Receptor
PDB id Resolution Class Description Source Keywords
2P98 1.7 Å EC: 3.4.11.18 E. COLI METHIONINE AMINOPEPTIDASE MONOMETALATED WITH INHIBITOR YE7 ESCHERICHIA COLI MONOMETALATED MONONUCLEAR MN(II)-FORM HYDROLASE ENZYME- INHIBITOR COMPLEX METALLOENZYME
Ref.: INHIBITION OF MONOMETALATED METHIONINE AMINOPEPTIDASE: INHIBITOR DISCOVERY AND CRYSTALLOGRAPHIC ANALYSIS. J.MED.CHEM. V. 50 5735 2007
Ligand
Ligand Chain:Residue Validity Ligand Warnings Binding Data NGL Viewer Molecular Weight (Da) Formula SMILES
MN A:264;
Part of Protein;
none;
submit data
54.938 Mn [Mn+2...
NA A:265;
Part of Protein;
none;
submit data
22.99 Na [Na+]
YE7 A:266;
Valid;
none;
ic50 = 0.64 uM
226.234 C12 H10 N4 O c1ccc...
View in 3D viewer
90% Homology Family
Leader
PDB id Resolution Class Description Source Keywords
1YVM 1.6 Å EC: 3.4.11.18 E. COLI METHIONINE AMINOPEPTIDASE IN COMPLEX WITH THIABENDAZOLE ESCHERICHIA COLI HYDROLASE(ALPHA-AMINOACYLPEPTIDE) METAL COMPLEX THIABENDAZOLE METHIONINE AMINOPEPTIDASE INHIBITOR
Ref.: METAL IONS AS COFACTORS FOR THE BINDING OF INHIBITORS TO METHIONINE AMINOPEPTIDASE: A CRITICAL VIEW OF THE RELEVANCE OF IN VITRO METALLOENZYME ASSAYS. ANGEW.CHEM.INT.ED.ENGL. V. 44 3620 2005
Members (36)
No: PDB id Binding Data Representative ligand Formula Smiles
The Class containing this family consists of a total of 8 families.
1 2GG0 ic50 = 1.7 uM U11 C16 H20 F3 N3 O5 C[C@@H](C(....
2 1YVM Ki = 0.4 uM TMG C10 H7 N3 S c1ccc2c(c1....
3 2GU6 - NLP C5 H14 N O3 P CCCC[C@H](....
4 2Q95 ic50 = 1.6 uM A05 C11 H6 Cl N O5 c1cc(c(cc1....
5 2GG8 ic50 = 25 uM U15 C20 H31 N3 O5 Cc1ccc(cc1....
6 2GTX - NLP C5 H14 N O3 P CCCC[C@H](....
7 2EVC ic50 = 0.29 uM FC3 C12 H7 F3 O3 c1ccc(c(c1....
8 4A6W ic50 = 1.9 uM 5C1 C10 H7 Cl N2 O3 c1ccc(c(c1....
9 2GG3 ic50 = 0.58 uM U13 C9 H7 F N6 [H]/N=C/1C....
10 3D27 ic50 = 55.7 uM W29 C12 H12 O2 S CCc1ccsc1c....
11 2GG7 ic50 = 1.75 uM U14 C10 H8 N6 O2 [H]/N=C1/C....
12 2GU5 - NLP C5 H14 N O3 P CCCC[C@H](....
13 1XNZ ic50 = 0.24 uM FCD C11 H7 Cl O3 c1ccc(c(c1....
14 4A6V ic50 = 1.9 uM IKY C11 H7 F3 N2 O3 c1ccc(c(c1....
15 1C21 - MET C5 H11 N O2 S CSCC[C@@H]....
16 2Q92 ic50 = 1.1 uM B23 C11 H7 N O5 c1ccc(c(c1....
17 1C27 - NLP C5 H14 N O3 P CCCC[C@H](....
18 1C24 - MPJ C4 H12 N O2 P S CSCC[C@H](....
19 2EVO ic50 = 0.067 uM CT0 C10 H13 N3 O2 S c1csc(n1)N....
20 2P99 ic50 = 1.16 uM YE6 C11 H9 Cl N2 O2 c1ccc(c(c1....
21 2GG9 ic50 = 3.5 uM U16 C22 H35 N3 O5 CC(C)C[C@H....
22 2Q94 ic50 = 0.37 uM A04 C12 H7 F3 O4 c1ccc(c(c1....
23 2P98 ic50 = 0.64 uM YE7 C12 H10 N4 O c1ccc2c(c1....
24 2GGB ic50 = 12 uM U17 C17 H33 N3 O6 CCCC[C@H](....
25 2EVM ic50 = 0.693 uM FC2 C11 H6 Cl2 O3 c1cc(c(cc1....
26 1C22 - MF3 C5 H8 F3 N O2 S C(CSC(F)(F....
