
FLU
|
C20 H12 O5
|
c1ccc(c(c1....
|
133
|
5EOR
|
- |
ASP VAL GLN THR GLY ARG ARG PRO TYR GLU
|
n/a
|
n/a
|
134
|
5JOP
|
- |
NAG GAL BGC GAL
|
n/a
|
n/a
|
135
|
3QCU
|
- |
NKN
|
C17 H35 O7 P
|
CCCCCCCCCC....
|
136
|
4ONF
|
- |
ASP ALA GLU PHE ARG HIS ASP
|
n/a
|
n/a
|
137
|
1KEL
|
Kd
=
52
nM |
AAH
|
C13 H19 N2 O7 P
|
c1cc(ccc1C....
|
138
|
1JGU
|
- |
HBC
|
C20 H21 N O
|
c1ccc(cc1)....
|
139
|
2DDQ
|
- |
HRB
|
C17 H27 N3 O5
|
CCCCC[C@@H....
|
140
|
2DQU
|
Ki
=
50
nM |
CPD
|
C28 H36 Cl2 F3 N6 O8 P
|
CCNC(=O)N(....
|
141
|
2DQT
|
Ki
=
50
nM |
CPD
|
C28 H36 Cl2 F3 N6 O8 P
|
CCNC(=O)N(....
|
142
|
6MQC
|
- |
ALA VAL GLY ILE GLY ALA VAL PHE
|
n/a
|
n/a
|
143
|
1JGL
|
Kd
=
2
nM |
EST
|
C18 H24 O2
|
C[C@]12CC[....
|
144
|
1A0Q
|
Ki
=
27
nM |
HEP
|
C15 H22 N O6 P
|
CCCC[C@H](....
|
145
|
2Z93
|
Kd
=
11.1
nM |
END
|
C17 H24 O7
|
C1C=CCO[C@....
|
146
|
2Z92
|
Kd
=
0.8
nM |
ENE
|
C22 H30 O8
|
C1C=CCO[C@....
|
147
|
2R0W
|
- |
ASP ALA GLU PHE ARG HIS ASP SER
|
n/a
|
n/a
|
148
|
5EOQ
|
- |
LYS ARG GLU ALA ILE VAL LYS ALA ASP GLU
|
n/a
|
n/a
|
149
|
3EYS
|
Kd
=
3000
nM |
PCA PHE ARG HIS ASP SER
|
n/a
|
n/a
|
150
|
2IPU
|
- |
ASP ALA GLU PHE ARG HIS ASP SER
|
n/a
|
n/a
|
151
|
2R0Z
|
Kd
=
3400
nM |
ALA LYS PHE ARG HIS ASP
|
n/a
|
n/a
|
152
|
6EV2
|
- |
BGC
|
C6 H12 O6
|
C([C@@H]1[....
|
153
|
4YHY
|
- |
M3L
|
C9 H21 N2 O2
|
C[N+](C)(C....
|
154
|
3TV3
|
- |
MAN AML MAN MAN MAN MAN MAN MAN MAN
|
n/a
|
n/a
|
155
|
3TWC
|
- |
MAN AML MAN MAN MAN MAN MAN MAN MAN
|
n/a
|
n/a
|
156
|
6B3D
|
- |
MAN MAN MAN MAN MAN MAN MAN
|
n/a
|
n/a
|
157
|
2V17
|
- |
THR ASP HIS GLY ALA GLU
|
n/a
|
n/a
|
158
|
1EAP
|
- |
HEP
|
C15 H22 N O6 P
|
CCCC[C@H](....
