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- PDB : .ZIP | .CSV
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- Class : .ZIP | .CSV
No: | PDB id | Binding Data | Representative ligand | Formula | Smiles |
---|---|---|---|---|---|
The Class containing this family consists of a total of 1 families. | |||||
1 | 1E81 | - | M91 | C34 H49 N5 O6 S | CSC[C@@H](.... |
2 | 4ZEA | - | IMI | C10 H17 N3 O2 S | C1[C@H]2[C.... |
3 | 3ER3 | Ki = 81 nM | 0EL | C51 H78 N8 O9 | NULL |
4 | 4Y4D | - | CFF | C8 H10 N4 O2 | Cn1cnc2c1C.... |
5 | 5LWT | - | 7B3 | C10 H13 N3 O | Cc1c2cnnc(.... |
6 | 1EPM | - | THR PHE GLN ALA PSA LEU ARG GLU | n/a | n/a |
7 | 1EED | Ki = 16.2 uM | 0EO | C34 H55 N3 O8 | CC(C)C[C@@.... |
8 | 3PMY | - | 41L | C15 H13 N3 O | c1ccc(cc1).... |
9 | 1OEX | - | BOC HIS PRO PHE ALA LOV ILE HIS | n/a | n/a |
10 | 4ER4 | Ki = 160 nM | PRO HIS PRO PHE HIS LAV ILE HIS LYS | n/a | n/a |
11 | 4LBT | Ki = 6 uM | 1TZ | C21 H24 N4 O | Cc1cc(c(c(.... |
12 | 3PWW | - | ROC | C38 H50 N6 O5 | CC(C)(C)NC.... |
13 | 4Y38 | Kd = 4 mM | 0A9 | C10 H13 N O2 | COC(=O)[C@.... |
14 | 2JJJ | - | 0QS | C36 H56 F2 N7 O8 S | CC(C)(C)S(.... |
15 | 1GVV | - | 0GM | C51 H61 N5 O6 | CC(C)C[C@H.... |
16 | 3PMU | - | F7L | C14 H20 F N O2 | c1ccc(c(c1.... |
17 | 5OJE | Ki = 6.1 uM | VSK | C22 H27 N3 O | Cc1cc(c(c(.... |
18 | 1GVT | - | 2ZS | C31 H48 N4 O7 S | CC(C)OC(=O.... |
19 | 1EPR | - | 0QS | C36 H56 F2 N7 O8 S | CC(C)(C)S(.... |
20 | 5MB5 | - | 46P | C8 H10 N4 S | Cc1c(sc(n1.... |
21 | 5MB7 | - | 4AV | C8 H9 Cl N2 O2 | CNCc1cc(cc.... |
22 | 4Y4G | - | GGB | C5 H12 N4 O3 | [H]/N=C(N).... |
23 | 3ER5 | Ki = 1 nM | PRO HIS PRO PHE HIS STA VAL ILE HIS LYS | n/a | n/a |
24 | 3URL | - | HIS SER LEU PHE HIS PUK THR PRO | n/a | n/a |
25 | 3PCZ | - | BAM | C7 H9 N2 | c1ccc(cc1).... |
26 | 2V00 | Kd = 0.22 mM | V15 | C12 H13 N3 O | c1ccc(cc1).... |
27 | 5LWR | - | 7B2 | C27 H29 Cl N9 O | Cc1c2cnn3c.... |
28 | 3PLL | - | F06 | C8 H9 Cl N2 S | [H]/N=C(N).... |
29 | 4ER2 | Ki = 0.5 nM | IVA VAL VAL STA ALA STA | n/a | n/a |
30 | 4LP9 | ic50 = 0.62 uM | SER LEU PHE HIS 22G THR PRO | n/a | n/a |