27 1C23 - MPH C4 H12 N O3 P S CSCC[C@H](....
28 2Q96 ic50 = 1.2 uM A18 C12 H9 Cl O3 c1ccc(c(c1....
29 2BB7 ic50 = 2.14 uM QMS C10 H10 N2 O2 S CS(=O)(=O)....
30 2GG2 ic50 = 0.25 uM U12 C10 H7 F3 N6 c1cc(cc(c1....
31 2GGC - MET C5 H11 N O2 S CSCC[C@@H]....
32 2GU4 - NLP C5 H14 N O3 P CCCC[C@H](....
33 2Q93 ic50 = 0.56 uM B21 C12 H10 O4 COc1ccccc1....
34 2GG5 ic50 = 0.25 uM U19 C10 H7 F3 N6 [H]/N=C1/C....
35 3MAT - AHH ALA LEU VAL 0A9 n/a n/a
36 2P9A ic50 = 6.56 uM YE6 C11 H9 Cl N2 O2 c1ccc(c(c1....
70% Homology Family (36)
No: PDB id Binding Data Representative ligand Formula Smiles
The Class containing this family consists of a total of 6 families.
1 2GG0 ic50 = 1.7 uM U11 C16 H20 F3 N3 O5 C[C@@H](C(....
2 1YVM Ki = 0.4 uM TMG C10 H7 N3 S c1ccc2c(c1....
3 2GU6 - NLP C5 H14 N O3 P CCCC[C@H](....
4 2Q95 ic50 = 1.6 uM A05 C11 H6 Cl N O5 c1cc(c(cc1....
5 2GG8 ic50 = 25 uM U15 C20 H31 N3 O5 Cc1ccc(cc1....
6 2GTX - NLP C5 H14 N O3 P CCCC[C@H](....
7 2EVC ic50 = 0.29 uM FC3 C12 H7 F3 O3 c1ccc(c(c1....
8 4A6W ic50 = 1.9 uM 5C1 C10 H7 Cl N2 O3 c1ccc(c(c1....
9 2GG3 ic50 = 0.58 uM U13 C9 H7 F N6 [H]/N=C/1C....
10 3D27 ic50 = 55.7 uM W29 C12 H12 O2 S CCc1ccsc1c....
11 2GG7 ic50 = 1.75 uM U14 C10 H8 N6 O2 [H]/N=C1/C....
12 2GU5 - NLP C5 H14 N O3 P CCCC[C@H](....
13 1XNZ ic50 = 0.24 uM FCD C11 H7 Cl O3 c1ccc(c(c1....
14 4A6V ic50 = 1.9 uM IKY C11 H7 F3 N2 O3 c1ccc(c(c1....
15 1C21 - MET C5 H11 N O2 S CSCC[C@@H]....
16 2Q92 ic50 = 1.1 uM B23 C11 H7 N O5 c1ccc(c(c1....
17 1C27 - NLP C5 H14 N O3 P CCCC[C@H](....
18 1C24 - MPJ C4 H12 N O2 P S CSCC[C@H](....
19 2EVO ic50 = 0.067 uM CT0 C10 H13 N3 O2 S c1csc(n1)N....
20 2P99 ic50 = 1.16 uM YE6 C11 H9 Cl N2 O2 c1ccc(c(c1....
21 2GG9 ic50 = 3.5 uM U16 C22 H35 N3 O5 CC(C)C[C@H....
22 2Q94 ic50 = 0.37 uM A04 C12 H7 F3 O4 c1ccc(c(c1....
23 2P98 ic50 = 0.64 uM YE7 C12 H10 N4 O c1ccc2c(c1....
24 2GGB ic50 = 12 uM U17 C17 H33 N3 O6 CCCC[C@H](....
25 2EVM ic50 = 0.693 uM FC2 C11 H6 Cl2 O3 c1cc(c(cc1....
26 1C22 - MF3 C5 H8 F3 N O2 S C(CSC(F)(F....
27 1C23 - MPH C4 H12 N O3 P S CSCC[C@H](....
28 2Q96 ic50 = 1.2 uM A18 C12 H9 Cl O3 c1ccc(c(c1....
29 2BB7 ic50 = 2.14 uM QMS C10 H10 N2 O2 S CS(=O)(=O)....
30 2GG2 ic50 = 0.25 uM U12 C10 H7 F3 N6 c1cc(cc(c1....
31 2GGC - MET C5 H11 N O2 S CSCC[C@@H]....
32 2GU4 - NLP C5 H14 N O3 P CCCC[C@H](....
33 2Q93 ic50 = 0.56 uM B21 C12 H10 O4 COc1ccccc1....
34 2GG5 ic50 = 0.25 uM U19 C10 H7 F3 N6 [H]/N=C1/C....
