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- Structure Biounit | Ligand Information
- PDB : .ZIP | .CSV
- Family 90% : .ZIP | .CSV
- Class : .ZIP | .CSV
No: | PDB id | Binding Data | Representative ligand | Formula | Smiles |
---|---|---|---|---|---|
The Class containing this family consists of a total of 4 families. | |||||
1 | 5EQR | - | TSV | C35 H44 F N5 O9 S | CC(C)(C)OC.... |
2 | 5ETX | - | 5RS | C36 H52 N6 O9 S | CCc1c(nc2c.... |
3 | 5VP9 | Ki = 1.03 nM | 9H7 | C38 H46 N6 O8 S2 | CC(C)(C)OC.... |
4 | 4WF8 | - | 2R9 | C35 H46 Cl N5 O9 S | CC(C)(C)[C.... |
5 | 3SU2 | Ki = 44.8 nM | TSV | C35 H44 F N5 O9 S | CC(C)(C)OC.... |
6 | 5EQS | - | 2R9 | C35 H46 Cl N5 O9 S | CC(C)(C)[C.... |
7 | 3RC5 | - | ACE GLN GLU ARG GLU VAL PRO CYS | n/a | n/a |
8 | 3M5M | - | ACE PHE ASP GLU MET GLU GLU CYS | n/a | n/a |
9 | 6NZV | - | L9J | C40 H54 F2 N6 O9 S | CC[C@@H]1[.... |
10 | 6PIZ | Ki = 27.9 nM | ON4 | C37 H48 N6 O9 S | Cc1c(nc2cc.... |
11 | 6PJ2 | Ki = 81 nM | OM7 | C40 H55 N7 O9 S | CC[C@H](C).... |
12 | 6PIW | Ki = 12.7 nM | OLV | C39 H52 N6 O9 S | Cc1c(nc2cc.... |
13 | 4WH6 | - | 2R9 | C35 H46 Cl N5 O9 S | CC(C)(C)[C.... |
14 | 6UE3 | Ki = 52 nM | 9H4 | C37 H50 N6 O9 S | Cc1c(nc2cc.... |
15 | 6CVW | Ki = 7.1 nM | FH1 | C37 H50 N6 O9 S | Cc1c(nc2cc.... |
16 | 3SV9 | - | SV6 | C36 H55 N7 O6 | CCC[C@@H](.... |
17 | 5EPN | Kd = 2.2 nM | 5R2 | C37 H50 N6 O9 S | CCc1c(nc2c.... |
18 | 3M5N | - | SER GLU CYS THR THR PRO CYS | n/a | n/a |
19 | 3SU0 | Ki = 162 nM | TSV | C35 H44 F N5 O9 S | CC(C)(C)OC.... |
20 | 3SU4 | Ki = 554 nM | SU3 | C38 H55 N5 O9 S | CC[C@@H]1C.... |
21 | 6CVY | Ki = 3.9 nM | FHD | C36 H49 Cl N6 O9 S | CCCCCOC(=O.... |
22 | 6PIX | Ki = 931 nM | OLY | C40 H55 N7 O10 S | Cc1c(nc2c(.... |
23 | 6PJ0 | Ki = 21.7 nM | OMV | C40 H54 N6 O9 S | CCC1(CCCC1.... |
24 | 6PIU | Ki = 9.68 nM | OL7 | C42 H57 N7 O10 S | Cc1c(nc2cc.... |
25 | 3SUE | Ki = 0.84 nM | SUE | C38 H50 N6 O9 S | CC(C)(C)[C.... |
26 | 6PIY | Ki = 46.4 nM | OMS | C38 H50 N6 O9 S | Cc1c(nc2cc.... |
27 | 3SU3 | Ki = 0.74 nM | SU3 | C38 H55 N5 O9 S | CC[C@@H]1C.... |
28 | 5VOJ | Ki = 3.6 nM | 9H4 | C37 H50 N6 O9 S | Cc1c(nc2cc.... |
29 | 6PIV | Ki = 2.3 nM | OLJ | C39 H50 N6 O9 S | Cc1c(nc2cc.... |
30 | 6CVX | Ki = 21 nM | FH4 | C39 H54 N6 O9 S | CC(C)c1c(n.... |
31 | 3SU6 | Ki = 958 nM | SU3 | C38 H55 N5 O9 S | CC[C@@H]1C.... |
32 | 3SUF | Ki = 27.8 nM | SUE | C38 H50 N6 O9 S | CC(C)(C)[C.... |
