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- PDB : .ZIP | .CSV
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- Class : .ZIP | .CSV
No: | PDB id | Binding Data | Representative ligand | Formula | Smiles |
---|---|---|---|---|---|
The Class containing this family consists of a total of 1 families. | |||||
1 | 1E81 | - | M91 | C34 H49 N5 O6 S | CSC[C@@H](.... |
2 | 4ZEA | - | IMI | C10 H17 N3 O2 S | C1[C@H]2[C.... |
3 | 3ER3 | Ki = 81 nM | 0EL | C51 H78 N8 O9 | NULL |
4 | 4Y4D | - | CFF | C8 H10 N4 O2 | Cn1cnc2c1C.... |
5 | 5LWT | - | 7B3 | C10 H13 N3 O | Cc1c2cnnc(.... |
6 | 1EPM | - | THR PHE GLN ALA PSA LEU ARG GLU | n/a | n/a |
7 | 1EED | Ki = 16.2 uM | 0EO | C34 H55 N3 O8 | CC(C)C[C@@.... |
8 | 3PMY | - | 41L | C15 H13 N3 O | c1ccc(cc1).... |
9 | 1OEX | - | BOC HIS PRO PHE ALA LOV ILE HIS | n/a | n/a |
10 | 4ER4 | Ki = 160 nM | PRO HIS PRO PHE HIS LAV ILE HIS LYS | n/a | n/a |
11 | 4LBT | Ki = 6 uM | 1TZ | C21 H24 N4 O | Cc1cc(c(c(.... |
12 | 3PWW | - | ROC | C38 H50 N6 O5 | CC(C)(C)NC.... |
13 | 4Y38 | Kd = 4 mM | 0A9 | C10 H13 N O2 | COC(=O)[C@.... |
14 | 2JJJ | - | 0QS | C36 H56 F2 N7 O8 S | CC(C)(C)S(.... |
15 | 1GVV | - | 0GM | C51 H61 N5 O6 | CC(C)C[C@H.... |
16 | 3PMU | - | F7L | C14 H20 F N O2 | c1ccc(c(c1.... |
17 | 5OJE | Ki = 6.1 uM | VSK | C22 H27 N3 O | Cc1cc(c(c(.... |
18 | 1GVT | - | 2ZS | C31 H48 N4 O7 S | CC(C)OC(=O.... |
19 | 1EPR | - | 0QS | C36 H56 F2 N7 O8 S | CC(C)(C)S(.... |
20 | 5MB5 | - | 46P | C8 H10 N4 S | Cc1c(sc(n1.... |
21 | 5MB7 | - | 4AV | C8 H9 Cl N2 O2 | CNCc1cc(cc.... |
22 | 4Y4G | - | GGB | C5 H12 N4 O3 | [H]/N=C(N).... |
23 | 3ER5 | Ki = 1 nM | PRO HIS PRO PHE HIS STA VAL ILE HIS LYS | n/a | n/a |
24 | 3URL | - | HIS SER LEU PHE HIS PUK THR PRO | n/a | n/a |
25 | 3PCZ | - | BAM | C7 H9 N2 | c1ccc(cc1).... |
26 | 2V00 | Kd = 0.22 mM | V15 | C12 H13 N3 O | c1ccc(cc1).... |
27 | 5LWR | - | 7B2 | C27 H29 Cl N9 O | Cc1c2cnn3c.... |
28 | 3PLL | - | F06 | C8 H9 Cl N2 S | [H]/N=C(N).... |
29 | 4ER2 | Ki = 0.5 nM | IVA VAL VAL STA ALA STA | n/a | n/a |
30 | 4LP9 | ic50 = 0.62 uM | SER LEU PHE HIS 22G THR PRO | n/a | n/a |
31 | 3PRS | - | RIT | C37 H48 N6 O5 S2 | CC(C)c1nc(.... |
32 | 1ENT | Ki = 110 nM | 0EM | C32 H52 N6 O7 P | NULL |
33 | 1E80 | - | 0GQ | C41 H64 N10 O6 | CC[C@H](C).... |
34 | 5LWS | - | 7B2 | C27 H29 Cl N9 O | Cc1c2cnn3c.... |
35 | 3PBD | - | F05 | C8 H8 N2 | c1ccc2c(c1.... |
36 | 1OD1 | - | 0QS | C36 H56 F2 N7 O8 S | CC(C)(C)S(.... |
37 | 3WZ6 | Ki = 1.1 uM | IXZ | C27 H25 N3 O2 S | c1ccc(cc1).... |
38 | 5ER1 | Ki = 960 nM | 0HT | C28 H48 N4 O5 | CC[C@H](C).... |
39 | 1OEW | - | SER THR | n/a | n/a |
40 | 1EPQ | Ki = 6.5 nM | 0QF | C31 H52 N4 O7 S2 | CCS[C@@H](.... |
41 | 5MB3 | - | 5GL | C13 H20 N2 O S | CCCN1C2=C(.... |
42 | 2JJI | - | 0QS | C36 H56 F2 N7 O8 S | CC(C)(C)S(.... |
43 | 3PCW | - | FBF | C8 H7 F3 N2 | [H]/N=C(/c.... |
44 | 3PGI | - | F41 | C14 H18 N2 O3 | c1cc2c(cc1.... |
45 | 4Y3J | Kd = 6.8 mM | HIC | C7 H11 N3 O2 | Cn1cc(nc1).... |
46 | 1GVW | Ki = 110 nM | 0EM | C32 H52 N6 O7 P | NULL |
47 | 5ER2 | Ki = 0.27 uM | 0EK | C50 H77 N9 O9 | NULL |
48 | 1EPP | Ki = 69 nM | 1Z1 | C32 H57 N7 O6 S2 | CC[C@H](C).... |
49 | 2ER7 | ic50 = 0.7 nM | BOC HIS PRO PHE HIS LOV ILE HIS | n/a | n/a |
50 | 4KUP | Ki = 6 uM | 1TZ | C21 H24 N4 O | Cc1cc(c(c(.... |
51 | 3WZ7 | Ki = 1.8 uM | IXY | C28 H30 N4 O2 S | c1ccc(cc1).... |
52 | 1EPO | Ki = 11 nM | 2Z3 | C32 H49 F2 N5 O7 | NULL |
53 | 1ER8 | - | DHI PRO PHE HIS LEU LEU VAL TYR | n/a | n/a |
54 | 3WZ8 | Ki = 1.5 uM | IXV | C27 H25 N3 O2 S | c1ccc(cc1).... |
55 | 3PI0 | - | F91 | C14 H14 N2 O2 | c1cc2c(cc1.... |
56 | 1GVU | Ki = 1 nM | PRO HIS PRO PHE HIS STA VAL ILE HIS LYS | n/a | n/a |