35 3MAT - AHH ALA LEU VAL 0A9 n/a n/a
36 2P9A ic50 = 6.56 uM YE6 C11 H9 Cl N2 O2 c1ccc(c(c1....
50% Homology Family (69)
No: PDB id Binding Data Representative ligand Formula Smiles
The Class containing this family consists of a total of 3 families.
1 2NQ6 ic50 = 1.5 uM HM4 C14 H16 N4 O3 S CC(C)(C)OC....
2 4U69 Ki = 54.8 uM Q07 C6 H16 N O3 P CCC[C@H](C....
3 2G6P ic50 = 0.6 uM HM2 C18 H17 Cl N4 Cc1c(c(nc(....
4 4U73 Ki = 6.6 uM Q02 C7 H10 N O3 P c1ccc(cc1)....
5 4IKT ic50 = 0.67 uM TFV C18 H16 Cl F3 N6 Cc1c(c(nc(....
6 4U6Z Ki = 3.9 uM Q07 C6 H16 N O3 P CCC[C@H](C....
7 4U70 Ki = 9.5 uM Q04 C8 H18 N O3 P C1CCC(CC1)....
8 4FLI ic50 = 3.59 uM Y16 C14 H26 N2 O6 CC(C)(C)/C....
9 4U6C Ki = 9.9 uM Q06 C8 H18 N O3 P C1CCC(C1)C....
10 4IKR ic50 = 0.59 uM PVP C16 H20 Cl N5 O Cc1c(c(nc(....
11 4FLK ic50 = 5.58 uM Y10 C21 H31 N O5 CC(C)(C)/C....
12 4IKU ic50 = 1.79 uM SHX C19 H18 Cl N5 O Cc1c(c(nc(....
13 2NQ7 ic50 = 2.9 uM HM5 C14 H16 N4 O2 S CC(C)(C)C(....
14 4FLL ic50 = 5.14 uM YZ6 C25 H35 N O6 CC(C)(C)/C....
15 4U71 Ki = 6 uM Q03 C7 H16 N O3 P C1CCC(CC1)....
16 4HXX - 1AY C28 H29 Cl2 N5 Cc1c(c(nc(....
17 4IKS ic50 = 7.23 uM TFD C18 H16 Cl F3 N6 Cc1c(c(nc(....
18 4U6E Ki = 111.6 uM Q02 C7 H10 N O3 P c1ccc(cc1)....
19 4U1B Ki = 4.9 uM Q08 C8 H20 N O3 P CCCC(CCC)[....
20 4FLJ ic50 = 7.45 uM Y08 C22 H38 N2 O6 CC(C)(C)/C....
21 2GG0 ic50 = 1.7 uM U11 C16 H20 F3 N3 O5 C[C@@H](C(....
22 1YVM Ki = 0.4 uM TMG C10 H7 N3 S c1ccc2c(c1....
23 2GU6 - NLP C5 H14 N O3 P CCCC[C@H](....
24 2Q95 ic50 = 1.6 uM A05 C11 H6 Cl N O5 c1cc(c(cc1....
25 2GG8 ic50 = 25 uM U15 C20 H31 N3 O5 Cc1ccc(cc1....
26 2GTX - NLP C5 H14 N O3 P CCCC[C@H](....
27 2EVC ic50 = 0.29 uM FC3 C12 H7 F3 O3 c1ccc(c(c1....
28 4A6W ic50 = 1.9 uM 5C1 C10 H7 Cl N2 O3 c1ccc(c(c1....
29 2GG3 ic50 = 0.58 uM U13 C9 H7 F N6 [H]/N=C/1C....
30 3D27 ic50 = 55.7 uM W29 C12 H12 O2 S CCc1ccsc1c....
31 2GG7 ic50 = 1.75 uM U14 C10 H8 N6 O2 [H]/N=C1/C....
32 2GU5 - NLP C5 H14 N O3 P CCCC[C@H](....
33 1XNZ ic50 = 0.24 uM FCD C11 H7 Cl O3 c1ccc(c(c1....
34 4A6V ic50 = 1.9 uM IKY C11 H7 F3 N2 O3 c1ccc(c(c1....
35 1C21 - MET C5 H11 N O2 S CSCC[C@@H]....
36 2Q92 ic50 = 1.1 uM B23 C11 H7 N O5 c1ccc(c(c1....
37 1C27 - NLP C5 H14 N O3 P CCCC[C@H](....
38 1C24 - MPJ C4 H12 N O2 P S CSCC[C@H](....
39 2EVO ic50 = 0.067 uM CT0 C10 H13 N3 O2 S c1csc(n1)N....
40 2P99 ic50 = 1.16 uM YE6 C11 H9 Cl N2 O2 c1ccc(c(c1....
41 2GG9 ic50 = 3.5 uM U16 C22 H35 N3 O5 CC(C)C[C@H....