31 | 3PRS | - | RIT | C37 H48 N6 O5 S2 | CC(C)c1nc(.... |
32 | 1ENT | Ki = 110 nM | 0EM | C32 H52 N6 O7 P | NULL |
33 | 1E80 | - | 0GQ | C41 H64 N10 O6 | CC[C@H](C).... |
34 | 5LWS | - | 7B2 | C27 H29 Cl N9 O | Cc1c2cnn3c.... |
35 | 3PBD | - | F05 | C8 H8 N2 | c1ccc2c(c1.... |
36 | 1OD1 | - | 0QS | C36 H56 F2 N7 O8 S | CC(C)(C)S(.... |
37 | 3WZ6 | Ki = 1.1 uM | IXZ | C27 H25 N3 O2 S | c1ccc(cc1).... |
38 | 5ER1 | Ki = 960 nM | 0HT | C28 H48 N4 O5 | CC[C@H](C).... |
39 | 1OEW | - | SER THR | n/a | n/a |
40 | 1EPQ | Ki = 6.5 nM | 0QF | C31 H52 N4 O7 S2 | CCS[C@@H](.... |
41 | 5MB3 | - | 5GL | C13 H20 N2 O S | CCCN1C2=C(.... |
42 | 2JJI | - | 0QS | C36 H56 F2 N7 O8 S | CC(C)(C)S(.... |
43 | 3PCW | - | FBF | C8 H7 F3 N2 | [H]/N=C(/c.... |
44 | 3PGI | - | F41 | C14 H18 N2 O3 | c1cc2c(cc1.... |
45 | 4Y3J | Kd = 6.8 mM | HIC | C7 H11 N3 O2 | Cn1cc(nc1).... |
46 | 1GVW | Ki = 110 nM | 0EM | C32 H52 N6 O7 P | NULL |
47 | 5ER2 | Ki = 0.27 uM | 0EK | C50 H77 N9 O9 | NULL |
48 | 1EPP | Ki = 69 nM | 1Z1 | C32 H57 N7 O6 S2 | CC[C@H](C).... |
49 | 2ER7 | ic50 = 0.7 nM | BOC HIS PRO PHE HIS LOV ILE HIS | n/a | n/a |
50 | 4KUP | Ki = 6 uM | 1TZ | C21 H24 N4 O | Cc1cc(c(c(.... |
51 | 3WZ7 | Ki = 1.8 uM | IXY | C28 H30 N4 O2 S | c1ccc(cc1).... |
52 | 1EPO | Ki = 11 nM | 2Z3 | C32 H49 F2 N5 O7 | NULL |
53 | 1ER8 | - | DHI PRO PHE HIS LEU LEU VAL TYR | n/a | n/a |
54 | 3WZ8 | Ki = 1.5 uM | IXV | C27 H25 N3 O2 S | c1ccc(cc1).... |
55 | 3PI0 | - | F91 | C14 H14 N2 O2 | c1cc2c(cc1.... |
56 | 1GVU | Ki = 1 nM | PRO HIS PRO PHE HIS STA VAL ILE HIS LYS | n/a | n/a |
57 | 1EPL | - | PRO LEU GLU PSA ARG LEU | n/a | n/a |
58 | 4Y3Y | Kd = 4.5 mM | DCL | C6 H15 N O | CC(C)C[C@@.... |
59 | 1E5O | - | 3AI | C23 H38 N4 O4 S | CC[C@H](C).... |
60 | 3PLD | - | F90 | C8 H9 Cl N2 S | [H]/N=C(N).... |
61 | 5MB0 | Kd = 1.4 mM | F91 | C14 H14 N2 O2 | c1cc2c(cc1.... |
62 | 2ER6 | Ki = 60 nM | PRO THR GLU PUK ARG GLU | n/a | n/a |
63 | 3URI | - | HIS PRO HIS LEU SER 13E ALA HIS | n/a | n/a |
64 | 4LHH | Ki = 6 uM | 1TZ | C21 H24 N4 O | Cc1cc(c(c(.... |
