Receptor
PDB id Resolution Class Description Source Keywords
3K4D 2.39 Å EC: 3.2.1.31 CRYSTAL STRUCTURE OF E. COLI BETA-GLUCURONIDASE WITH THE GLU LACTAM INHIBITOR BOUND ESCHERICHIA COLI ALPHA/BETA BARREL SUGAR-BINDING DOMAIN BETA-SANDWICH DOMAIGLYCOSYL HYDROLASE GLUCARO-D-LACTAM GLYCOSIDASE HYDROLASHYDROLASE-HYDROLASE INHIBITOR COMPLEX
Ref.: ALLEVIATING CANCER DRUG TOXICITY BY INHIBITING A BA ENZYME. SCIENCE V. 330 831 2010
Ligand
Ligand Chain:Residue Validity Ligand Warnings Binding Data NGL Viewer Molecular Weight (Da) Formula SMILES
EVA A:604;
B:604;
Valid;
Valid;
none;
none;
Ki = 7750 nM
191.139 C6 H9 N O6 [C@@H...
View in 3D viewer
90% Homology Family
Leader
PDB id Resolution Class Description Source Keywords
3LPF 2.26 Å EC: 3.2.1.31 STRUCTURE OF E. COLI BETA-GLUCURONIDASE BOUND WITH A NOVEL, INHIBITOR 1-((6,7-DIMETHYL-2-OXO-1,2-DIHYDROQUINOLIN-3-YL)M( 2-HYDROXYETHYL)-3-(3-METHOXYPHENYL)THIOUREA ESCHERICHIA COLI ALPHA/BETA BARREL SUGAR-BINDING DOMAIN BETA-SANDWICH DOMAIGLYCOSYL HYDROLASE BETA-GLUCURONIDASE INHIBITOR GLYCOSIDAHYDROLASE HYDROLASE-HYDROLASE INHIBITOR COMPLEX
Ref.: ALLEVIATING CANCER DRUG TOXICITY BY INHIBITING A BA ENZYME. SCIENCE V. 330 831 2010
Members (3)
No: PDB id Binding Data Representative ligand Formula Smiles
The Class containing this family consists of a total of 4 families.
1 3K4D Ki = 7750 nM EVA C6 H9 N O6 [C@@H]1([C....
2 5CZK Ki = 1.9 uM 57Z C21 H23 N3 O3 S Cc1cc(c2c(....
3 3LPF Ki = 208 nM Z77 C22 H25 N3 O3 S Cc1cc2c(cc....
70% Homology Family (3)
No: PDB id Binding Data Representative ligand Formula Smiles
The Class containing this family consists of a total of 4 families.
1 3K4D Ki = 7750 nM EVA C6 H9 N O6 [C@@H]1([C....
2 5CZK Ki = 1.9 uM 57Z C21 H23 N3 O3 S Cc1cc(c2c(....
3 3LPF Ki = 208 nM Z77 C22 H25 N3 O3 S Cc1cc2c(cc....
50% Homology Family (10)
No: PDB id Binding Data Representative ligand Formula Smiles
The Class containing this family consists of a total of 214 families.
1 3K4D Ki = 7750 nM EVA C6 H9 N O6 [C@@H]1([C....
2 5CZK Ki = 1.9 uM 57Z C21 H23 N3 O3 S Cc1cc(c2c(....
3 3LPF Ki = 208 nM Z77 C22 H25 N3 O3 S Cc1cc2c(cc....
4 6JZ5 - BDP C6 H10 O7 [C@@H]1([C....
5 6JZ7 - CKU C9 H17 N O4 CCCN1C[C@@....
6 6JZ3 - CN0 C6 H11 N O5 C1[C@@H]([....
7 6JZ4 - EVA C6 H9 N O6 [C@@H]1([C....
8 6JZ6 - CKX C9 H17 N O4 CCC[C@H]1[....
9 6JZ8 - GCB C6 H8 O7 [C@@H]1([C....
10 6JZ2 - SJ5 C6 H11 N O4 C1[C@@H]([....