42 2Q94 ic50 = 0.37 uM A04 C12 H7 F3 O4 c1ccc(c(c1....
43 2P98 ic50 = 0.64 uM YE7 C12 H10 N4 O c1ccc2c(c1....
44 2GGB ic50 = 12 uM U17 C17 H33 N3 O6 CCCC[C@H](....
45 2EVM ic50 = 0.693 uM FC2 C11 H6 Cl2 O3 c1cc(c(cc1....
46 1C22 - MF3 C5 H8 F3 N O2 S C(CSC(F)(F....
47 1C23 - MPH C4 H12 N O3 P S CSCC[C@H](....
48 2Q96 ic50 = 1.2 uM A18 C12 H9 Cl O3 c1ccc(c(c1....
49 2BB7 ic50 = 2.14 uM QMS C10 H10 N2 O2 S CS(=O)(=O)....
50 2GG2 ic50 = 0.25 uM U12 C10 H7 F3 N6 c1cc(cc(c1....
51 2GGC - MET C5 H11 N O2 S CSCC[C@@H]....
52 2GU4 - NLP C5 H14 N O3 P CCCC[C@H](....
53 2Q93 ic50 = 0.56 uM B21 C12 H10 O4 COc1ccccc1....
54 2GG5 ic50 = 0.25 uM U19 C10 H7 F3 N6 [H]/N=C1/C....
55 3MAT - AHH ALA LEU VAL 0A9 n/a n/a
56 2P9A ic50 = 6.56 uM YE6 C11 H9 Cl N2 O2 c1ccc(c(c1....
57 4IU6 - FZ1 C24 H23 N5 O COc1ccc(cc....
58 1QXZ ic50 = 19 uM M3C C8 H14 N2 O2 S2 CSCC[C@@H]....
59 1QXY ic50 = 16 uM M2C C10 H16 N2 O2 S CSCC[C@@H]....
60 1QXW ic50 = 7 uM M1C C10 H22 N2 O2 CCCC[C@@H]....
61 3IU9 ic50 = 0.24 uM T07 C9 H8 Cl2 N4 S c1cc(c(cc1....
62 3IU7 ic50 = 16 uM FCD C11 H7 Cl O3 c1ccc(c(c1....
63 3PKE - Y10 C21 H31 N O5 CC(C)(C)/C....
64 3PKB ic50 = 0.62 uM Y16 C14 H26 N2 O6 CC(C)(C)/C....
65 3PKA ic50 = 0.54 uM Y02 C23 H37 N O6 Cc1cc(c(c(....
66 3PKC ic50 = 0.96 uM Y08 C22 H38 N2 O6 CC(C)(C)/C....
67 3IU8 ic50 = 0.58 uM T03 C9 H8 F N3 S c1cc(ccc1C....
68 3PKD ic50 = 0.76 uM Y10 C21 H31 N O5 CC(C)(C)/C....
69 1YJ3 - MET C5 H11 N O2 S CSCC[C@@H]....
Polypharmacology
Similar Ligands (2D)
Ligand no: 1; Ligand: YE7; Similar ligands found: 1
No: Ligand ECFP6 Tc MDL keys Tc
1 YE7 1 1
Similar Ligands (3D)
Ligand no: 1; Ligand: YE7; Similar ligands found: 736
No: Ligand Similarity coefficient
1 RGK 0.9635
2 YE6 0.9622
3 F40 0.9620
4 NKI 0.9595
5 WLH 0.9541
6 1V3 0.9523
7 2GQ 0.9520
8 TCR 0.9495
9 JCZ 0.9470
10 W8L 0.9467
11 CDJ 0.9458
12 H2W 0.9454
13 IDZ 0.9454
14 7L4 0.9436
15 1V1 0.9425
16 DFL 0.9420
17 20D 0.9409
18 A73 0.9400
19 PIQ 0.9400
20 2P3 0.9392
21 5NN 0.9385
22 AMR 0.9381
23 5V7 0.9381
24 2QU 0.9375
25 FCD 0.9369
26 1FE 0.9368
27 AGI 0.9368
28 3WL 0.9352
29 II4 0.9347
30 1V4 0.9342
31 P4L 0.9338
32 25F 0.9337
33 SZ5 0.9337
34 QUB 0.9332
35 D80 0.9324
36 LL1 0.9321
37 QIV 0.9314
38 5WT 0.9312
39 3F4 0.9312
40 5B2 0.9310
41 DDC 0.9309
42 2JX 0.9307
43 C09 0.9306
44 5E5 0.9303
45 EV2 0.9302
46 A63 0.9301
47 E9L 0.9297
48 Q0K 0.9297
49 TRP 0.9294
50 JVD 0.9288
51 9CE 0.9281
52 IOP 0.9281
53 M78 0.9279
54 UN9 0.9275
55 DXK 0.9272
56 9BF 0.9271
57 4AU 0.9264
58 I2E 0.9263
59 M3W 0.9261
60 0DF 0.9259
61 3GX 0.9251
62 GNV 0.9244
63 ITE 0.9244
64 4ZF 0.9242
65 NRA 0.9241
66 Q5M 0.9241
67 5F8 0.9240