57 | 1EPL | - | PRO LEU GLU PSA ARG LEU | n/a | n/a |
58 | 4Y3Y | Kd = 4.5 mM | DCL | C6 H15 N O | CC(C)C[C@@.... |
59 | 1E5O | - | 3AI | C23 H38 N4 O4 S | CC[C@H](C).... |
60 | 3PLD | - | F90 | C8 H9 Cl N2 S | [H]/N=C(N).... |
61 | 5MB0 | Kd = 1.4 mM | F91 | C14 H14 N2 O2 | c1cc2c(cc1.... |
62 | 2ER6 | Ki = 60 nM | PRO THR GLU PUK ARG GLU | n/a | n/a |
63 | 3URI | - | HIS PRO HIS LEU SER 13E ALA HIS | n/a | n/a |
64 | 4LHH | Ki = 6 uM | 1TZ | C21 H24 N4 O | Cc1cc(c(c(.... |
65 | 4Y48 | - | GLY PRO | n/a | n/a |
66 | 1E82 | - | M90 | C34 H49 N5 O6 S | CSC[C@@H](.... |
67 | 1EPN | - | 2ZS | C31 H48 N4 O7 S | CC(C)OC(=O.... |
68 | 2ER9 | Ki = 40 nM | BOC HIS PRO PHE HIS STA LEU PHE | n/a | n/a |
69 | 4Y4J | Kd = 3.4 mM | LNR | C8 H11 N O3 | c1cc(c(cc1.... |
70 | 1GVX | Ki = 60 nM | PRO THR GLU PUK ARG GLU | n/a | n/a |
71 | 3PM4 | - | F5N | C15 H13 N3 O | c1ccc(cc1).... |
72 | 3PB5 | - | F63 | C11 H12 N2 O2 | CNCc1ccc(o.... |
73 | 4ZE6 | Kd = 3.3 mM | 011 | C7 H15 N O2 | C(CCCN)CCC.... |
74 | 3PBZ | - | F02 | C11 H17 N3 O | CCN(CC)c1c.... |
75 | 4ER1 | Ki = 0.24 uM | 0ZP | C51 H68 N5 O4 | CC[C@H](C).... |
76 | 5RBV | - | RQD | C10 H12 F N O2 | COC(=O)[C@.... |
77 | 5RCG | - | REG | C11 H20 N2 O2 | C1CCC(C1)N.... |
78 | 5R1U | - | T9G | C9 H13 N O | CC[C@H](c1.... |
79 | 5RC3 | - | RAY | C11 H14 F N O3 | COCCOCC(=O.... |
80 | 5R21 | - | R9Y | C11 H16 N2 | CN1CCCc2c1.... |
81 | 5RCE | - | RE4 | C11 H13 N5 | Cc1cc(nc(n.... |
82 | 5RBS | - | R8V | C9 H9 N O2 | CN1[C@H](c.... |
83 | 5RBU | - | R97 | C10 H10 N2 S | Cc1csc(n1).... |
84 | 5R2C | - | RE4 | C11 H13 N5 | Cc1cc(nc(n.... |
85 | 5R20 | - | R9V | C14 H19 N O | c1ccc(cc1).... |
86 | 5RCC | - | RDV | C12 H22 N2 O | C1CCC(C1)C.... |
87 | 5RC4 | - | RB7 | C11 H16 Br N O2 S | Cc1cc(ccc1.... |
88 | 5R25 | - | RBJ | C8 H11 N O | CNCc1ccc(c.... |
89 | 5HCT | Ki = 0.0254 uM | 61P | C30 H30 N8 O2 | c1ccc2c(c1.... |
90 | 5R1W | - | R8Y | C10 H13 N O3 S | CCN(CCC(=O.... |
91 | 5R23 | - | RAY | C11 H14 F N O3 | COCCOCC(=O.... |
92 | 5RC5 | - | RBG | C10 H20 N2 O | CC(C)(C)NC.... |
93 | 5RCB | - | RDM | C12 H15 N O3 | CC(=O)N[C@.... |
94 | 5RC6 | - | RBJ | C8 H11 N O | CNCc1ccc(c.... |
95 | 5RBQ | - | R8P | C8 H9 N O3 | C[C@@H](c1.... |
96 | 5R1V | - | R8S | C5 H8 N4 O | COc1ccnc(n.... |
97 | 5R1Z | - | R9M | C6 H7 N O2 S | c1csc(n1)C.... |
98 | 5R2B | - | RDY | C12 H15 N O4 | C[C@@H](C(.... |
99 | 5RC7 | - | AES | C8 H10 F N O2 S | c1cc(ccc1C.... |
100 | 5RBO | - | R8A | C6 H8 N2 O | c1cc(c(nc1.... |
101 | 5R26 | - | RCV | C10 H13 N O3 | COC(=O)COc.... |
102 | 5R1Y | - | R9J | C11 H15 N O2 | Cc1ccc(cc1.... |
103 | 5RBZ | - | R9S | C9 H11 N O | Cc1ccccc1C.... |
104 | 5R1X | - | RQD | C10 H12 F N O2 | COC(=O)[C@.... |
105 | 5RC8 | - | RCV | C10 H13 N O3 | COC(=O)COc.... |
106 | 5RC9 | - | RD4 | C9 H12 N2 O | [H]/N=C(c1.... |
107 | 5RBY | - | R9M | C6 H7 N O2 S | c1csc(n1)C.... |
108 | 5RCF | - | RE7 | C13 H16 F N3 | C[C@H](c1c.... |
109 | 5R24 | - | RB7 | C11 H16 Br N O2 S | Cc1cc(ccc1.... |
110 | 5R28 | - | RDJ | C9 H15 N3 O2 S | CCNC(=O)CS.... |
111 | 5RBT | - | RA7 | C8 H12 N2 O2 S | c1c(sc(n1).... |
112 | 5RCD | - | RDY | C12 H15 N O4 | C[C@@H](C(.... |
113 | 5RBR | - | R8S | C5 H8 N4 O | COc1ccnc(n.... |
114 | 5R2D | - | REG | C11 H20 N2 O2 | C1CCC(C1)N.... |
115 | 5RC0 | - | R9V | C14 H19 N O | c1ccc(cc1).... |
116 | 5R29 | - | RDM | C12 H15 N O3 | CC(=O)N[C@.... |
117 | 5R1T | - | R8A | C6 H8 N2 O | c1cc(c(nc1.... |
118 | 5R2A | - | RDV | C12 H22 N2 O | C1CCC(C1)C.... |
119 | 5R27 | - | RD4 | C9 H12 N2 O | [H]/N=C(c1.... |
120 | 5RBX | - | R9J | C11 H15 N O2 | Cc1ccc(cc1.... |