|
159
|
6C5J
|
Kd
=
68.5
nM |
GP1 Z9M KDO KDO KDO
|
n/a
|
n/a
|
160
|
4M7J
|
Kd
=
0.781
uM |
KDA KDO KDO
|
n/a
|
n/a
|
161
|
6C5H
|
Kd
=
370
nM |
GP1 Z9M KDO KDO KDO
|
n/a
|
n/a
|
162
|
5T78
|
Kd
=
43
nM |
NGA ALA PRO ASP THR ARG PRO ALA PRO
|
n/a
|
n/a
|
163
|
5T6P
|
Kd
=
880
nM |
ALA PRO ASP THR ARG PRO ALA PRO
|
n/a
|
n/a
|
164
|
4TUO
|
- |
GLC GAL SIA NGA SIA
|
n/a
|
n/a
|
165
|
1DL7
|
Kd
=
0.32
uM |
NCH
|
C11 H18 N2 O6 P
|
C[N+](C)(C....
|
166
|
2HKF
|
- |
LEU PRO GLY GLU GLU ASP LEU PRO GLY
|
n/a
|
n/a
|
167
|
1MFE
|
- |
MAN GLA ABE
|
n/a
|
n/a
|
168
|
1MFB
|
- |
RAM MAN GLA ABE RAM MAN GLA
|
n/a
|
n/a
|
169
|
1MFD
|
Kd
=
4.9
uM |
MMA GLA ABE
|
n/a
|
n/a
|
170
|
1MFC
|
- |
RAM MAN GLA ABE
|
n/a
|
n/a
|
171
|
1LO3
|
- |
AN1
|
C18 H16 O2
|
Cc1c2ccccc....
|
172
|
1LO0
|
- |
BC1
|
C19 H17 N3 O3
|
CN1c2ccccc....
|
173
|
1LO2
|
- |
OX1
|
C18 H16 O4
|
CC12c3cccc....
|
174
|
3BZ4
|
- |
EAG RAM RAM GLC RAM NAG RAM RAM GLC RAM
|
n/a
|
n/a
|
175
|
3C6S
|
- |
RAM NAG RAM RAM RAM NAG RAM RAM RAM GLC GLC
|
n/a
|
n/a
|
176
|
6DWI
|
- |
HD4
|
C13 H26 N O13 P
|
CC(=O)N[C@....
|
177
|
6UBI
|
- |
ALA VAL GLY ILE GLY ALA VAL PHE
|
n/a
|
n/a
|
178
|
1M7D
|
Ka
=
1700000
M^-1 |
MAG RAE RAM
|
n/a
|
n/a
|
179
|
1M7I
|
Ka
=
250000
M^-1 |
RAO NAG RAM RAM RAM
|
n/a
|
n/a
|
180
|
1PZ5
|
Kd
=
4
uM |
MET ASP TRP ASN MET HIS ALA ALA
|
n/a
|
n/a
|
181
|
5TKK
|
- |
ALA VAL GLY ILE GLY ALA VAL PHE
|
n/a
|
n/a
|
182
|
2BJM
|
Ka
<
100000
M^-1 |
ANF
|
C14 H10 O
|
c1ccc2c(c1....
|
183
|
1A6V
|
- |
NPC
|
C14 H17 N2 O6
|
c1cc(c(cc1....
|
184
|
1OAU
|
Kd
=
20
nM |
DNF SER
|
n/a
|
n/a
|
185
|
1A6W
|
- |
NIP
|
C14 H16 I N2 O6
|
c1c(cc(c(c....
|
186
|
1XF2
|
- |
DT DT DT
|
n/a
|
n/a
|
187
|
2OMN
|
- |
IPH
|
C6 H6 O
|
c1ccc(cc1)....
|
188
|
2YKL
|
- |
NLD
|
C17 H25 N3 O3
|
CCNC(=O)CC....
|
189
|
2YK1
|
Kd
=
7.4
nM |
NCT
|
C10 H14 N2
|
C[N@@]1CCC....
|
190
|
6MQE
|
- |
ALA VAL GLY ILE GLY ALA VAL PHE
|
n/a
|
n/a
|
191
|
6DF1
|
- |
LEU PTR LEU
|
n/a
|
n/a
|
192
|
6DZR
|
- |
FLC
|
C6 H5 O7
|
C(C(=O)[O-....