68 MN QAY 0.9239
69 6DQ 0.9233
70 JTA 0.9232
71 LIG 0.9230
72 J38 0.9222
73 L07 0.9220
74 VT3 0.9216
75 RSV 0.9215
76 ZHA 0.9214
77 B21 0.9213
78 XG1 0.9212
79 52F 0.9211
80 6ZW 0.9208
81 N1E 0.9208
82 IKY 0.9207
83 5WN 0.9203
84 27M 0.9201
85 LI7 0.9201
86 0UL 0.9201
87 C0W 0.9200
88 Y3L 0.9199
89 57D 0.9193
90 DRG 0.9192
91 9JT 0.9191
92 S60 0.9191
93 S98 0.9191
94 D87 0.9189
95 5WK 0.9189
96 ZZA 0.9188
97 IQZ 0.9187
98 C4E 0.9187
99 AVA 0.9186
100 A6W 0.9186
101 08C 0.9185
102 5FL 0.9183
103 39Z 0.9180
104 JP2 0.9179
105 G14 0.9177
106 1AJ 0.9171
107 49P 0.9170
108 5TZ 0.9169
109 M4N 0.9165
110 P83 0.9165
111 L1T 0.9162
112 BIK 0.9161
113 VM1 0.9160
114 5SJ 0.9158
115 NAR 0.9156
116 H75 0.9154
117 BGU 0.9152
118 2WU 0.9151
119 X2M 0.9151
120 8G6 0.9150
121 7FU 0.9147
122 6JM 0.9145
123 AJG 0.9145
124 3D8 0.9145
125 AVX 0.9144
126 YZ9 0.9144
127 6XC 0.9144
128 5WW 0.9143
129 VUP 0.9141
130 NIF 0.9141
131 27F 0.9141
132 CX4 0.9140
133 JBZ 0.9139
134 YEX 0.9135
135 1Q4 0.9134
136 X0T 0.9133
137 JFS 0.9132
138 ZEA 0.9132
139 1EL 0.9130
140 ODK 0.9129
141 91F 0.9129
142 WG8 0.9129
143 7EH 0.9127
144 A9B 0.9127
145 0LO 0.9124
146 3VX 0.9123
147 CX6 0.9122
148 LP8 0.9122
149 NAL 0.9121
150 833 0.9120
151 CZ0 0.9117
152 5ER 0.9117
153 47V 0.9116
154 L3L 0.9115
155 5TY 0.9113
156 2QV 0.9112
157 0OK 0.9110
158 EWG 0.9108
159 HH6 0.9104
160 A5H 0.9103
161 Z21 0.9102
162 3VQ 0.9100
163 HA6 0.9099
164 AP6 0.9098
165 363 0.9096
166 ZYQ 0.9096
167 KMP 0.9095
168 1QP 0.9094
169 O9Q 0.9091
170 DX2 0.9091
171 DX7 0.9091
172 RVE 0.9089
173 SU9 0.9088
174 4FF 0.9088
175 2JK 0.9086
176 1FL 0.9085
177 TXW 0.9084
178 CUE 0.9084
179 ET0 0.9083
180 5P3 0.9082
181 4CN 0.9082
182 6BK 0.9080
183 272 0.9080
184 LR2 0.9079
185 DTR 0.9078
186 6TJ 0.9077
187 XJ2 0.9075
188 1UZ 0.9075
189 KWB 0.9074
190 FER 0.9074
191 R4E 0.9074
192 HBO 0.9071
193 3JC 0.9068
194 PRL 0.9067
195 AXX 0.9066
196 ZIP 0.9065
197 HRD 0.9064
198 GNJ 0.9064
199 6JO 0.9062
200 LEL 0.9058
201 1HP 0.9057
202 FC2 0.9057
203 1V8 0.9052
204 338 0.9052
205 2J1 0.9052
206 78Y 0.9051
207 GO2 0.9050
208 BA5 0.9050
209 S62 0.9049
210 AJ1 0.9049
211 OX2 0.9046
212 QUE 0.9045
213 1XS 0.9044
214 D25 0.9044
215 N91 0.9043
216 SNJ 0.9042
217 JTF 0.9041
218 H4B 0.9041
219 2D2 0.9038
220 TMG 0.9038
221 FCW 0.9036
222 HRM 0.9036
223 5F5 0.9035
224 34L 0.9035
225 22T 0.9034
226 KLE 0.9033
227 S1D 0.9033
228 LTN 0.9032
229 JMG 0.9032
230 1DR 0.9030
231 4HG 0.9029
232 LUM 0.9029
233 ZRK 0.9027
234 4GU 0.9025
235 0FR 0.9025
236 BRY 0.9024
237 NK5 0.9024
238 JSX 0.9024
239 2LW 0.9023
240 ZSP 0.9023
241 ZME 0.9022
242 RUG 0.9022
243 5VU 0.9021