121 | 5RC1 | - | R9Y | C11 H16 N2 | CN1CCCc2c1.... |
122 | 5RCA | - | RDJ | C9 H15 N3 O2 S | CCNC(=O)CS.... |
123 | 5R22 | - | RA7 | C8 H12 N2 O2 S | c1c(sc(n1).... |
124 | 5RC2 | - | R8Y | C10 H13 N O3 S | CCN(CCC(=O.... |
125 | 5RBW | - | R9G | C12 H15 N O2 | COc1cccc(c.... |
126 | 5RBP | - | SYG | C9 H13 N O | CC[C@@H](c.... |
127 | 1PPM | Ki = 1600 nM | 0P1 | C29 H40 N3 O9 P | C[C@@H](C(.... |
128 | 2WED | Ki = 0.8 uM | PP6 | C29 H32 N2 O7 P | CC(C)[C@H].... |
129 | 1APU | Ki = 1.6 nM | IVA VAL VAL 32L | n/a | n/a |
130 | 2WEC | Ki = 110 uM | PP5 | C28 H32 N2 O7 P | CC(C)[C@@H.... |
131 | 1APW | Ki = 10 nM | IVA VAL VAL DFI NME | n/a | n/a |
132 | 1PPL | Ki = 2.8 nM | 1Z7 | C30 H50 N3 O8 P | CC(C)C[C@H.... |
133 | 2WEB | Ki = 7.6 uM | PP4 | C28 H32 N2 O7 P | CC(C)[C@@H.... |
134 | 2WEA | - | PP6 | C29 H32 N2 O7 P | CC(C)[C@H].... |
135 | 1BXO | Ki = 0.1 nM | PP7 | C30 H47 N4 O9 P | CC(C)C[C@@.... |
136 | 1APT | - | IVA VAL VAL LTA | n/a | n/a |
137 | 1PPK | Ki = 22 nM | IVV | C24 H46 N3 O7 P | CCOC(=O)C[.... |
138 | 1BXQ | Ki = 42 nM | PP8 | C29 H47 N4 O9 P | CC(C)C[C@H.... |
139 | 1APV | Ki = 1 nM | IVA VAL VAL DFO NME | n/a | n/a |
140 | 1IZE | - | IVA VAL VAL STA ALA STA | n/a | n/a |
141 | 3EMY | - | IVA VAL VAL STA ALA STA | n/a | n/a |
No: | PDB id | Binding Data | Representative ligand | Formula | Smiles |
---|---|---|---|---|---|
The Class containing this family consists of a total of 1 families. | |||||
1 | 1E81 | - | M91 | C34 H49 N5 O6 S | CSC[C@@H](.... |
2 | 4ZEA | - | IMI | C10 H17 N3 O2 S | C1[C@H]2[C.... |
3 | 3ER3 | Ki = 81 nM | 0EL | C51 H78 N8 O9 | NULL |
4 | 4Y4D | - | CFF | C8 H10 N4 O2 | Cn1cnc2c1C.... |
5 | 5LWT | - | 7B3 | C10 H13 N3 O | Cc1c2cnnc(.... |
6 | 1EPM | - | THR PHE GLN ALA PSA LEU ARG GLU | n/a | n/a |
7 | 1EED | Ki = 16.2 uM | 0EO | C34 H55 N3 O8 | CC(C)C[C@@.... |
8 | 3PMY | - | 41L | C15 H13 N3 O | c1ccc(cc1).... |
9 | 1OEX | - | BOC HIS PRO PHE ALA LOV ILE HIS | n/a | n/a |
10 | 4ER4 | Ki = 160 nM | PRO HIS PRO PHE HIS LAV ILE HIS LYS | n/a | n/a |
11 | 4LBT | Ki = 6 uM | 1TZ | C21 H24 N4 O | Cc1cc(c(c(.... |
12 | 3PWW | - | ROC | C38 H50 N6 O5 | CC(C)(C)NC.... |
13 | 4Y38 | Kd = 4 mM | 0A9 | C10 H13 N O2 | COC(=O)[C@.... |
14 | 2JJJ | - | 0QS | C36 H56 F2 N7 O8 S | CC(C)(C)S(.... |
15 | 1GVV | - | 0GM | C51 H61 N5 O6 | CC(C)C[C@H.... |
16 | 3PMU | - | F7L | C14 H20 F N O2 | c1ccc(c(c1.... |
17 | 5OJE | Ki = 6.1 uM | VSK | C22 H27 N3 O | Cc1cc(c(c(.... |
18 | 1GVT | - | 2ZS | C31 H48 N4 O7 S | CC(C)OC(=O.... |
19 | 1EPR | - | 0QS | C36 H56 F2 N7 O8 S | CC(C)(C)S(.... |
20 | 5MB5 | - | 46P | C8 H10 N4 S | Cc1c(sc(n1.... |
21 | 5MB7 | - | 4AV | C8 H9 Cl N2 O2 | CNCc1cc(cc.... |
22 | 4Y4G | - | GGB | C5 H12 N4 O3 | [H]/N=C(N).... |
23 | 3ER5 | Ki = 1 nM | PRO HIS PRO PHE HIS STA VAL ILE HIS LYS | n/a | n/a |
24 | 3URL | - | HIS SER LEU PHE HIS PUK THR PRO | n/a | n/a |
25 | 3PCZ | - | BAM | C7 H9 N2 | c1ccc(cc1).... |
26 | 2V00 | Kd = 0.22 mM | V15 | C12 H13 N3 O | c1ccc(cc1).... |
27 | 5LWR | - | 7B2 | C27 H29 Cl N9 O | Cc1c2cnn3c.... |
28 | 3PLL | - | F06 | C8 H9 Cl N2 S | [H]/N=C(N).... |
29 | 4ER2 | Ki = 0.5 nM | IVA VAL VAL STA ALA STA | n/a | n/a |
30 | 4LP9 | ic50 = 0.62 uM | SER LEU PHE HIS 22G THR PRO | n/a | n/a |
31 | 3PRS | - | RIT | C37 H48 N6 O5 S2 | CC(C)c1nc(.... |
32 | 1ENT | Ki = 110 nM | 0EM | C32 H52 N6 O7 P | NULL |
33 | 1E80 | - | 0GQ | C41 H64 N10 O6 | CC[C@H](C).... |
34 | 5LWS | - | 7B2 | C27 H29 Cl N9 O | Cc1c2cnn3c.... |
35 | 3PBD | - | F05 | C8 H8 N2 | c1ccc2c(c1.... |
36 | 1OD1 | - | 0QS | C36 H56 F2 N7 O8 S | CC(C)(C)S(.... |
37 | 3WZ6 | Ki = 1.1 uM | IXZ | C27 H25 N3 O2 S | c1ccc(cc1).... |