Polypharmacology
Similar Ligands (2D)
Ligand no: 1; Ligand: EVA; Similar ligands found: 1
No: Ligand ECFP6 Tc MDL keys Tc
1 EVA 1 1
Similar Ligands (3D)
Ligand no: 1; Ligand: EVA; Similar ligands found: 1138
No: Ligand Similarity coefficient
1 BDP 1.0000
2 GCB 1.0000
3 15L 1.0000
4 GCU 0.9971
5 BGC 0.9854
6 LGC 0.9787
7 GLC 0.9775
8 SHG 0.9747
9 IJZ 0.9741
10 GAL 0.9741
11 G3F 0.9740
12 GCS 0.9719
13 FOT 0.9699
14 SYA 0.9698
15 GCW 0.9695
16 GTR 0.9687
17 4AA 0.9685
18 DHK 0.9670
19 Q6T 0.9652
20 9PY 0.9652
21 5WY 0.9651
22 CN0 0.9647
23 AKH 0.9634
24 HJP 0.9617
25 C2U 0.9607
26 4XV 0.9596
27 BNT 0.9587
28 42C 0.9581
29 KBG 0.9579
30 GDE 0.9579
31 ASO 0.9574
32 JTH 0.9568
33 8S0 0.9560
34 4Z4 0.9552
35 E7Z 0.9545
36 CFF 0.9545
37 8XQ 0.9541
38 4XS 0.9538
39 PFB 0.9523
40 3IT 0.9521
41 3MG 0.9511
42 L7T 0.9500
43 0P6 0.9497
44 5NE 0.9496
45 KGK 0.9488
46 QSH 0.9485
47 HKD 0.9481
48 94B 0.9478
49 7ZE 0.9476
50 IFL 0.9473
51 GLT 0.9469
52 HQD 0.9466
53 ICO 0.9462
54 SOE 0.9457
55 23J 0.9456
56 149 0.9454
57 GOG 0.9451
58 TTY 0.9451
59 NOJ 0.9450
60 FE DB1 0.9450
61 3F0 0.9449
62 DBH 0.9448
63 3M0 0.9441
64 GOX 0.9439
65 ADA 0.9437
66 3HA 0.9437
67 DIU 0.9435
68 GTQ 0.9433
69 ALL 0.9431
70 K3Q 0.9431
71 8GK 0.9430
72 948 0.9427
73 HNQ 0.9425
74 57O 0.9424
75 FGZ 0.9421
76 1GN 0.9420
77 5RG 0.9420
78 PA1 0.9418
79 GCV 0.9416
80 2FG 0.9415
81 LKA 0.9415
82 5QX 0.9415
83 QPR 0.9413
84 9MG 0.9411
85 INE 0.9410
86 9TZ 0.9409
87 NOY 0.9405
88 KFH 0.9403
89 BMA 0.9401
90 AZ9 0.9400
91 DPZ 0.9393
92 DOR 0.9390
93 G5V 0.9389
94 G2F 0.9387
95 3Z8 0.9387
96 UFV 0.9383
97 6CS 0.9382
98 82I 0.9381
99 60Q 0.9376
100 APZ 0.9376
101 ORO 0.9374
102 3WA 0.9374
103 2H5 0.9373
104 5RN 0.9373
105 5NS 0.9372
106 DOB 0.9367
107 SJ5 0.9367
108 FA0 0.9364
109 YIO 0.9363
110 BHA 0.9363
111 D1X 0.9363
112 PXL 0.9361
113 4NC 0.9358
114 SKM 0.9357
115 5M0 0.9354
116 4ME 0.9353
117 8CM 0.9353
118 3DO 0.9352
119 LCN 0.9350
120 4M0 0.9350
121 9KH 0.9349
122 A7W 0.9348
123 TEP 0.9346
124 MAN 0.9345
125 DQA 0.9344
126 25W 0.9343
127 Q88 0.9340
128 OA3 0.9339
129 ES0 0.9337
130 5MK 0.9336
131 UNC 0.9335
132 MO8 0.9335
133 GLF 0.9334
134 54G 0.9334
135 K5W 0.9333
136 CWS 0.9331
137 KUF 0.9327
138 TTL 0.9327
139 KT7 0.9325
140 CWM 0.9319
141 7NI 0.9318
142 6XI 0.9312
143 NID 0.9310
144 XX2 0.9309
145 WOO 0.9308
146 GLA 0.9308
147 DIN 0.9307
148 M2K 0.9303
149 2ZQ 0.9301
150 GIV 0.9301
151 5CU 0.9299
152 IPB 0.9299
153 2D0 0.9299
154 0N7 0.9298
155 BK9 0.9296
156 HXX 0.9293
157 M0Q 0.9293
158 XXR 0.9293
159 DHB 0.9291
160 VNL 0.9291
161 5RO 0.9290
162 12Q 0.9286
163 92K 0.9285
164 FA3 0.9284
165 1LQ 0.9284
166 M1E 0.9283
167 CLZ 0.9282
168 KJY 0.9281