244 KU1 0.9021
245 VBC 0.9019
246 P7V 0.9018
247 FT6 0.9017
248 V1T 0.9016
249 108 0.9015
250 3SU 0.9014
251 EY2 0.9014
252 7G2 0.9013
253 30G 0.9013
254 3IL 0.9013
255 FNT 0.9012
256 6QT 0.9011
257 L5D 0.9011
258 0SY 0.9010
259 8CC 0.9009
260 HBI 0.9006
261 68A 0.9006
262 G6P 0.9005
263 K7H 0.9003
264 2UD 0.9002
265 LU2 0.9001
266 96Z 0.9001
267 MR4 0.9000
268 JF8 0.8998
269 4UM 0.8998
270 4I8 0.8995
271 OPA 0.8995
272 KLV 0.8993
273 JRO 0.8993
274 B2E 0.8991
275 3WN 0.8990
276 3WO 0.8990
277 774 0.8990
278 B23 0.8986
279 GVI 0.8986
280 7I2 0.8984
281 H35 0.8983
282 9UL 0.8983
283 9OF 0.8983
284 4YE 0.8982
285 78P 0.8981
286 H7S 0.8980
287 CHQ 0.8978
288 OCZ 0.8978
289 NYJ 0.8976
290 OTA 0.8974
291 801 0.8974
292 BIO 0.8974
293 0H5 0.8972
294 9F8 0.8972
295 NIY 0.8971
296 MUX 0.8969
297 STV 0.8968
298 GEN 0.8968
299 CKA 0.8966
300 FQX 0.8966
301 MBP 0.8963
302 1QV 0.8962
303 2FX 0.8962
304 1X8 0.8961
305 D9Z 0.8960
306 EQA 0.8958
307 LC1 0.8958
308 19E 0.8956
309 26C 0.8956
310 B4L 0.8948
311 IQQ 0.8948
312 Q4G 0.8947
313 4Z9 0.8946
314 NEU 0.8943
315 6C8 0.8943
316 J1K 0.8943
317 0SX 0.8942
318 6MW 0.8942
319 9XZ 0.8942
320 SDN 0.8940
321 7MX 0.8939
322 40N 0.8937
323 GNG 0.8937
324 PUE 0.8936
325 BBY 0.8935
326 18E 0.8934
327 97K 0.8931
328 U13 0.8930
329 FF2 0.8930
330 6FB 0.8927
331 DHC 0.8926
332 EVO 0.8926
333 D64 0.8925
334 8M5 0.8924
335 ZRL 0.8922
336 BG6 0.8920
337 COL 0.8920
338 DNQ 0.8919
339 O9T 0.8917
340 SGW 0.8916
341 NFZ 0.8915
342 BHF 0.8915
343 5GV 0.8914
344 4BL 0.8913
345 28A 0.8912
346 DK1 0.8910
347 MKN 0.8909
348 5TO 0.8908
349 6FG 0.8907
350 X8E 0.8906
351 M3F 0.8904
352 344 0.8904
353 AUV 0.8904
354 4AB 0.8902
355 GJK 0.8902
356 NU3 0.8902
357 M5H 0.8901
358 55D 0.8899
359 AQN 0.8899
360 FY8 0.8899
361 8NX 0.8898
362 BJ4 0.8898
363 F5C 0.8896
364 0K7 0.8895
365 XCG 0.8895
366 AC2 0.8894
367 FHV 0.8890
368 0NJ 0.8890
369 HNT 0.8889
370 O9Z 0.8888
371 5OR 0.8886
372 CTE 0.8883
373 5H6 0.8883
374 LWS 0.8882
375 245 0.8879
376 DFV 0.8879
377 6KT 0.8879
378 LOT 0.8876
379 78U 0.8876
380 QMS 0.8875
381 Q9T 0.8874
382 GOE 0.8872
383 PJK 0.8870
384 MD6 0.8869
385 U4J 0.8869
386 M9N 0.8866
387 EES 0.8866
388 IQ5 0.8866
389 6HP 0.8865
390 0ON 0.8864
391 GA2 0.8863
392 BUX 0.8862
393 3DE 0.8862
394 WUB 0.8861
395 4R1 0.8860
396 5E1 0.8860
397 JWS 0.8859
398 4BX 0.8859
399 H2B 0.8858
400 5XL 0.8858
401 4BY 0.8857
402 LFQ 0.8857
403 U7E 0.8856
404 5GT 0.8855
405 C9M 0.8854
406 ML1 0.8853
407 X0U 0.8853
408 V2Z 0.8852
409 KYN 0.8851
410 BBP 0.8851
411 ANC 0.8851
412 1V0 0.8850
413 20N 0.8849
414 KLS 0.8847
415 RCV 0.8844
416 4FE 0.8844
417 BPU 0.8844