38 | 5ER1 | Ki = 960 nM | 0HT | C28 H48 N4 O5 | CC[C@H](C).... |
39 | 1OEW | - | SER THR | n/a | n/a |
40 | 1EPQ | Ki = 6.5 nM | 0QF | C31 H52 N4 O7 S2 | CCS[C@@H](.... |
41 | 5MB3 | - | 5GL | C13 H20 N2 O S | CCCN1C2=C(.... |
42 | 2JJI | - | 0QS | C36 H56 F2 N7 O8 S | CC(C)(C)S(.... |
43 | 3PCW | - | FBF | C8 H7 F3 N2 | [H]/N=C(/c.... |
44 | 3PGI | - | F41 | C14 H18 N2 O3 | c1cc2c(cc1.... |
45 | 4Y3J | Kd = 6.8 mM | HIC | C7 H11 N3 O2 | Cn1cc(nc1).... |
46 | 1GVW | Ki = 110 nM | 0EM | C32 H52 N6 O7 P | NULL |
47 | 5ER2 | Ki = 0.27 uM | 0EK | C50 H77 N9 O9 | NULL |
48 | 1EPP | Ki = 69 nM | 1Z1 | C32 H57 N7 O6 S2 | CC[C@H](C).... |
49 | 2ER7 | ic50 = 0.7 nM | BOC HIS PRO PHE HIS LOV ILE HIS | n/a | n/a |
50 | 4KUP | Ki = 6 uM | 1TZ | C21 H24 N4 O | Cc1cc(c(c(.... |
51 | 3WZ7 | Ki = 1.8 uM | IXY | C28 H30 N4 O2 S | c1ccc(cc1).... |
52 | 1EPO | Ki = 11 nM | 2Z3 | C32 H49 F2 N5 O7 | NULL |
53 | 1ER8 | - | DHI PRO PHE HIS LEU LEU VAL TYR | n/a | n/a |
54 | 3WZ8 | Ki = 1.5 uM | IXV | C27 H25 N3 O2 S | c1ccc(cc1).... |
55 | 3PI0 | - | F91 | C14 H14 N2 O2 | c1cc2c(cc1.... |
56 | 1GVU | Ki = 1 nM | PRO HIS PRO PHE HIS STA VAL ILE HIS LYS | n/a | n/a |
57 | 1EPL | - | PRO LEU GLU PSA ARG LEU | n/a | n/a |
58 | 4Y3Y | Kd = 4.5 mM | DCL | C6 H15 N O | CC(C)C[C@@.... |
59 | 1E5O | - | 3AI | C23 H38 N4 O4 S | CC[C@H](C).... |
60 | 3PLD | - | F90 | C8 H9 Cl N2 S | [H]/N=C(N).... |
61 | 5MB0 | Kd = 1.4 mM | F91 | C14 H14 N2 O2 | c1cc2c(cc1.... |
62 | 2ER6 | Ki = 60 nM | PRO THR GLU PUK ARG GLU | n/a | n/a |
63 | 3URI | - | HIS PRO HIS LEU SER 13E ALA HIS | n/a | n/a |
64 | 4LHH | Ki = 6 uM | 1TZ | C21 H24 N4 O | Cc1cc(c(c(.... |
65 | 4Y48 | - | GLY PRO | n/a | n/a |
66 | 1E82 | - | M90 | C34 H49 N5 O6 S | CSC[C@@H](.... |
67 | 1EPN | - | 2ZS | C31 H48 N4 O7 S | CC(C)OC(=O.... |
68 | 2ER9 | Ki = 40 nM | BOC HIS PRO PHE HIS STA LEU PHE | n/a | n/a |
69 | 4Y4J | Kd = 3.4 mM | LNR | C8 H11 N O3 | c1cc(c(cc1.... |
70 | 1GVX | Ki = 60 nM | PRO THR GLU PUK ARG GLU | n/a | n/a |
71 | 3PM4 | - | F5N | C15 H13 N3 O | c1ccc(cc1).... |
72 | 3PB5 | - | F63 | C11 H12 N2 O2 | CNCc1ccc(o.... |
73 | 4ZE6 | Kd = 3.3 mM | 011 | C7 H15 N O2 | C(CCCN)CCC.... |
74 | 3PBZ | - | F02 | C11 H17 N3 O | CCN(CC)c1c.... |
75 | 4ER1 | Ki = 0.24 uM | 0ZP | C51 H68 N5 O4 | CC[C@H](C).... |
76 | 3OWN | Ki = 34 nM | 3OX | C37 H48 N4 O7 S | CC(C)CNC(=.... |
77 | 2G21 | - | L1B | C19 H24 N5 O | CCc1c(c(nc.... |
78 | 4RYC | ic50 = 0.08 uM | 3ZK | C27 H39 N3 O6 S | Cc1ccc(cc1.... |
79 | 3D91 | Kd = 131 pM | REM | C33 H50 N4 O6 S | CC(C)(C)S(.... |
80 | 1BIL | ic50 = 0.5 nM | 0IU | C34 H53 N5 O5 S | NULL |
81 | 3KM4 | ic50 = 1.3 nM | 22X | C28 H45 Cl N4 O3 | CC(=O)NCCC.... |
82 | 2G24 | - | 7IG | C19 H19 F2 N5 | CCc1c(c(nc.... |
83 | 2IL2 | Kd = 79 nM | LIX | C32 H38 N6 O5 S | CCc1c(c(nc.... |
84 | 5SY3 | ic50 = 43 uM | 74Z | C15 H15 N3 O S | c1cc(oc1)C.... |
85 | 4Q1N | ic50 = 0.2 nM | 2Y9 | C26 H42 N4 O4 | CCOC[C@@H].... |
86 | 2I4Q | ic50 = 0.007 uM | UA4 | C25 H27 F2 N5 O3 | CCc1c(c(nc.... |
87 | 2BKS | ic50 = 37 nM | PZ1 | C34 H41 N3 O6 | COc1ccccc1.... |
88 | 4S1G | Ki = 0.6 nM | 43T | C24 H29 F N4 O2 | C[C@@H](c1.... |
89 | 4XX3 | Ki = 56 nM | 70X | C23 H28 N4 O2 | [H]/N=C1/N.... |
90 | 2G1S | - | 4IG | C24 H25 F2 N5 O3 | CCc1c(c(nc.... |
91 | 2G20 | - | L1A | C33 H50 N6 O7 S2 | CC(C)C[C@@.... |
92 | 5SXN | ic50 = 11 uM | 74U | C19 H15 N3 O | c1ccc(cc1).... |
93 | 3G70 | ic50 = 0.4 nM | A5T | C33 H32 Cl3 F2 N3 O2 | c1cc(c(c(c.... |
94 | 2G1Y | - | 5IG | C20 H27 N5 O3 | CCc1c(c(nc.... |
95 | 2G1R | - | 3IG | C20 H26 N6 O3 | CCc1c(c(nc.... |
96 | 4GJC | ic50 = 0.09 uM | 0MJ | C27 H29 N3 O4 S | Cc1ccc(cc1.... |
97 | 4GJ8 | - | 0LW | C20 H23 N O S | c1ccc2c(c1.... |