|
193
|
5ALB
|
- |
TIQ
|
C23 H28 F2 N6 O4 S
|
CCCSc1nc(c....
|
194
|
5ALC
|
- |
TIQ
|
C23 H28 F2 N6 O4 S
|
CCCSc1nc(c....
|
195
|
1NGP
|
- |
NPA
|
C8 H7 N O5
|
c1cc(c(cc1....
|
196
|
4ODV
|
- |
GP1 Z9M
|
n/a
|
n/a
|
197
|
1KEG
|
- |
DT 64T DT DT
|
n/a
|
n/a
|
198
|
1EHL
|
- |
5HT DT
|
n/a
|
n/a
|
199
|
1C1E
|
- |
ENH
|
C10 H5 Cl6 N O2
|
CN1C(=O)[C....
|
200
|
1CLY
|
- |
NAG NON FUC GAL FUC
|
n/a
|
n/a
|
201
|
1CT8
|
Kd
=
0.3
uM |
TAA
|
C20 H21 Cl2 F3 N3 O8 P
|
c1cc(ccc1C....
|
202
|
1CE1
|
- |
GLY THR SER SER PRO SER ALA ASP
|
n/a
|
n/a
|
203
|
6DW2
|
- |
HD4
|
C13 H26 N O13 P
|
CC(=O)N[C@....
|
204
|
1T66
|
- |
FLU
|
C20 H12 O5
|
c1ccc(c(c1....
|
205
|
3GHB
|
- |
LYS GLY VAL ARG ILE GLY PRO GLY GLN ALA
|
n/a
|
n/a
|
206
|
2W65
|
- |
ALA CIR GLY LEU THR GLY ARG HYP GLY
|
n/a
|
n/a
|
207
|
5DYO
|
- |
FLU
|
C20 H12 O5
|
c1ccc(c(c1....
|
208
|
4UIN
|
Kd
=
24
nM |
QI9
|
C20 H24 N2 O2
|
COc1ccc2c(....
|
209
|
3V0W
|
Kd
=
32
nM |
KDO KDO GM0 GM0 GLC GMH GLC GLA GLC PA1
|
n/a
|
n/a
|
210
|
3IFL
|
- |
ASP ALA GLU PHE ARG HIS ASP
|
n/a
|
n/a
|
211
|
3IFO
|
- |
ASP ALA GLU PHE ARG HIS ASP
|
n/a
|
n/a
|
212
|
2CGR
|
Kd
=
53
nM |
GAS
|
C23 H20 N4 O2
|
c1ccc(cc1)....
|
213
|
1YNK
|
- |
SC5
|
C18 H26 N4 O2
|
C[C@H](c1c....
|
214
|
1I7Z
|
Kd
=
0.4
uM |
COC
|
C17 H21 N O4
|
C[N@]1[C@H....
|
215
|
2O5Z
|
Kd
=
110
mM |
ANO
|
C19 H28 O2
|
C[C@]12CCC....
|
216
|
25C8
|
- |
GEP
|
C19 H29 N2 O3
|
C[N+]1(CCC....
|
217
|
35C8
|
- |
NOX
|
C18 H26 N2 O4
|
c1cc(ccc1C....
|
218
|
1FL3
|
Kd
=
0.16
uM |
SPB
|
C19 H19 N O3
|
c1ccc(cc1)....
|
219
|
3CFB
|
- |
SPB
|
C19 H19 N O3
|
c1ccc(cc1)....
|
220
|
1UB5
|
- |
SPB
|
C19 H19 N O3
|
c1ccc(cc1)....
|
221
|
6LRA
|
Kd
=
0.41
uM |
VAL GLN ILE ILE ASN LYS
|
n/a
|
n/a
|
222
|
1IND
|
Ka
=
11000000000
M^-1 |
EOT
|
C20 H28 N4 O9 S
|
c1cc(ccc1C....