418 LR8 0.8843
419 1UR 0.8842
420 S0D 0.8842
421 GNY 0.8842
422 CSN 0.8842
423 N2M 0.8842
424 ASE 0.8842
425 5ZM 0.8839
426 IXM 0.8839
427 XEV 0.8839
428 MR5 0.8838
429 4G2 0.8838
430 7O4 0.8838
431 LFN 0.8837
432 7MW 0.8837
433 LF5 0.8836
434 O82 0.8836
435 657 0.8834
436 F18 0.8834
437 CNI 0.8834
438 3WK 0.8831
439 XI7 0.8829
440 28S 0.8829
441 1EB 0.8829
442 4L2 0.8828
443 RFZ 0.8828
444 CC6 0.8827
445 3D1 0.8826
446 FSE 0.8826
447 6DH 0.8825
448 64F 0.8825
449 3ZB 0.8823
450 THA 0.8823
451 NPX 0.8823
452 WV7 0.8823
453 BVS 0.8822
454 4K2 0.8822
455 D8Q 0.8822
456 6QF 0.8821
457 3AK 0.8821
458 6C5 0.8820
459 HWB 0.8819
460 QR2 0.8816
461 SSY 0.8816
462 8XL 0.8814
463 NPS 0.8813
464 SLS 0.8811
465 DX8 0.8810
466 KP2 0.8810
467 4NR 0.8808
468 6C4 0.8807
469 CWE 0.8806
470 KYA 0.8805
471 ZTW 0.8804
472 PLP 0.8804
473 39R 0.8804
474 P93 0.8803
475 EZL 0.8802
476 GDL 0.8801
477 EQU 0.8800
478 5WS 0.8800
479 N0Z 0.8798
480 9KZ 0.8796
481 22L 0.8793
482 CG 0.8792
483 OQC 0.8792
484 27K 0.8791
485 GO8 0.8790
486 8NB 0.8789
487 OUG 0.8789
488 RHN 0.8788
489 CIY 0.8788
490 P9I 0.8788
491 K48 0.8788
492 7M5 0.8787
493 SKF 0.8785
494 UN4 0.8784
495 5EZ 0.8783
496 F36 0.8782
497 K25 0.8781
498 IOS 0.8781
499 5AD 0.8780
500 122 0.8780
501 CR4 0.8780
502 E1T 0.8780
503 BMZ 0.8779
504 N7I 0.8778
505 OLU 0.8778
506 PTS 0.8778
507 SJK 0.8778
508 NDG 0.8777
509 8D6 0.8777
510 6H2 0.8777
511 HMZ 0.8777
512 5WM 0.8777
513 X48 0.8777
514 BDI 0.8774
515 HWH 0.8773
516 G2V 0.8770
517 2PV 0.8769
518 NDD 0.8768
519 0JD 0.8768
520 PE2 0.8767
521 1R5 0.8767
522 SRO 0.8767
523 8SK 0.8766
524 2PK 0.8765
525 5KN 0.8765
526 36I 0.8765
527 3J8 0.8764
528 BP7 0.8764
529 5F1 0.8763
530 0MB 0.8761
531 6ZE 0.8759
532 NWD 0.8758
533 8RK 0.8756
534 JMM 0.8755
535 ANF 0.8755
536 D2G 0.8754
537 6GP 0.8753
538 MR6 0.8753
539 BHS 0.8752
540 3Y7 0.8748
541 9NB 0.8748
542 DT7 0.8745
543 GNM 0.8745
544 4MB 0.8744
545 PNX 0.8743
546 IQW 0.8743
547 3D3 0.8742
548 E1K 0.8741
549 B61 0.8740
550 KWV 0.8739
551 CR1 0.8739
552 A7H 0.8739
553 7LU 0.8739
554 0FK 0.8739
555 L22 0.8734
556 THM 0.8734
557 DNA 0.8731
558 BMC 0.8730
559 9TF 0.8730
560 Q8G 0.8729
561 IDD 0.8729
562 4NP 0.8727
563 120 0.8725
564 5P7 0.8725
565 1YL 0.8723
566 54X 0.8723
567 IBP 0.8722
568 CDY 0.8721
569 8HC 0.8720
570 7M2 0.8719
571 0NX 0.8718
572 AA 0.8715
573 5M2 0.8715
574 4MP 0.8714
575 1A7 0.8714
576 GB4 0.8713
577 4V2 0.8712
578 0XR 0.8709
579 4GP 0.8709
580 5DE 0.8707
581 MIL 0.8706
582 EMU 0.8706
583 6P3 0.8706
584 8YH 0.8706
585 JY4 0.8705
586 3R4 0.8705
587 WA2 0.8705
588 7G0 0.8703
589 HA5 0.8703
590 92P 0.8702
591 CMG 0.8702