169 AFR 0.9279
170 KJH 0.9279
171 DBJ 0.9276
172 091 0.9276
173 LZ2 0.9275
174 VK3 0.9274
175 IV2 0.9270
176 NTM 0.9266
177 LT2 0.9262
178 OXC 0.9262
179 7WR 0.9260
180 4HC 0.9260
181 NTZ 0.9259
182 Z5P 0.9259
183 BEA 0.9258
184 I3A 0.9256
185 ZWZ 0.9255
186 2CZ 0.9254
187 34D 0.9254
188 X09 0.9253
189 B60 0.9250
190 M0W 0.9250
191 MHK 0.9245
192 7VS 0.9245
193 URC 0.9244
194 PYQ 0.9242
195 G6D 0.9241
196 DBX 0.9239
197 F5B 0.9238
198 B57 0.9238
199 R8V 0.9236
200 NDM 0.9235
201 209 0.9234
202 2KA 0.9234
203 GRE 0.9234
204 HLZ 0.9231
205 X6X 0.9228
206 67N 0.9224
207 GAF 0.9223
208 SX1 0.9223
209 EMZ 0.9222
210 UEG 0.9222
211 M1Q 0.9222
212 SOR 0.9221
213 12B 0.9219
214 KYA 0.9219
215 86J 0.9218
216 HQT 0.9217
217 O2A 0.9216
218 PXM 0.9215
219 0FK 0.9214
220 MWP 0.9213
221 6F0 0.9213
222 FLV 0.9213
223 GXL 0.9212
224 MAQ 0.9212
225 C2Y 0.9212
226 FA6 0.9211
227 AIN 0.9209
228 7HQ 0.9209
229 IPZ 0.9209
230 MRW 0.9206
231 KBB 0.9205
232 8WT 0.9205
233 61M 0.9204
234 XAN 0.9204
235 8W9 0.9201
236 SWA 0.9201
237 TOF 0.9200
238 N8Y 0.9199
239 6M1 0.9199
240 LZM 0.9198
241 FBU 0.9197
242 NVU 0.9196
243 RPQ 0.9196
244 6M4 0.9194
245 7W1 0.9193
246 QIC 0.9192
247 INO 0.9191
248 DNA 0.9190
249 DQN 0.9190
250 3FH 0.9189
251 39A 0.9188
252 COU 0.9188
253 93K 0.9186
254 UFO 0.9185
255 4MU 0.9184
256 MBG 0.9183
257 JBQ 0.9183
258 AW5 0.9183
259 FHN 0.9182
260 H33 0.9182
261 YSO 0.9182
262 P9P 0.9182
263 UAN 0.9181
264 JKZ 0.9181
265 KLW 0.9181
266 JBK 0.9181
267 IFP 0.9181
268 5WX 0.9177
269 EXO 0.9176
270 DNF 0.9176
271 MA3 0.9175
272 ISE 0.9172
273 G1O 0.9170
274 A13 0.9169
275 J9W 0.9169
276 JND 0.9168
277 23A 0.9167
278 RXA 0.9167
279 X0V 0.9165
280 AZ8 0.9165
281 TSR 0.9164
282 DEE 0.9164
283 M1A 0.9163
284 R9S 0.9161
285 EYK 0.9161
286 329 0.9160
287 MJ2 0.9160
288 UQ 0.9159
289 42A 0.9159
290 9DG 0.9157
291 0LH 0.9155
292 K17 0.9155
293 5NU 0.9154
294 GTL 0.9153
295 PE0 0.9153
296 NQ 0.9153
297 FBV 0.9153
298 2LY 0.9153
299 MYJ 0.9153
300 5IQ 0.9152
301 MNM 0.9151
302 FBT 0.9151
303 1P7 0.9150
304 PHT 0.9150
305 5SG 0.9150
306 P3K 0.9149
307 SHA 0.9149
308 ZB1 0.9147
309 1X7 0.9147
310 MT5 0.9147
311 KIB 0.9147
312 DGJ 0.9143
313 KJ5 0.9143
314 MIG 0.9142
315 2EC 0.9141
316 F12 0.9138
317 GLG 0.9137
318 7D2 0.9135
319 MUA 0.9135
320 JKE 0.9135
321 EJZ 0.9134
322 LSA 0.9133
323 8TX 0.9133
324 MT0 0.9132
325 9TW 0.9132
326 173 0.9132
327 5CL 0.9131
328 CHB 0.9131
329 Q7A 0.9131
330 1SQ 0.9130
331 INS 0.9130
332 AJ2 0.9129
333 TFU 0.9129
334 680 0.9128
335 N5J 0.9128
336 KIA 0.9127
337 BDF 0.9126
338 1NP 0.9126
339 F31 0.9125
340 JPZ 0.9125
341 JBH 0.9125
342 2HO 0.9125
343 7B4 0.9125
344 G4D 0.9124
345 GYP 0.9124
346 LYL 0.9123