|
223
|
1ZEA
|
Kd
=
6
uM |
DVA DPR GLY DSN DGN DHI DTY DAS DSN
|
n/a
|
n/a
|
224
|
1MEX
|
- |
RAC
|
C18 H18 N2 O5
|
CN(C)C(=O)....
|
225
|
1UM5
|
- |
SS1
|
C8 H10 O
|
C[C@@H](c1....
|
226
|
1UM4
|
- |
SH4
|
C17 H19 N O4 P
|
C[C@@H](c1....
|
227
|
1VPO
|
Kd
=
0.000000064
M |
TES
|
C19 H28 O2
|
C[C@]12CC[....
|
228
|
1C5C
|
Kd
=
110
nM |
TK4
|
C12 H11 N O7 S2
|
CC(=O)Nc1c....
|
229
|
2PCP
|
Kd
=
2
nM |
1PC
|
C17 H25 N
|
c1ccc(cc1)....
|
230
|
1D6V
|
Kd
=
670
nM |
HOP
|
C23 H27 N O4
|
c1ccc(cc1)....
|
231
|
1Q0Y
|
Kd
~
1
nM |
MOI
|
C17 H19 N O3
|
C[N@]1CC[C....
|
232
|
6CDO
|
- |
ALA VAL GLY ILE GLY ALA VAL PHE
|
n/a
|
n/a
|
233
|
6IDG
|
Kd
=
0.000000064
M |
64T 5PY
|
n/a
|
n/a
|
234
|
4YHK
|
ic50
=
4.6
nM |
4CC
|
C25 H25 N7 O3
|
[H]/N=C(c1....
|
235
|
4YHM
|
Kd
=
173
pM |
4CC
|
C25 H25 N7 O3
|
[H]/N=C(c1....
|
236
|
4YHO
|
Kd
=
18
pM |
4CC
|
C25 H25 N7 O3
|
[H]/N=C(c1....
|
237
|
4YHI
|
ic50
=
4.6
nM |
4CC
|
C25 H25 N7 O3
|
[H]/N=C(c1....
|
238
|
3O6M
|
Kd
=
33
nM |
PRO LYS LEU GLU PRO TRP LYS HIS PRO
|
n/a
|
n/a
|
239
|
1IGJ
|
Kd
=
0.1
nM |
DGX
|
C41 H64 O14
|
C[C@@H]1[C....
|
240
|
1UZ8
|
Ka
=
93000
M^-1 |
MAG FUC GAL
|
n/a
|
n/a
|
241
|
4ODT
|
- |
GP1 Z9M
|
n/a
|
n/a
|
242
|
1RUM
|
- |
BEZ
|
C7 H6 O2
|
c1ccc(cc1)....
|
243
|
1ND0
|
- |
DP4
|
C14 H23 N O Si
|
C[N+]1(CCC....
|
244
|
3LEY
|
- |
LEU LEU GLU LEU ASP LYS TRP ALA NH2
|
n/a
|
n/a
|
245
|
1RUP
|
- |
BEZ
|
C7 H6 O2
|
c1ccc(cc1)....
|
246
|
1RU9
|
- |
BEZ
|
C7 H6 O2
|
c1ccc(cc1)....
|
247
|
1RUL
|
- |
BEZ
|
C7 H6 O2
|
c1ccc(cc1)....
|
248
|
3LEX
|
Kd
=
6.44
nM |
LEU LEU GLU LEU ASP LYS TRP ALA NH2
|
n/a
|
n/a
|
249
|
1RUK
|
- |
BEZ
|
C7 H6 O2
|
c1ccc(cc1)....
|
250
|
1NCW
|
- |
BEZ
|
C7 H6 O2
|
c1ccc(cc1)....
|
251
|
1RUA
|
- |
BEZ
|
C7 H6 O2
|
c1ccc(cc1)....
|
252
|
6BE4
|
- |
NAG NAG NAG NAG NAG
|
n/a
|
n/a
|
253
|
6BE3
|
- |
NAG
|
C8 H15 N O6
|
CC(=O)N[C@....
|