65 | 4Y48 | - | GLY PRO | n/a | n/a |
66 | 1E82 | - | M90 | C34 H49 N5 O6 S | CSC[C@@H](.... |
67 | 1EPN | - | 2ZS | C31 H48 N4 O7 S | CC(C)OC(=O.... |
68 | 2ER9 | Ki = 40 nM | BOC HIS PRO PHE HIS STA LEU PHE | n/a | n/a |
69 | 4Y4J | Kd = 3.4 mM | LNR | C8 H11 N O3 | c1cc(c(cc1.... |
70 | 1GVX | Ki = 60 nM | PRO THR GLU PUK ARG GLU | n/a | n/a |
71 | 3PM4 | - | F5N | C15 H13 N3 O | c1ccc(cc1).... |
72 | 3PB5 | - | F63 | C11 H12 N2 O2 | CNCc1ccc(o.... |
73 | 4ZE6 | Kd = 3.3 mM | 011 | C7 H15 N O2 | C(CCCN)CCC.... |
74 | 3PBZ | - | F02 | C11 H17 N3 O | CCN(CC)c1c.... |
75 | 4ER1 | Ki = 0.24 uM | 0ZP | C51 H68 N5 O4 | CC[C@H](C).... |
76 | 5RBV | - | RQD | C10 H12 F N O2 | COC(=O)[C@.... |
77 | 5RCG | - | REG | C11 H20 N2 O2 | C1CCC(C1)N.... |
78 | 5R1U | - | T9G | C9 H13 N O | CC[C@H](c1.... |
79 | 5RC3 | - | RAY | C11 H14 F N O3 | COCCOCC(=O.... |
80 | 5R21 | - | R9Y | C11 H16 N2 | CN1CCCc2c1.... |
81 | 5RCE | - | RE4 | C11 H13 N5 | Cc1cc(nc(n.... |
82 | 5RBS | - | R8V | C9 H9 N O2 | CN1[C@H](c.... |
83 | 5RBU | - | R97 | C10 H10 N2 S | Cc1csc(n1).... |
84 | 5R2C | - | RE4 | C11 H13 N5 | Cc1cc(nc(n.... |
85 | 5R20 | - | R9V | C14 H19 N O | c1ccc(cc1).... |
86 | 5RCC | - | RDV | C12 H22 N2 O | C1CCC(C1)C.... |
87 | 5RC4 | - | RB7 | C11 H16 Br N O2 S | Cc1cc(ccc1.... |
88 | 5R25 | - | RBJ | C8 H11 N O | CNCc1ccc(c.... |
89 | 5HCT | Ki = 0.0254 uM | 61P | C30 H30 N8 O2 | c1ccc2c(c1.... |
90 | 5R1W | - | R8Y | C10 H13 N O3 S | CCN(CCC(=O.... |
91 | 5R23 | - | RAY | C11 H14 F N O3 | COCCOCC(=O.... |
92 | 5RC5 | - | RBG | C10 H20 N2 O | CC(C)(C)NC.... |
93 | 5RCB | - | RDM | C12 H15 N O3 | CC(=O)N[C@.... |
94 | 5RC6 | - | RBJ | C8 H11 N O | CNCc1ccc(c.... |
95 | 5RBQ | - | R8P | C8 H9 N O3 | C[C@@H](c1.... |
96 | 5R1V | - | R8S | C5 H8 N4 O | COc1ccnc(n.... |
97 | 5R1Z | - | R9M | C6 H7 N O2 S | c1csc(n1)C.... |
98 | 5R2B | - | RDY | C12 H15 N O4 | C[C@@H](C(.... |
99 | 5RC7 | - | AES | C8 H10 F N O2 S | c1cc(ccc1C.... |
100 | 5RBO | - | R8A | C6 H8 N2 O | c1cc(c(nc1.... |
101 | 5R26 | - | RCV | C10 H13 N O3 | COC(=O)COc.... |
102 | 5R1Y | - | R9J | C11 H15 N O2 | Cc1ccc(cc1.... |