347 LNR 0.9123
348 ES1 0.9123
349 4YS 0.9122
350 5NI 0.9121
351 ODO 0.9121
352 JB5 0.9121
353 6VD 0.9120
354 AMG 0.9119
355 HHA 0.9119
356 495 0.9119
357 SAL 0.9119
358 EUG 0.9118
359 4M4 0.9118
360 DFB 0.9117
361 V55 0.9117
362 Q24 0.9117
363 2HQ 0.9115
364 HQY 0.9115
365 PDC 0.9114
366 IFM 0.9113
367 SKA 0.9113
368 LDP 0.9112
369 FH2 0.9111
370 1LM 0.9111
371 0JD 0.9110
372 8H8 0.9110
373 7B3 0.9110
374 O72 0.9109
375 QM1 0.9109
376 24W 0.9108
377 QX4 0.9108
378 5Q0 0.9107
379 4FS 0.9106
380 FDK 0.9103
381 HA5 0.9103
382 BE2 0.9103
383 ES5 0.9102
384 FUL 0.9102
385 HPT 0.9101
386 AQO 0.9100
387 FYU 0.9100
388 AZF 0.9099
389 FBG 0.9099
390 5WV 0.9099
391 FDB 0.9098
392 OCH 0.9098
393 M1H 0.9097
394 3U4 0.9095
395 XQG 0.9094
396 DMJ 0.9094
397 0HO 0.9092
398 5XC 0.9091
399 7MH 0.9091
400 RAT 0.9090
401 7ME 0.9090
402 7VJ 0.9090
403 M4E 0.9089
404 VNJ 0.9088
405 3HB 0.9088
406 F0J 0.9087
407 M6N 0.9087
408 4TU 0.9086
409 2ZM 0.9085
410 95Z 0.9085
411 NBG 0.9084
412 2AQ 0.9084
413 03V 0.9083
414 T6C 0.9083
415 CTS 0.9082
416 EKZ 0.9080
417 AJV 0.9080
418 3PF 0.9079
419 3RI 0.9077
420 3SK 0.9077
421 QSB 0.9077
422 JLZ 0.9076
423 B62 0.9074
424 IHB 0.9074
425 ZXD 0.9073
426 L99 0.9073
427 ISN 0.9073
428 GUN 0.9073
429 RM1 0.9071
430 GJS 0.9070
431 2CL 0.9070
432 DHQ 0.9069
433 BCF 0.9068
434 37T 0.9068
435 M5K 0.9066
436 4JQ 0.9066
437 97T 0.9066
438 28N 0.9066
439 S76 0.9064
440 GM7 0.9063
441 8OZ 0.9063
442 BZ3 0.9062
443 PCI 0.9061
444 H5B 0.9060
445 4CS 0.9060
446 4SV 0.9059
447 OHP 0.9059
448 KTA 0.9058
449 JUG 0.9058
450 4FH 0.9058
451 3A9 0.9058
452 ES6 0.9058
453 0HN 0.9058
454 HZQ 0.9057
455 PRZ 0.9057
456 OXZ 0.9056
457 GCO 0.9054
458 8WO 0.9054
459 K2P 0.9052
460 SXS 0.9052
461 ES7 0.9052
462 J9Q 0.9048
463 GIM 0.9048
464 IF7 0.9047
465 293 0.9046
466 BBF 0.9046
467 FHB 0.9046
468 DNC 0.9046
469 BTE 0.9045
470 2FY 0.9044
471 AZA 0.9044
472 ASC 0.9043
473 XAZ 0.9043
474 HMU 0.9043
475 ADZ 0.9042
476 GV9 0.9041
477 HFB 0.9041
478 92P 0.9041
479 MEW 0.9040
480 NNO 0.9040
481 IBF 0.9040
482 6OT 0.9040
483 QBK 0.9040
484 EA1 0.9036
485 QX2 0.9036
486 EGR 0.9035
487 8ZE 0.9033
488 SVD 0.9033
489 I6G 0.9033
490 TVP 0.9032
491 DQU 0.9031
492 0FN 0.9031
493 3NT 0.9031
494 MS9 0.9029
495 4A3 0.9029
496 6AP 0.9028
497 HPA 0.9028
498 3NY 0.9027
499 5WU 0.9025
500 9KT 0.9025
501 6ME 0.9024
502 B53 0.9022
503 R9Y 0.9022
504 P84 0.9022
505 5QY 0.9022
506 9FL 0.9022
507 SR4 0.9021
508 N3W 0.9021
509 3HM 0.9021
510 FB1 0.9021
511 3R6 0.9020
512 226 0.9020
513 XHP 0.9020
514 3RK 0.9020
515 SRO 0.9020
516 06B 0.9020
517 H42 0.9019
518 4XH 0.9019
519 RMN 0.9018
520 IGA 0.9018
521 32X 0.9018
522 D07 0.9017
523 HH8 0.9017