33 | 3SU1 | Ki = 208 nM | TSV | C35 H44 F N5 O9 S | CC(C)(C)OC.... |
34 | 3SU5 | Ki = 2635 nM | SU3 | C38 H55 N5 O9 S | CC[C@@H]1C.... |
35 | 6PJ1 | Ki = 16 nM | GKM | C39 H52 N6 O9 S | Cc1c(nc2cc.... |
36 | 5EQQ | Kd = 6.7 nM | 5RS | C36 H52 N6 O9 S | CCc1c(nc2c.... |
37 | 3SUG | Ki = 620 nM | SUE | C38 H50 N6 O9 S | CC(C)(C)[C.... |
38 | 3SUD | Ki = 0.14 nM | SUE | C38 H50 N6 O9 S | CC(C)(C)[C.... |
39 | 3M5O | - | ACE THR GLU ASP VAL VAL CYS CYS | n/a | n/a |
40 | 5ESB | - | SU3 | C38 H55 N5 O9 S | CC[C@@H]1C.... |
41 | 6NZT | - | L9P | C40 H52 F4 N6 O9 S | CC[C@@H]1[.... |
42 | 5EPY | - | 5R2 | C37 H50 N6 O9 S | CCc1c(nc2c.... |
43 | 3M5L | - | TSV | C35 H44 F N5 O9 S | CC(C)(C)OC.... |
44 | 4NWL | - | 2R9 | C35 H46 Cl N5 O9 S | CC(C)(C)[C.... |
45 | 6BQJ | - | Z1B | C39 H49 F2 N5 O9 S | CC(C)(C)[C.... |
46 | 6BQK | ic50 = 1 nM | Z1E | C34 H44 Cl F2 N5 O9 S | CC(C)(C)[C.... |
47 | 4NWK | - | 2R8 | C35 H47 N5 O9 S | CC(C)(C)[C.... |
48 | 7D5L | ic50 = 4.8 nM | GXO | C40 H51 F4 N5 O9 S | CC[C@@H]1C.... |
No: | PDB id | Binding Data | Representative ligand | Formula | Smiles |
---|---|---|---|---|---|
The Class containing this family consists of a total of 2 families. | |||||
1 | 5EQR | - | TSV | C35 H44 F N5 O9 S | CC(C)(C)OC.... |
2 | 5ETX | - | 5RS | C36 H52 N6 O9 S | CCc1c(nc2c.... |
3 | 5VP9 | Ki = 1.03 nM | 9H7 | C38 H46 N6 O8 S2 | CC(C)(C)OC.... |
4 | 4WF8 | - | 2R9 | C35 H46 Cl N5 O9 S | CC(C)(C)[C.... |
5 | 3SU2 | Ki = 44.8 nM | TSV | C35 H44 F N5 O9 S | CC(C)(C)OC.... |
6 | 5EQS | - | 2R9 | C35 H46 Cl N5 O9 S | CC(C)(C)[C.... |
7 | 3RC5 | - | ACE GLN GLU ARG GLU VAL PRO CYS | n/a | n/a |
8 | 3M5M | - | ACE PHE ASP GLU MET GLU GLU CYS | n/a | n/a |
9 | 6NZV | - | L9J | C40 H54 F2 N6 O9 S | CC[C@@H]1[.... |
10 | 6PIZ | Ki = 27.9 nM | ON4 | C37 H48 N6 O9 S | Cc1c(nc2cc.... |
11 | 6PJ2 | Ki = 81 nM | OM7 | C40 H55 N7 O9 S | CC[C@H](C).... |
12 | 6PIW | Ki = 12.7 nM | OLV | C39 H52 N6 O9 S | Cc1c(nc2cc.... |
13 | 4WH6 | - | 2R9 | C35 H46 Cl N5 O9 S | CC(C)(C)[C.... |
14 | 6UE3 | Ki = 52 nM | 9H4 | C37 H50 N6 O9 S | Cc1c(nc2cc.... |
15 | 6CVW | Ki = 7.1 nM | FH1 | C37 H50 N6 O9 S | Cc1c(nc2cc.... |
16 | 3SV9 | - | SV6 | C36 H55 N7 O6 | CCC[C@@H](.... |
17 | 5EPN | Kd = 2.2 nM | 5R2 | C37 H50 N6 O9 S | CCc1c(nc2c.... |
18 | 3M5N | - | SER GLU CYS THR THR PRO CYS | n/a | n/a |
19 | 3SU0 | Ki = 162 nM | TSV | C35 H44 F N5 O9 S | CC(C)(C)OC.... |
20 | 3SU4 | Ki = 554 nM | SU3 | C38 H55 N5 O9 S | CC[C@@H]1C.... |