98 | 5SY2 | ic50 = 11 uM | 74V | C18 H25 N5 O2 | CCN([C@H]1.... |
99 | 5KOS | ic50 = 1.5 nM | 6VS | C27 H46 N6 O4 | CC(C)CN([C.... |
100 | 3G72 | ic50 = 0.8 nM | A6T | C33 H32 Cl3 F2 N3 O2 | c1cc(c(c(c.... |
101 | 3G6Z | ic50 = 0.2 nM | A7T | C35 H39 Cl2 N3 O3 | Cc1cccc(c1.... |
102 | 3GW5 | ic50 = 0.47 nM | 72X | C28 H46 Cl N3 O3 | CNC[C@H](C.... |
103 | 3SFC | ic50 = 0.003 uM | S53 | C32 H29 F N4 O2 | Cc1ccc(cc1.... |
104 | 2IKO | Kd = 3571 nM | 7IG | C19 H19 F2 N5 | CCc1c(c(nc.... |
105 | 3K1W | - | BFX | C31 H31 Br Cl F N2 O2 | c1ccc(c(c1.... |
106 | 4XX4 | Ki = 44 nM | 70Y | C25 H30 N4 O2 | [H]/N=C1/N.... |
107 | 2FS4 | ic50 = 37 nM | PZ1 | C34 H41 N3 O6 | COc1ccccc1.... |
108 | 2BKT | ic50 = 23 nM | RPF | C31 H37 N3 O5 | COc1ccccc1.... |
109 | 4GJ5 | - | 0LR | C22 H23 N O | c1ccc(cc1).... |
110 | 2G22 | - | 6IG | C27 H35 N5 O | CCc1c(c(nc.... |
111 | 1RNE | ic50 = 2 nM | C60 | C39 H63 N5 O6 S | CCCCNC(=O).... |
112 | 2G26 | - | 3LG | C32 H35 N3 O7 | COc1ccccc1.... |
113 | 4Y6M | - | 48Q | C39 H52 N4 O4 | CCCN(CCC)C.... |
114 | 5YIE | Ki = 5.6 nM | 8VF | C39 H51 N5 O6 S | CCN(CCN)c1.... |
115 | 5YID | Ki = 4 nM | K95 | C37 H44 N4 O6 S2 | CC1([C@H](.... |
116 | 2IGX | - | A1T | C41 H49 N5 O2 | CCCCCc1ccc.... |
117 | 5YIC | Ki = 1.3 nM | 8VO | C37 H45 N5 O6 S2 | CC1([C@H](.... |
118 | 4CKU | ic50 = 0.15 uM | P2F | C38 H52 N4 O6 S | CCCN(CCC)C.... |
119 | 1XDH | - | IVA VAL VAL STA ALA STA | n/a | n/a |
120 | 1LF2 | - | R37 | C32 H41 N3 O4 | Cc1cccc(c1.... |
121 | 5YIB | Ki = 3.3 nM | 8VC | C40 H53 N5 O6 S | Cc1cc(cc(c.... |
122 | 1LEE | - | R36 | C32 H41 N3 O4 | Cc1cccc(c1.... |
123 | 5YIA | Ki = 3 nM | 8V9 | C37 H44 N4 O7 S2 | CC1([C@H](.... |
124 | 1XE5 | - | 5FE | C29 H47 F6 N5 O9 | C[C@@H](C(.... |
125 | 5RBV | - | RQD | C10 H12 F N O2 | COC(=O)[C@.... |
126 | 5RCG | - | REG | C11 H20 N2 O2 | C1CCC(C1)N.... |
127 | 5R1U | - | T9G | C9 H13 N O | CC[C@H](c1.... |
128 | 5RC3 | - | RAY | C11 H14 F N O3 | COCCOCC(=O.... |
129 | 5R21 | - | R9Y | C11 H16 N2 | CN1CCCc2c1.... |
130 | 5RCE | - | RE4 | C11 H13 N5 | Cc1cc(nc(n.... |
131 | 5RBS | - | R8V | C9 H9 N O2 | CN1[C@H](c.... |
132 | 5RBU | - | R97 | C10 H10 N2 S | Cc1csc(n1).... |
133 | 5R2C | - | RE4 | C11 H13 N5 | Cc1cc(nc(n.... |
134 | 5R20 | - | R9V | C14 H19 N O | c1ccc(cc1).... |
135 | 5RCC | - | RDV | C12 H22 N2 O | C1CCC(C1)C.... |
136 | 5RC4 | - | RB7 | C11 H16 Br N O2 S | Cc1cc(ccc1.... |
137 | 5R25 | - | RBJ | C8 H11 N O | CNCc1ccc(c.... |
138 | 5HCT | Ki = 0.0254 uM | 61P | C30 H30 N8 O2 | c1ccc2c(c1.... |
139 | 5R1W | - | R8Y | C10 H13 N O3 S | CCN(CCC(=O.... |
140 | 5R23 | - | RAY | C11 H14 F N O3 | COCCOCC(=O.... |
141 | 5RC5 | - | RBG | C10 H20 N2 O | CC(C)(C)NC.... |
142 | 5RCB | - | RDM | C12 H15 N O3 | CC(=O)N[C@.... |
143 | 5RC6 | - | RBJ | C8 H11 N O | CNCc1ccc(c.... |
144 | 5RBQ | - | R8P | C8 H9 N O3 | C[C@@H](c1.... |
145 | 5R1V | - | R8S | C5 H8 N4 O | COc1ccnc(n.... |
146 | 5R1Z | - | R9M | C6 H7 N O2 S | c1csc(n1)C.... |
147 | 5R2B | - | RDY | C12 H15 N O4 | C[C@@H](C(.... |
148 | 5RC7 | - | AES | C8 H10 F N O2 S | c1cc(ccc1C.... |
149 | 5RBO | - | R8A | C6 H8 N2 O | c1cc(c(nc1.... |
150 | 5R26 | - | RCV | C10 H13 N O3 | COC(=O)COc.... |
151 | 5R1Y | - | R9J | C11 H15 N O2 | Cc1ccc(cc1.... |
152 | 5RBZ | - | R9S | C9 H11 N O | Cc1ccccc1C.... |
153 | 5R1X | - | RQD | C10 H12 F N O2 | COC(=O)[C@.... |
154 | 5RC8 | - | RCV | C10 H13 N O3 | COC(=O)COc.... |
155 | 5RC9 | - | RD4 | C9 H12 N2 O | [H]/N=C(c1.... |
156 | 5RBY | - | R9M | C6 H7 N O2 S | c1csc(n1)C.... |
157 | 5RCF | - | RE7 | C13 H16 F N3 | C[C@H](c1c.... |
158 | 5R24 | - | RB7 | C11 H16 Br N O2 S | Cc1cc(ccc1.... |