524 75K 0.9016
525 GXY 0.9015
526 4HM 0.9015
527 4SX 0.9015
528 2AK 0.9014
529 JXZ 0.9014
530 6NT 0.9014
531 0W8 0.9013
532 5OB 0.9013
533 1KH 0.9013
534 1XN 0.9012
535 DRL 0.9011
536 HMH 0.9011
537 AY4 0.9011
538 PHH 0.9010
539 LI6 0.9008
540 QWW 0.9008
541 1F1 0.9008
542 A2F 0.9007
543 290 0.9004
544 QAS 0.9004
545 4P0 0.9003
546 X05 0.9003
547 141 0.9002
548 GZ8 0.9002
549 HH5 0.9002
550 M5N 0.9000
551 H6B 0.8999
552 2AL 0.8999
553 LXC 0.8999
554 KKN 0.8998
555 NCD 0.8996
556 PFL 0.8996
557 IBM 0.8996
558 K32 0.8996
559 ABV 0.8995
560 261 0.8995
561 HDL 0.8994
562 BCU 0.8994
563 BTY 0.8993
564 FP1 0.8993
565 F05 0.8993
566 TSS 0.8992
567 6GU 0.8992
568 GJP 0.8992
569 QAT 0.8991
570 HIO 0.8991
571 AEZ 0.8990
572 44V 0.8989
573 8HC 0.8988
574 24B 0.8987
575 7HP 0.8987
576 BZX 0.8985
577 GT0 0.8984
578 RAM 0.8984
579 FA1 0.8983
580 YH7 0.8983
581 MVL 0.8982
582 D3M 0.8981
583 HX3 0.8981
584 61O 0.8980
585 FRU 0.8980
586 F3B 0.8979
587 M3S 0.8978
588 NAG 0.8978
589 IP0 0.8978
590 5JQ 0.8977
591 AS3 0.8977
592 1P3 0.8977
593 7WV 0.8976
594 TAG 0.8975
595 XQ0 0.8974
596 MQN 0.8974
597 OTW 0.8973
598 44W 0.8973
599 FDR 0.8973
600 DHY 0.8973
601 2A7 0.8972
602 15N 0.8972
603 3OC 0.8972
604 XX3 0.8971
605 1WD 0.8971
606 PEY 0.8970
607 HTP 0.8970
608 CBF 0.8969
609 EV0 0.8969
610 4RU 0.8969
611 3C1 0.8969
612 MFB 0.8969
613 1DW 0.8968
614 JDN 0.8968
615 GAB 0.8968
616 H7Y 0.8967
617 4ZC 0.8967
618 0FO 0.8967
619 KOJ 0.8967
620 JXW 0.8967
621 HA7 0.8966
622 JXN 0.8966
623 53C 0.8965
624 ESI 0.8965
625 IOS 0.8964
626 RHU 0.8964
627 FUC 0.8963
628 MR1 0.8962
629 ADE 0.8962
630 B55 0.8961
631 4KL 0.8961
632 0F9 0.8961
633 NSP 0.8960
634 6AI 0.8960
635 RNS 0.8958
636 TQU 0.8958
637 27B 0.8956
638 4YO 0.8956
639 MMA 0.8956
640 3Z7 0.8955
641 3MB 0.8955
642 NGO 0.8954
643 10L 0.8954
644 HHR 0.8953
645 PH2 0.8953
646 6R8 0.8952
647 MT8 0.8952
648 TBS 0.8951
649 7CT 0.8951
650 LDR 0.8951
651 FXH 0.8951
652 N2Z 0.8950
653 G3E 0.8950
654 ICT 0.8949
655 AZG 0.8949
656 YQA 0.8948
657 51R 0.8948
658 BOA 0.8948
659 OMD 0.8947
660 1HN 0.8946
661 CFP 0.8946
662 S3B 0.8945
663 I1N 0.8945
664 ADK 0.8944
665 PQ0 0.8944
666 FCB 0.8942
667 2ZV 0.8942
668 BSP 0.8942
669 APS 0.8942
670 T9G 0.8941
671 F1A 0.8941
672 GC2 0.8941
673 OVV 0.8941
674 NLA 0.8939
675 ZVO 0.8939
676 NDH 0.8938
677 FUF 0.8938
678 ZZ8 0.8936
679 ZZT 0.8936
680 8WQ 0.8934
681 7W4 0.8934
682 C9E 0.8934
683 DX4 0.8934
684 F81 0.8934
685 MVN 0.8933
686 XYP 0.8933
687 SYR 0.8932
688 1XA 0.8932
689 PHB 0.8932
690 E7R 0.8931
691 1XM 0.8931
692 9AP 0.8931
693 XQK 0.8931
694 MSN 0.8930
695 0CU 0.8930
696 0R0 0.8928
697 6M9 0.8928
698 AC6 0.8928
699 KJU 0.8928
700 3DM 0.8927
701 JR2 0.8926
