1
|
5AMB
|
- |
MET VAL GLY GLY VAL VAL ILE ALA
|
n/a
|
n/a
|
2
|
4CA6
|
Ki
=
180
nM |
3EF
|
C38 H38 N3 O9 P
|
c1ccc(cc1)....
|
3
|
2XYD
|
Ki
=
150
nM |
3ES
|
C38 H38 N3 O9 P
|
c1ccc(cc1)....
|
4
|
6TT1
|
- |
1IU
|
C19 H29 N8 O5 P
|
C[C@H](CP(....
|
5
|
4BZS
|
Ki
=
75
nM |
K26
|
C25 H34 N3 O8 P
|
CC[C@H](C)....
|
6
|
5AMA
|
- |
ASP SER
|
n/a
|
n/a
|
7
|
6F9R
|
Ki
=
10.6
uM |
D0W
|
C25 H33 N3 O10
|
CC(=O)N[C@....
|
8
|
6H5X
|
- |
FT8
|
C19 H24 N2 O4 S2
|
c1ccc(cc1)....
|
9
|
4UFB
|
- |
LYS PRO
|
n/a
|
n/a
|
10
|
3NXQ
|
- |
RX4
|
C21 H31 N4 O8 P
|
C[C@H](C[P....
|
11
|
6F9V
|
Ki
=
171.9
nM |
D0Z
|
C26 H40 N4 O9 S
|
CS(=O)(=O)....
|
12
|
5AM9
|
- |
GLU VAL
|
n/a
|
n/a
|
13
|
6TT4
|
- |
FT8
|
C19 H24 N2 O4 S2
|
c1ccc(cc1)....
|
14
|
5AM8
|
- |
PHE ARG HIS ASP SER GLY TYR
|
n/a
|
n/a
|
15
|
6TT3
|
- |
BJ2
|
C18 H28 N4 O8
|
C[C@@H](C(....
|
16
|
4BXK
|
Ki
=
11.21
nM |
1IU
|
C19 H29 N8 O5 P
|
C[C@H](CP(....
|
17
|
6EN6
|
Ki
=
11.45
nM |
BJ2
|
C18 H28 N4 O8
|
C[C@@H](C(....
|
18
|
6EN5
|
Ki
=
11.45
nM |
BJ2
|
C18 H28 N4 O8
|
C[C@@H](C(....
|
19
|
4UFA
|
- |
SAC ASP
|
n/a
|
n/a
|
20
|
3ZQZ
|
- |
SLC
|
C9 H13 N O3 Se
|
C=C(C[SeH]....
|
21
|
2X8Z
|
Ki
=
11
nM |
X8Z
|
C9 H15 N O3 S
|
C[C@H](CS)....
|
22
|
2X97
|
Ki
=
2200
nM |
RX4
|
C21 H31 N4 O8 P
|
C[C@H](C[P....
|
23
|
2X93
|
- |
X93
|
C22 H30 N2 O5
|
C[C@@H](C(....
|
24
|
1J36
|
Ki
=
18
nM |
LPR
|
C21 H31 N3 O5
|
c1ccc(cc1)....
|
25
|
2X96
|
Ki
=
94
uM |
RX3
|
C33 H36 N3 O7 P
|
c1ccc(cc1)....
|
26
|
5A2R
|
- |
MLT
|
C4 H6 O5
|
C([C@H](C(....
|
27
|
4AA1
|
Ki
=
76
uM |
ASP ARG VAL TYR ILE HIS PRO PHE
|
n/a
|
n/a
|
28
|
2X90
|
- |
EAL
|
C18 H24 N2 O5
|
C[C@@H](C(....
|
29
|
2X92
|
- |
X92
|
C21 H28 N2 O5
|
C[C@@H](C(....
|
30
|
1J37
|
Ki
=
1.1
nM |
X8Z
|
C9 H15 N O3 S
|
C[C@H](CS)....
|
31
|
4CA8
|
Ki
=
120
nM |
3ES
|
C38 H38 N3 O9 P
|
c1ccc(cc1)....
|
32
|
2X8Y
|
- |
FLC
|
C6 H5 O7
|
C(C(=O)[O-....
|
33
|
2X94
|
- |
X94
|
C17 H28 N2 O5
|
CCC[C@@H](....
|
34
|
4CA7
|
Ki
=
24
nM |
3EF
|
C38 H38 N3 O9 P
|
c1ccc(cc1)....
|
35
|
4ASQ
|
- |
ARG PRO PRO GLY PHE SER PRO PHE ARG
|
n/a
|
n/a
|
36
|
2XHM
|
- |
K26
|
C25 H34 N3 O8 P
|
CC[C@H](C)....
|
37
|
2X95
|
- |
X95
|
C27 H34 N4 O5
|
c1ccc(cc1)....
|
38
|
4ASR
|
- |
ARG PRO PRO GLY PHE THR PRO PHE ARG
|
n/a
|
n/a
|
39
|
2X91
|
Ki
=
180
nM |
LPR
|
C21 H31 N3 O5
|
c1ccc(cc1)....
|
40
|
6F9U
|
- |
D0W
|
C25 H33 N3 O10
|
CC(=O)N[C@....
|
41
|
1UZF
|
- |
MCO
|
C9 H15 N O3 S
|
C[C@H](CS)....
|
42
|
3BKK
|
Ki
=
0.83
uM |
KAF
|
C28 H30 N2 O6
|
c1ccc(cc1)....
|
43
|
1O8A
|
- |
NXA
|
C4 H7 N O4
|
C[C@@H](C(....
|
44
|
2XY9
|
Ki
=
0.65
nM |
3ES
|
C38 H38 N3 O9 P
|
c1ccc(cc1)....
|
45
|
3L3N
|
- |
LSW
|
C27 H34 N4 O5
|
c1ccc(cc1)....
|
46
|
1UZE
|
- |
EAL
|
C18 H24 N2 O5
|
C[C@@H](C(....
|
47
|
6H5W
|
- |
FT8
|
C19 H24 N2 O4 S2
|
c1ccc(cc1)....
|
48
|
4BZR
|
- |
K26
|
C25 H34 N3 O8 P
|
CC[C@H](C)....
|
49
|
4APH
|
Ki
=
4
uM |
ASP ARG VAL TYR ILE HIS PRO PHE
|
n/a
|
n/a
|
50
|
2YDM
|
ic50
=
36.4
nM |
SLC
|
C9 H13 N O3 Se
|
C=C(C[SeH]....
|
51
|
1O86
|
- |
GLY
|
C2 H5 N O2
|
C(C(=O)O)N
|
52
|
6F9T
|
- |
D0Z
|
C26 H40 N4 O9 S
|
CS(=O)(=O)....
|
53
|
3BKL
|
Ki
=
0.679
uM |
KAW
|
C30 H31 N3 O6
|
c1ccc(cc1)....
|
54
|
4CA5
|
Ki
=
0.41
nM |
3EF
|
C38 H38 N3 O9 P
|
c1ccc(cc1)....
|
55
|
4C2P
|
- |
X8Z
|
C9 H15 N O3 S
|
C[C@H](CS)....
|
56
|
2OC2
|
Ki
=
3
nM |
RX3
|
C33 H36 N3 O7 P
|
c1ccc(cc1)....
|
57
|
6S1Z
|
ic50
=
1.5
nM |
KS8
|
C23 H34 N O5 P
|
c1ccc(cc1)....
|
58
|
6S1Y
|
- |
KSN
|
C10 H16 N2 O7
|
C(CC(=O)N[....
|