21 | 6CVY | Ki = 3.9 nM | FHD | C36 H49 Cl N6 O9 S | CCCCCOC(=O.... |
22 | 6PIX | Ki = 931 nM | OLY | C40 H55 N7 O10 S | Cc1c(nc2c(.... |
23 | 6PJ0 | Ki = 21.7 nM | OMV | C40 H54 N6 O9 S | CCC1(CCCC1.... |
24 | 6PIU | Ki = 9.68 nM | OL7 | C42 H57 N7 O10 S | Cc1c(nc2cc.... |
25 | 3SUE | Ki = 0.84 nM | SUE | C38 H50 N6 O9 S | CC(C)(C)[C.... |
26 | 6PIY | Ki = 46.4 nM | OMS | C38 H50 N6 O9 S | Cc1c(nc2cc.... |
27 | 3SU3 | Ki = 0.74 nM | SU3 | C38 H55 N5 O9 S | CC[C@@H]1C.... |
28 | 5VOJ | Ki = 3.6 nM | 9H4 | C37 H50 N6 O9 S | Cc1c(nc2cc.... |
29 | 6PIV | Ki = 2.3 nM | OLJ | C39 H50 N6 O9 S | Cc1c(nc2cc.... |
30 | 6CVX | Ki = 21 nM | FH4 | C39 H54 N6 O9 S | CC(C)c1c(n.... |
31 | 3SU6 | Ki = 958 nM | SU3 | C38 H55 N5 O9 S | CC[C@@H]1C.... |
32 | 3SUF | Ki = 27.8 nM | SUE | C38 H50 N6 O9 S | CC(C)(C)[C.... |
33 | 3SU1 | Ki = 208 nM | TSV | C35 H44 F N5 O9 S | CC(C)(C)OC.... |
34 | 3SU5 | Ki = 2635 nM | SU3 | C38 H55 N5 O9 S | CC[C@@H]1C.... |
35 | 6PJ1 | Ki = 16 nM | GKM | C39 H52 N6 O9 S | Cc1c(nc2cc.... |
36 | 5EQQ | Kd = 6.7 nM | 5RS | C36 H52 N6 O9 S | CCc1c(nc2c.... |
37 | 3SUG | Ki = 620 nM | SUE | C38 H50 N6 O9 S | CC(C)(C)[C.... |
38 | 3SUD | Ki = 0.14 nM | SUE | C38 H50 N6 O9 S | CC(C)(C)[C.... |
39 | 3M5O | - | ACE THR GLU ASP VAL VAL CYS CYS | n/a | n/a |
40 | 5ESB | - | SU3 | C38 H55 N5 O9 S | CC[C@@H]1C.... |
41 | 6NZT | - | L9P | C40 H52 F4 N6 O9 S | CC[C@@H]1[.... |
42 | 5EPY | - | 5R2 | C37 H50 N6 O9 S | CCc1c(nc2c.... |
43 | 3M5L | - | TSV | C35 H44 F N5 O9 S | CC(C)(C)OC.... |
44 | 4NWL | - | 2R9 | C35 H46 Cl N5 O9 S | CC(C)(C)[C.... |
45 | 6BQJ | - | Z1B | C39 H49 F2 N5 O9 S | CC(C)(C)[C.... |
46 | 6BQK | ic50 = 1 nM | Z1E | C34 H44 Cl F2 N5 O9 S | CC(C)(C)[C.... |
47 | 4NWK | - | 2R8 | C35 H47 N5 O9 S | CC(C)(C)[C.... |
48 | 7D5L | ic50 = 4.8 nM | GXO | C40 H51 F4 N5 O9 S | CC[C@@H]1C.... |
This union binding pocket(no: 1) in the query (biounit: 3sud.bio3) has 23 residues | |||
---|---|---|---|
No: | Leader PDB | Ligand | Sequence Similarity |
This union binding pocket(no: 2) in the query (biounit: 3sud.bio1) has 52 residues | |||
---|---|---|---|
No: | Leader PDB | Ligand | Sequence Similarity |
This union binding pocket(no: 3) in the query (biounit: 3sud.bio2) has 58 residues | |||
---|---|---|---|
No: | Leader PDB | Ligand | Sequence Similarity |
This union binding pocket(no: 4) in the query (biounit: 3sud.bio4) has 24 residues | |||
---|---|---|---|
No: | Leader PDB | Ligand | Sequence Similarity |