702 TBP 0.8926
703 IPM 0.8924
704 14O 0.8924
705 4JT 0.8924
706 NPO 0.8924
707 VOH 0.8923
708 3MA 0.8923
709 2MN 0.8921
710 CTL 0.8921
711 52C 0.8921
712 2HU 0.8920
713 3GQ 0.8920
714 MZB 0.8920
715 FBB 0.8919
716 NMJ 0.8919
717 8IG 0.8918
718 9ZE 0.8917
719 270 0.8916
720 AX7 0.8916
721 0TU 0.8916
722 KTW 0.8916
723 PRF 0.8916
724 PD2 0.8915
725 5VL 0.8915
726 3C2 0.8914
727 35C 0.8914
728 39O 0.8914
729 9FE 0.8914
730 0W1 0.8914
731 M6Z 0.8913
732 1AL 0.8911
733 SRT 0.8911
734 67X 0.8911
735 ARP 0.8911
736 URQ 0.8910
737 SYV 0.8910
738 1WG 0.8908
739 2BG 0.8908
740 GLO 0.8907
741 GIO 0.8907
742 N2I 0.8905
743 BP1 0.8905
744 SYG 0.8905
745 GTZ 0.8903
746 5B1 0.8903
747 2FQ 0.8902
748 F60 0.8901
749 2LP 0.8900
750 9EW 0.8899
751 5H1 0.8898
752 JYB 0.8897
753 2A9 0.8896
754 ET2 0.8896
755 LT8 0.8894
756 9DA 0.8894
757 X8D 0.8893
758 ZZ3 0.8892
759 GOO 0.8891
760 XXG 0.8891
761 BRV 0.8891
762 3ID 0.8891
763 0RW 0.8890
764 9HX 0.8890
765 PAB 0.8889
766 2MI 0.8887
767 ONR 0.8887
768 1U6 0.8886
769 K22 0.8886
770 5MI 0.8886
771 ABI 0.8885
772 5MB 0.8885
773 F9Y 0.8884
774 EPR 0.8884
775 5JL 0.8882
776 G12 0.8882
777 DIG 0.8882
778 7MX 0.8881
779 7WA 0.8881
780 GYE 0.8881
781 SE2 0.8880
782 BCP 0.8878
783 XCZ 0.8877
784 Q02 0.8876
785 6BL 0.8873
786 XM0 0.8873
787 3XX 0.8872
788 PZI 0.8871
789 DIE 0.8871
790 VXX 0.8870
791 AHR 0.8870
792 TH7 0.8870
793 64C 0.8870
794 NGT 0.8869
795 DX3 0.8869
796 6FZ 0.8868
797 J5I 0.8868
798 XXP 0.8867
799 JAW 0.8867
800 TGX 0.8866
801 HMQ 0.8864
802 JFD 0.8862
803 BSX 0.8862
804 JBE 0.8862
805 A29 0.8862
806 EDR 0.8861
807 6MP 0.8858
808 2CK 0.8857
809 2K4 0.8856
810 1KP 0.8856
811 2CQ 0.8855
812 5OF 0.8851
813 K2T 0.8851
814 QY9 0.8850
815 HBD 0.8850
816 LAO 0.8849
817 FCR 0.8848
818 RIB 0.8847
819 ES9 0.8846
820 6NI 0.8845
821 AX3 0.8843
822 QUZ 0.8841
823 5GU 0.8840
824 BZJ 0.8839
825 RM4 0.8839
826 EOL 0.8838
827 CKU 0.8837
828 9R5 0.8836
829 SWD 0.8835
830 DHS 0.8834
831 SF9 0.8833
832 FBW 0.8831
833 NK 0.8831
834 CLW 0.8831
835 PM6 0.8830
836 4XR 0.8829
837 TWO 0.8828
838 3BZ 0.8828
839 1Y6 0.8825
840 HHT 0.8824
841 EQT 0.8823
842 1LN 0.8823
843 DMD 0.8820
844 OW4 0.8819
845 NK2 0.8818
846 ZZ2 0.8817
847 XIY 0.8817
848 B2J 0.8816
849 54X 0.8816
850 EXD 0.8815
851 PX7 0.8813
852 4MA 0.8813
853 OVM 0.8812
854 289 0.8811
855 68A 0.8811
856 NGW 0.8810
857 JIF 0.8810
858 QMS 0.8809
859 505 0.8809
860 DC5 0.8809
861 I3C 0.8809
862 HBA 0.8809
863 JFJ 0.8808
864 ES2 0.8808
865 ZYR 0.8808
866 WCE 0.8808
867 1P8 0.8806
868 ARB 0.8805
869 2GS 0.8803
870 2C2 0.8803
871 JZ3 0.8803
872 NOK 0.8802
873 8GC 0.8802
874 TLA 0.8801
875 MFU 0.8801
876 TSU 0.8801
877 15E 0.8801
878 ENL 0.8800