159 | 5R28 | - | RDJ | C9 H15 N3 O2 S | CCNC(=O)CS.... |
160 | 5RBT | - | RA7 | C8 H12 N2 O2 S | c1c(sc(n1).... |
161 | 5RCD | - | RDY | C12 H15 N O4 | C[C@@H](C(.... |
162 | 5RBR | - | R8S | C5 H8 N4 O | COc1ccnc(n.... |
163 | 5R2D | - | REG | C11 H20 N2 O2 | C1CCC(C1)N.... |
164 | 5RC0 | - | R9V | C14 H19 N O | c1ccc(cc1).... |
165 | 5R29 | - | RDM | C12 H15 N O3 | CC(=O)N[C@.... |
166 | 5R1T | - | R8A | C6 H8 N2 O | c1cc(c(nc1.... |
167 | 5R2A | - | RDV | C12 H22 N2 O | C1CCC(C1)C.... |
168 | 5R27 | - | RD4 | C9 H12 N2 O | [H]/N=C(c1.... |
169 | 5RBX | - | R9J | C11 H15 N O2 | Cc1ccc(cc1.... |
170 | 5RC1 | - | R9Y | C11 H16 N2 | CN1CCCc2c1.... |
171 | 5RCA | - | RDJ | C9 H15 N3 O2 S | CCNC(=O)CS.... |
172 | 5R22 | - | RA7 | C8 H12 N2 O2 S | c1c(sc(n1).... |
173 | 5RC2 | - | R8Y | C10 H13 N O3 S | CCN(CCC(=O.... |
174 | 5RBW | - | R9G | C12 H15 N O2 | COc1cccc(c.... |
175 | 5RBP | - | SYG | C9 H13 N O | CC[C@@H](c.... |
176 | 1PPM | Ki = 1600 nM | 0P1 | C29 H40 N3 O9 P | C[C@@H](C(.... |
177 | 2WED | Ki = 0.8 uM | PP6 | C29 H32 N2 O7 P | CC(C)[C@H].... |
178 | 1APU | Ki = 1.6 nM | IVA VAL VAL 32L | n/a | n/a |
179 | 2WEC | Ki = 110 uM | PP5 | C28 H32 N2 O7 P | CC(C)[C@@H.... |
180 | 1APW | Ki = 10 nM | IVA VAL VAL DFI NME | n/a | n/a |
181 | 1PPL | Ki = 2.8 nM | 1Z7 | C30 H50 N3 O8 P | CC(C)C[C@H.... |
182 | 2WEB | Ki = 7.6 uM | PP4 | C28 H32 N2 O7 P | CC(C)[C@@H.... |
183 | 2WEA | - | PP6 | C29 H32 N2 O7 P | CC(C)[C@H].... |
184 | 1BXO | Ki = 0.1 nM | PP7 | C30 H47 N4 O9 P | CC(C)C[C@@.... |
185 | 1APT | - | IVA VAL VAL LTA | n/a | n/a |
186 | 1PPK | Ki = 22 nM | IVV | C24 H46 N3 O7 P | CCOC(=O)C[.... |
187 | 1BXQ | Ki = 42 nM | PP8 | C29 H47 N4 O9 P | CC(C)C[C@H.... |
188 | 1APV | Ki = 1 nM | IVA VAL VAL DFO NME | n/a | n/a |
189 | 1SMR | - | PIV HIS PRO PHE HIS LPL TYR TYR SER | n/a | n/a |
190 | 1QRP | - | HH0 | C36 H60 N5 O10 P | C[C@@H](C(.... |
191 | 1PSO | - | IVA VAL VAL STA ALA STA | n/a | n/a |
192 | 2QZX | ic50 = 6 nM | IVA VAL VAL STA ALA STA | n/a | n/a |
193 | 2JXR | Ki = 90 nM | 2Z3 | C32 H49 F2 N5 O7 | NULL |
194 | 1FQ5 | Ki = 4 nM | 0GM | C51 H61 N5 O6 | CC(C)C[C@H.... |
195 | 1QS8 | - | IVA VAL VAL STA ALA STA | n/a | n/a |
196 | 1ZAP | Ki = 0.17 nM | A70 | C42 H70 N6 O5 | CCCC[C@@H].... |
197 | 1IZE | - | IVA VAL VAL STA ALA STA | n/a | n/a |
198 | 1WKR | - | IVA VAL VAL STA ALA STA | n/a | n/a |
199 | 5N7Q | - | IVA VAL VAL STA ALA STA | n/a | n/a |
200 | 5N70 | Kd ~ 3 nM | ALA PHE ARG ILE PRO LEU THR ARG | n/a | n/a |
201 | 3EMY | - | IVA VAL VAL STA ALA STA | n/a | n/a |
202 | 2H6T | Ki = 60 nM | IVA VAL VAL STA ALA STA | n/a | n/a |
203 | 3FV3 | Ki = 0.3 nM | IVA VAL VAL STA ALA STA | n/a | n/a |
204 | 3QVI | - | K95 | C37 H44 N4 O6 S2 | CC1([C@H](.... |
205 | 3APR | - | DHI PRO PHE HIS PUK VAL TYR | n/a | n/a |
206 | 6APR | Ki < 17 nM | IVA VAL VAL STA ALA STA | n/a | n/a |
207 | 5APR | Ki < 17 nM | HIS PRO PHE CYS STA LEU PHE DHL | n/a | n/a |
208 | 4APR | Ki = 200 nM | IVA HIS PRO PHE HIS STA LEU PHE | n/a | n/a |
209 | 1CZI | - | PRO PHI SMC NOR | n/a | n/a |
No: | Ligand | Similarity coefficient |
---|---|---|
1 | 3VS | 0.9352 |
2 | 9NB | 0.9254 |
3 | Y3L | 0.9233 |
4 | 6P3 | 0.9228 |
5 | LQ2 | 0.9218 |
6 | VC3 | 0.9214 |
7 | RYV | 0.9210 |
8 | 6FB | 0.9206 |
9 | PQS | 0.9204 |
10 | PQM | 0.9196 |
11 | XCG | 0.9178 |
12 | 1A5 | 0.9177 |
13 | KLS | 0.9174 |
14 | 4BY | 0.9173 |
15 | AES | 0.9165 |
16 | HRM | 0.9163 |
17 | 0SY | 0.9154 |
18 | A5Q | 0.9145 |
19 | K3D | 0.9141 |
20 | AZM | 0.9136 |
21 | 0UL | 0.9130 |
22 | I3E | 0.9127 |
23 | OLU | 0.9126 |
24 | 856 | 0.9124 |
25 | QIV | 0.9113 |
26 | 4I8 | 0.9112 |
27 | A7N | 0.9109 |