592 HHS 0.8701
593 E3X 0.8700
594 KMY 0.8700
595 A5Q 0.8700
596 JHY 0.8696
597 2K8 0.8695
598 MJW 0.8694
599 RKV 0.8694
600 OAI 0.8693
601 397 0.8692
602 124 0.8692
603 NAG 0.8692
604 7KE 0.8690
605 MUR 0.8689
606 1HR 0.8689
607 B56 0.8689
608 1SF 0.8688
609 1ZC 0.8686
610 EST 0.8685
611 UN3 0.8685
612 6C9 0.8684
613 549 0.8684
614 JF5 0.8682
615 H5B 0.8682
616 CK2 0.8677
617 BL7 0.8677
618 AZY 0.8676
619 X2L 0.8676
620 DH2 0.8675
621 DBE 0.8675
622 S0E 0.8673
623 L03 0.8673
624 JAH 0.8672
625 HUL 0.8672
626 B0K 0.8671
627 CC5 0.8670
628 BZJ 0.8670
629 8Y7 0.8668
630 EAE 0.8668
631 0J4 0.8665
632 795 0.8665
633 M6Z 0.8664
634 D26 0.8664
635 1HN 0.8664
636 EUE 0.8662
637 8HH 0.8662
638 M4E 0.8661
639 4HB 0.8661
640 A64 0.8659
641 P80 0.8659
642 JGY 0.8657
643 A05 0.8656
644 MFZ 0.8656
645 GLP 0.8654
646 1CE 0.8654
647 1OT 0.8652
648 P9E 0.8652
649 2UV 0.8652
650 PMP 0.8651
651 GJP 0.8651
652 3QV 0.8650
653 15N 0.8648
654 4KL 0.8646
655 O53 0.8645
656 92O 0.8642
657 3C3 0.8640
658 RF2 0.8639
659 121 0.8638
660 9AP 0.8637
661 X6W 0.8637
662 AJ4 0.8636
663 GJG 0.8633
664 761 0.8632
665 LDR 0.8632
666 G1P 0.8632
667 HFT 0.8631
668 MFR 0.8629
669 3N0 0.8628
670 DE7 0.8627
671 MS0 0.8626
672 5RP 0.8623
673 U14 0.8622
674 5E2 0.8622
675 XYP XYP 0.8622
676 8HG 0.8621
677 A8D 0.8621
678 E3U 0.8621
679 62D 0.8620
680 OSY 0.8619
681 6SD 0.8616
682 A6P 0.8616
683 4RU 0.8610
684 MZM 0.8610
685 AH9 0.8608
686 XIF XYP 0.8608
687 3VS 0.8608
688 BXS 0.8607
689 CXH 0.8604
690 9ZE 0.8603
691 DAH 0.8600
692 KTW 0.8599
693 ALR 0.8599
694 FZM 0.8598
695 4Z1 0.8598
696 IA2 0.8593
697 51Y 0.8591
698 4RG 0.8588
699 F02 0.8588
700 RDT 0.8585
701 D1G 0.8584
702 U12 0.8584
703 AN3 0.8584
704 AJY 0.8583
705 DQH 0.8581
706 9FE 0.8578
707 YIP 0.8578
708 EV3 0.8577
709 5DN 0.8576
710 F2W 0.8570
711 NPL 0.8570
712 2L2 0.8570
713 BPY 0.8570
714 6J9 0.8570
715 J6W 0.8569
716 IMH 0.8566
717 GI3 0.8566
718 EI1 0.8566
719 IIH 0.8563
720 JOH 0.8562
721 7FZ 0.8562
722 7GP 0.8562
723 HJ7 0.8557
724 D3G 0.8552
725 4F8 0.8550
726 TID 0.8550
727 SG2 0.8549
728 A7Q 0.8547
729 XDL XYP 0.8536
730 ALH 0.8534
731 ESI 0.8533
732 TXQ 0.8532
733 S7S 0.8530
734 27B 0.8527
735 0RY 0.8511
736 N4E 0.8507
Similar Binding Sites (Proteins are less than 50% similar to leader)
Pocket No.: 1; Query (leader) PDB : 1YVM; Ligand: TMG; Similar sites found with APoc: No similar binding sites found, or similarity not calculated due to duplicate pocket.
This union binding pocket(no: 1) in the query (biounit: 1yvm.bio1) has 18 residues
No: Leader PDB Ligand Sequence Similarity
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