879 42J 0.8799
880 1WC 0.8799
881 XYS 0.8797
882 2O6 0.8796
883 CIT 0.8795
884 150 0.8795
885 PBZ 0.8795
886 717 0.8794
887 3AB 0.8794
888 7N0 0.8793
889 FX1 0.8793
890 D48 0.8793
891 4P5 0.8793
892 6DP 0.8791
893 0GZ 0.8791
894 OTD 0.8791
895 NFQ 0.8790
896 OTR 0.8790
897 ALA PRO 0.8789
898 PQK 0.8789
899 NDG 0.8788
900 45C 0.8788
901 GNM 0.8788
902 39U 0.8787
903 G1P 0.8787
904 CKX 0.8784
905 MIC 0.8783
906 IAC 0.8783
907 MAJ 0.8781
908 M3Q 0.8780
909 CIP 0.8779
910 P72 0.8779
911 Z82 0.8779
912 790 0.8778
913 2D3 0.8778
914 1M2 0.8777
915 12M 0.8777
916 URF 0.8777
917 MQB 0.8776
918 069 0.8775
919 H62 0.8774
920 CDV 0.8773
921 94W 0.8773
922 JB8 0.8771
923 HQJ 0.8771
924 TRC 0.8769
925 8XL 0.8769
926 KP6 0.8768
927 Q71 0.8768
928 TIU 0.8768
929 5VJ 0.8767
930 GL1 0.8764
931 II6 0.8764
932 FLC 0.8764
933 NPY 0.8762
934 1FF 0.8761
935 ISZ 0.8761
936 GLS 0.8760
937 L3Q 0.8759
938 SVN 0.8758
939 3C7 0.8757
940 GLY PRO 0.8757
941 FCA 0.8756
942 TC7 0.8755
943 8NX 0.8755
944 7A2 0.8754
945 HLD 0.8754
946 3SL 0.8753
947 8G0 0.8752
948 582 0.8751
949 GZL 0.8751
950 APG 0.8750
951 286 0.8749
952 BZ2 0.8748
953 PBA 0.8748
954 1IT 0.8747
955 BHO 0.8747
956 6X9 0.8746
957 9RW 0.8745
958 R8A 0.8745
959 45L 0.8745
960 S7B 0.8744
961 J9T 0.8743
962 SMN 0.8740
963 2TQ 0.8740
964 REL 0.8739
965 A2G 0.8739
966 FBS 0.8738
967 X8Z 0.8737
968 WBU 0.8736
969 BPU 0.8736
970 NIZ 0.8735
971 MCT 0.8734
972 PRY 0.8730
973 SAN 0.8730
974 AMS 0.8730
975 AAS 0.8730
976 GDL 0.8728
977 4J8 0.8727
978 7I2 0.8723
979 5HN 0.8723
980 0XT 0.8723
981 5FN 0.8722
982 CH9 0.8721
983 A9P 0.8719
984 V1T 0.8719
985 SW7 0.8719
986 CFI 0.8718
987 IPT 0.8717
988 GZQ 0.8717
989 MCO 0.8716
990 KYD 0.8716
991 XFE 0.8714
992 5DI 0.8713
993 BEN 0.8713
994 PJW 0.8712
995 449 0.8712
996 4NG 0.8711
997 20J 0.8711
998 2XX 0.8707
999 SLC 0.8707
1000 XUL 0.8706
1001 SFU 0.8706
1002 BEZ 0.8706
1003 CWJ 0.8701
1004 JZ4 0.8700
1005 3AL 0.8700
1006 12T 0.8700
1007 XYL 0.8700
1008 W8G 0.8699
1009 E35 0.8698
1010 I4D 0.8696
1011 HDH 0.8696
1012 1U1 0.8696
1013 HHS 0.8688
1014 ZZZ 0.8687
1015 7FF 0.8687
1016 2PG 0.8684
1017 L1Q 0.8684
1018 GL4 0.8682
1019 AMH 0.8681
1020 ICB 0.8681
1021 HBO 0.8681
1022 L5V 0.8681
1023 6LW 0.8680
1024 GIF 0.8680
1025 FEH 0.8679
1026 FSW 0.8678
1027 3R9 0.8677
1028 IPD 0.8676
1029 ES4 0.8675
1030 AJY 0.8675
1031 JG8 0.8674
1032 6PC 0.8673
1033 TRA 0.8672
1034 NGA 0.8671
1035 SDD 0.8671
1036 260 0.8669
1037 BNS 0.8668
1038 0MK 0.8667
1039 KIF 0.8665
1040 BPY 0.8664
1041 PSV 0.8663
1042 E3D 0.8661
1043 CKA 0.8661
1044 PYD 0.8660
1045 ROI 0.8660
1046 GNL 0.8659
1047 K6X 0.8659
1048 A9O 0.8658
1049 Q77 0.8658
1050 F6P 0.8657
1051 LRH 0.8657
1052 TT4 0.8657