28 | LR8 | 0.9106 |
29 | KMY | 0.9103 |
30 | QBP | 0.9100 |
31 | N91 | 0.9097 |
32 | 8NB | 0.9097 |
33 | 2PV | 0.9095 |
34 | TMG | 0.9095 |
35 | 6KT | 0.9091 |
36 | 4JE | 0.9089 |
37 | 4CN | 0.9086 |
38 | PRL | 0.9083 |
39 | S0D | 0.9079 |
40 | 2PK | 0.9069 |
41 | CNI | 0.9069 |
42 | 2QC | 0.9068 |
43 | ZHA | 0.9068 |
44 | 3VX | 0.9065 |
45 | F4K | 0.9062 |
46 | 3ZB | 0.9061 |
47 | 4CM | 0.9054 |
48 | 4NP | 0.9054 |
49 | 7FU | 0.9051 |
50 | RNO | 0.9046 |
51 | TID | 0.9044 |
52 | AJ1 | 0.9043 |
53 | 1OT | 0.9042 |
54 | JBZ | 0.9034 |
55 | M4N | 0.9031 |
56 | L15 | 0.9031 |
57 | SNO | 0.9030 |
58 | ZRK | 0.9028 |
59 | N4E | 0.9028 |
60 | FZM | 0.9026 |
61 | ITE | 0.9023 |
62 | S7J | 0.9023 |
63 | FBF | 0.9017 |
64 | N1E | 0.9017 |
65 | 4NB | 0.9014 |
66 | 4MB | 0.9012 |
67 | FF2 | 0.9010 |
68 | 1OS | 0.9000 |
69 | UNJ | 0.8998 |
70 | JA5 | 0.8993 |
71 | 3W8 | 0.8991 |
72 | 3AE | 0.8988 |
73 | EUE | 0.8985 |
74 | FYR | 0.8984 |
75 | 7EH | 0.8984 |
76 | 4UM | 0.8982 |
77 | 2FX | 0.8981 |
78 | K4V | 0.8978 |
79 | S0E | 0.8977 |
80 | 4NZ | 0.8976 |
81 | 657 | 0.8975 |
82 | 8V8 | 0.8975 |
83 | MKN | 0.8974 |
84 | A7H | 0.8972 |
85 | 3W6 | 0.8968 |
86 | 3W3 | 0.8968 |
87 | 4NS | 0.8968 |
88 | L14 | 0.8967 |
89 | 1EB | 0.8966 |
90 | AJG | 0.8963 |
91 | ZEC | 0.8962 |
92 | 8CC | 0.8959 |
93 | PNP | 0.8958 |
94 | 5TT | 0.8957 |
95 | S98 | 0.8956 |
96 | JAH | 0.8953 |
97 | AM4 | 0.8952 |
98 | V1T | 0.8952 |
99 | J1K | 0.8951 |
100 | 245 | 0.8950 |
101 | X0U | 0.8950 |
102 | 1ZC | 0.8942 |
103 | 6SD | 0.8938 |
104 | 5LA | 0.8938 |
105 | 7MW | 0.8937 |
106 | 4BL | 0.8937 |
107 | 3VQ | 0.8936 |
108 | ANN | 0.8935 |
109 | NPX | 0.8929 |
110 | OQC | 0.8925 |
111 | RSV | 0.8924 |
112 | SWX | 0.8924 |
113 | PNZ | 0.8923 |
114 | 428 | 0.8920 |
115 | 1OU | 0.8919 |
116 | ZYX | 0.8917 |
117 | 72D | 0.8917 |
118 | 2WU | 0.8915 |
119 | BQ2 | 0.8912 |
120 | AMH | 0.8912 |
121 | NPS | 0.8910 |
122 | 5SJ | 0.8910 |
123 | 14N | 0.8910 |
124 | VD9 | 0.8910 |
125 | 5GV | 0.8905 |
126 | BGU | 0.8899 |
127 | 5E5 | 0.8894 |
128 | 833 | 0.8892 |
129 | C53 | 0.8886 |
130 | K97 | 0.8884 |
131 | K7H | 0.8878 |
132 | J6W | 0.8878 |
133 | 4FC | 0.8877 |
134 | KLV | 0.8875 |
135 | 5TY | 0.8873 |
136 | N2M | 0.8873 |
137 | LR5 | 0.8872 |
138 | YE6 | 0.8870 |
139 | 0NJ | 0.8870 |
140 | PPN | 0.8870 |
141 | 2P3 | 0.8869 |
142 | FCW | 0.8869 |
143 | HNT | 0.8868 |
144 | T1N | 0.8867 |
145 | WA1 | 0.8867 |
146 | 363 | 0.8866 |
147 | 0F3 | 0.8866 |
148 | FQX | 0.8865 |
149 | S7D | 0.8853 |
150 | 397 | 0.8852 |
151 | 68B | 0.8850 |
152 | AH9 | 0.8847 |
153 | FHV | 0.8844 |
154 | 7N8 | 0.8842 |
155 | 4BZ | 0.8842 |
156 | FBC | 0.8840 |
157 | 7O4 | 0.8839 |
158 | E3X | 0.8838 |
159 | 47V | 0.8838 |
160 | E7S | 0.8838 |
161 | ESP | 0.8837 |
162 | 2O8 | 0.8836 |
163 | GO2 | 0.8835 |
164 | KLE | 0.8834 |
165 | A9B | 0.8832 |
166 | JMG | 0.8831 |
167 | 6H2 | 0.8831 |
168 | ESX | 0.8830 |
169 | LZ5 | 0.8830 |
170 | 5RP | 0.8830 |
171 | 26C | 0.8829 |
172 | ZZA | 0.8828 |
173 | 0OK | 0.8827 |
174 | G14 | 0.8827 |
175 | MR6 | 0.8820 |
176 | LOT | 0.8816 |
177 | 92G | 0.8816 |
178 | 2J1 | 0.8815 |
179 | FER | 0.8815 |
180 | IBP | 0.8815 |
181 | 3R4 | 0.8814 |
182 | KW7 | 0.8813 |
183 | WV7 | 0.8811 |
184 | 4AU | 0.8811 |
185 | 4AF | 0.8810 |
186 | D26 | 0.8810 |
187 | RYY | 0.8805 |
188 | 3XR | 0.8804 |
189 | D25 | 0.8803 |
190 | JCZ | 0.8803 |
191 | GJP | 0.8802 |
192 | 5O6 | 0.8801 |
193 | 0FR | 0.8797 |
194 | CIY | 0.8795 |
195 | M83 | 0.8795 |
196 | 2JX | 0.8794 |
197 | PIQ | 0.8792 |
198 | OSP | 0.8792 |
199 | 9FH | 0.8790 |
200 | M78 | 0.8790 |
201 | 549 | 0.8789 |
202 | A6Z | 0.8789 |
203 | 4BX | 0.8789 |
204 | 6L6 | 0.8787 |