1053 6KT 0.8656
1054 FAN 0.8654
1055 RSO 0.8653
1056 S0G 0.8652
1057 E5X 0.8652
1058 GVG 0.8652
1059 2K8 0.8652
1060 4VP 0.8651
1061 9CA 0.8651
1062 PYG 0.8649
1063 B0D 0.8646
1064 ARW 0.8646
1065 PBC 0.8641
1066 V6F 0.8641
1067 H76 0.8639
1068 MIF 0.8637
1069 NCA 0.8635
1070 3CU 0.8634
1071 B5D 0.8634
1072 SQ7 0.8633
1073 SER PRO 0.8630
1074 GSY 0.8630
1075 CFA 0.8629
1076 MXN 0.8628
1077 GJZ 0.8628
1078 7MU 0.8627
1079 BAM 0.8627
1080 SBI 0.8623
1081 SF6 0.8623
1082 RJY 0.8620
1083 OVP 0.8620
1084 3C4 0.8620
1085 FBM 0.8620
1086 7A3 0.8620
1087 AUD 0.8619
1088 RIP 0.8617
1089 RB5 0.8614
1090 DFU 0.8614
1091 3TJ 0.8614
1092 9GP 0.8614
1093 FIX 0.8613
1094 1A7 0.8613
1095 PAC 0.8611
1096 TIY 0.8610
1097 ANN 0.8609
1098 FUD 0.8608
1099 36E 0.8608
1100 TZE 0.8607
1101 NCT 0.8606
1102 CCV 0.8604
1103 BPS 0.8602
1104 CXF 0.8601
1105 BM3 0.8595
1106 PEZ 0.8595
1107 826 0.8594
1108 4TE 0.8594
1109 JF2 0.8592
1110 PZA 0.8591
1111 UNU 0.8590
1112 NIO 0.8590
1113 2SX 0.8585
1114 BRT 0.8585
1115 TYL 0.8583
1116 MXX 0.8582
1117 HLR 0.8579
1118 QSC 0.8579
1119 GF4 0.8575
1120 ROR 0.8570
1121 4NM 0.8569
1122 428 0.8567
1123 ESP 0.8567
1124 CGB 0.8561
1125 4WL 0.8559
1126 F9P 0.8559
1127 LIP 0.8559
1128 GAG 0.8558
1129 ST2 0.8557
1130 VC2 0.8557
1131 KDF 0.8556
1132 1Z8 0.8554
1133 9BF 0.8552
1134 PBR 0.8550
1135 6UA 0.8546
1136 YCP 0.8545
1137 NPA 0.8511
1138 RH1 0.8510
Similar Binding Sites (Proteins are less than 50% similar to leader)
Pocket No.: 1; Query (leader) PDB : 3LPF; Ligand: Z77; Similar sites found with APoc: No similar binding sites found, or similarity not calculated due to duplicate pocket.
This union binding pocket(no: 1) in the query (biounit: 3lpf.bio1) has 28 residues
No: Leader PDB Ligand Sequence Similarity
Pocket No.: 2; Query (leader) PDB : 3LPF; Ligand: Z77; Similar sites found with APoc: No similar binding sites found, or similarity not calculated due to duplicate pocket.
This union binding pocket(no: 2) in the query (biounit: 3lpf.bio1) has 28 residues
No: Leader PDB Ligand Sequence Similarity
Pocket No.: 3; Query (leader) PDB : 3LPF; Ligand: Z77; Similar sites found with APoc: No similar binding sites found, or similarity not calculated due to duplicate pocket.
This union binding pocket(no: 3) in the query (biounit: 3lpf.bio1) has 28 residues
No: Leader PDB Ligand Sequence Similarity
Pocket No.: 4; Query (leader) PDB : 3LPF; Ligand: Z77; Similar sites found with APoc: No similar binding sites found, or similarity not calculated due to duplicate pocket.
This union binding pocket(no: 4) in the query (biounit: 3lpf.bio1) has 28 residues
No: Leader PDB Ligand Sequence Similarity
APoc FAQ
Feedback