205 | AWE | 0.8787 |
206 | ODK | 0.8786 |
207 | S0A | 0.8785 |
208 | LUM | 0.8783 |
209 | 1KN | 0.8779 |
210 | SKF | 0.8779 |
211 | EZL | 0.8779 |
212 | EVF | 0.8779 |
213 | EES | 0.8777 |
214 | DHC | 0.8777 |
215 | 5H6 | 0.8777 |
216 | A5P | 0.8776 |
217 | 80G | 0.8775 |
218 | TEF | 0.8774 |
219 | ST3 | 0.8774 |
220 | RA7 | 0.8774 |
221 | BP7 | 0.8773 |
222 | DT7 | 0.8770 |
223 | 12T | 0.8769 |
224 | F2W | 0.8769 |
225 | 8D6 | 0.8766 |
226 | DVQ | 0.8764 |
227 | 27K | 0.8764 |
228 | 4HB | 0.8763 |
229 | RKN | 0.8763 |
230 | 9JT | 0.8763 |
231 | YI6 | 0.8762 |
232 | TFM | 0.8761 |
233 | BIO | 0.8760 |
234 | L22 | 0.8759 |
235 | X48 | 0.8758 |
236 | TJM | 0.8756 |
237 | S60 | 0.8755 |
238 | ZTW | 0.8752 |
239 | 801 | 0.8750 |
240 | V2Z | 0.8745 |
241 | 15E | 0.8744 |
242 | GVY | 0.8742 |
243 | N7I | 0.8738 |
244 | 0ON | 0.8738 |
245 | EE8 | 0.8735 |
246 | L2K | 0.8733 |
247 | 4NM | 0.8732 |
248 | M4S | 0.8731 |
249 | TYR | 0.8730 |
250 | D9Z | 0.8729 |
251 | 120 | 0.8728 |
252 | 3QV | 0.8725 |
253 | EAT | 0.8724 |
254 | BFL | 0.8724 |
255 | PPY | 0.8722 |
256 | ZYQ | 0.8721 |
257 | 5B2 | 0.8720 |
258 | PTR | 0.8720 |
259 | NDD | 0.8719 |
260 | 5VU | 0.8719 |
261 | 1DR | 0.8717 |
262 | E5X | 0.8717 |
263 | 259 | 0.8713 |
264 | J38 | 0.8712 |
265 | X2M | 0.8709 |
266 | MR4 | 0.8709 |
267 | 4AB | 0.8706 |
268 | 5ER | 0.8706 |
269 | WCU | 0.8705 |
270 | SSC | 0.8705 |
271 | NAG | 0.8704 |
272 | ERZ | 0.8703 |
273 | AN3 | 0.8702 |
274 | ZRL | 0.8701 |
275 | 5GT | 0.8698 |
276 | F18 | 0.8698 |
277 | PH3 | 0.8696 |
278 | NK5 | 0.8695 |
279 | F4E | 0.8695 |
280 | GNM | 0.8695 |
281 | A6W | 0.8691 |
282 | 613 | 0.8691 |
283 | ENO | 0.8689 |
284 | GB5 | 0.8685 |
285 | DDU | 0.8685 |
286 | AAN | 0.8683 |
287 | 122 | 0.8679 |
288 | BMZ | 0.8679 |
289 | CR4 | 0.8679 |
290 | 28A | 0.8678 |
291 | R52 | 0.8677 |
292 | I2E | 0.8677 |
293 | 1XS | 0.8677 |
294 | 68A | 0.8675 |
295 | BX4 | 0.8673 |
296 | DBS | 0.8670 |
297 | 27B | 0.8669 |
298 | EQW | 0.8667 |
299 | 4RU | 0.8664 |
300 | 2PW | 0.8663 |
301 | 4V2 | 0.8663 |
302 | LR2 | 0.8663 |
303 | BIK | 0.8662 |
304 | 4CF | 0.8662 |
305 | HC4 | 0.8661 |
306 | B1J | 0.8660 |
307 | 5WK | 0.8660 |
308 | DAH | 0.8659 |
309 | E1K | 0.8659 |
310 | PTB | 0.8657 |
311 | A5K | 0.8657 |
312 | X6W | 0.8653 |
313 | LO1 | 0.8652 |
314 | 0NX | 0.8652 |
315 | GOE | 0.8647 |
316 | 121 | 0.8640 |
317 | 92O | 0.8638 |
318 | SOJ | 0.8637 |
319 | U13 | 0.8637 |
320 | 4FF | 0.8634 |
321 | ICB | 0.8630 |
322 | MSR | 0.8629 |
323 | 2D2 | 0.8627 |
324 | STX | 0.8625 |
325 | 6N4 | 0.8622 |
326 | C4E | 0.8619 |
327 | A5E | 0.8618 |
328 | X0W | 0.8616 |
329 | BVS | 0.8613 |
330 | JMM | 0.8611 |
331 | 4FE | 0.8608 |
332 | 36E | 0.8608 |
333 | THA | 0.8606 |
334 | EN1 | 0.8604 |
335 | 9R5 | 0.8600 |
336 | AVX | 0.8599 |
337 | SNV | 0.8598 |
338 | BSU | 0.8596 |
339 | ENW | 0.8595 |
340 | PLP | 0.8595 |
341 | 0DF | 0.8593 |
342 | SJK | 0.8591 |
343 | CTE | 0.8588 |
344 | YE7 | 0.8588 |
345 | YZ9 | 0.8585 |
346 | LC1 | 0.8584 |
347 | EZ1 | 0.8584 |
348 | Z70 | 0.8584 |
349 | 9ZE | 0.8583 |
350 | SNU | 0.8580 |
351 | 0XR | 0.8580 |
352 | 3N1 | 0.8577 |
353 | A51 | 0.8573 |
354 | 2L1 | 0.8571 |
355 | 3D1 | 0.8571 |
356 | CBE | 0.8568 |
357 | MUX | 0.8564 |
358 | 5OR | 0.8563 |
359 | CK2 | 0.8560 |
360 | MMJ | 0.8559 |
361 | RES | 0.8559 |
362 | HBO | 0.8558 |
363 | 1Q1 | 0.8553 |
364 | 6QF | 0.8551 |
365 | HAR | 0.8546 |
366 | S62 | 0.8540 |
367 | 5F1 | 0.8536 |
368 | ALE | 0.8527 |
This union binding pocket(no: 1) in the query (biounit: 4er2.bio1) has 39 residues | |||
---|---|---|---|
No: | Leader PDB | Ligand | Sequence Similarity |
1 | 1J71 | THR ILE THR SER | 42.4242 |