103 | 5RBZ | - | R9S | C9 H11 N O | Cc1ccccc1C.... |
104 | 5R1X | - | RQD | C10 H12 F N O2 | COC(=O)[C@.... |
105 | 5RC8 | - | RCV | C10 H13 N O3 | COC(=O)COc.... |
106 | 5RC9 | - | RD4 | C9 H12 N2 O | [H]/N=C(c1.... |
107 | 5RBY | - | R9M | C6 H7 N O2 S | c1csc(n1)C.... |
108 | 5RCF | - | RE7 | C13 H16 F N3 | C[C@H](c1c.... |
109 | 5R24 | - | RB7 | C11 H16 Br N O2 S | Cc1cc(ccc1.... |
110 | 5R28 | - | RDJ | C9 H15 N3 O2 S | CCNC(=O)CS.... |
111 | 5RBT | - | RA7 | C8 H12 N2 O2 S | c1c(sc(n1).... |
112 | 5RCD | - | RDY | C12 H15 N O4 | C[C@@H](C(.... |
113 | 5RBR | - | R8S | C5 H8 N4 O | COc1ccnc(n.... |
114 | 5R2D | - | REG | C11 H20 N2 O2 | C1CCC(C1)N.... |
115 | 5RC0 | - | R9V | C14 H19 N O | c1ccc(cc1).... |
116 | 5R29 | - | RDM | C12 H15 N O3 | CC(=O)N[C@.... |
117 | 5R1T | - | R8A | C6 H8 N2 O | c1cc(c(nc1.... |
118 | 5R2A | - | RDV | C12 H22 N2 O | C1CCC(C1)C.... |
119 | 5R27 | - | RD4 | C9 H12 N2 O | [H]/N=C(c1.... |
120 | 5RBX | - | R9J | C11 H15 N O2 | Cc1ccc(cc1.... |
121 | 5RC1 | - | R9Y | C11 H16 N2 | CN1CCCc2c1.... |
122 | 5RCA | - | RDJ | C9 H15 N3 O2 S | CCNC(=O)CS.... |
123 | 5R22 | - | RA7 | C8 H12 N2 O2 S | c1c(sc(n1).... |
124 | 5RC2 | - | R8Y | C10 H13 N O3 S | CCN(CCC(=O.... |
125 | 5RBW | - | R9G | C12 H15 N O2 | COc1cccc(c.... |
126 | 5RBP | - | SYG | C9 H13 N O | CC[C@@H](c.... |
127 | 1PPM | Ki = 1600 nM | 0P1 | C29 H40 N3 O9 P | C[C@@H](C(.... |
128 | 2WED | Ki = 0.8 uM | PP6 | C29 H32 N2 O7 P | CC(C)[C@H].... |
129 | 1APU | Ki = 1.6 nM | IVA VAL VAL 32L | n/a | n/a |
130 | 2WEC | Ki = 110 uM | PP5 | C28 H32 N2 O7 P | CC(C)[C@@H.... |
131 | 1APW | Ki = 10 nM | IVA VAL VAL DFI NME | n/a | n/a |
132 | 1PPL | Ki = 2.8 nM | 1Z7 | C30 H50 N3 O8 P | CC(C)C[C@H.... |
133 | 2WEB | Ki = 7.6 uM | PP4 | C28 H32 N2 O7 P | CC(C)[C@@H.... |
134 | 2WEA | - | PP6 | C29 H32 N2 O7 P | CC(C)[C@H].... |
135 | 1BXO | Ki = 0.1 nM | PP7 | C30 H47 N4 O9 P | CC(C)C[C@@.... |
136 | 1APT | - | IVA VAL VAL LTA | n/a | n/a |
137 | 1PPK | Ki = 22 nM | IVV | C24 H46 N3 O7 P | CCOC(=O)C[.... |
138 | 1BXQ | Ki = 42 nM | PP8 | C29 H47 N4 O9 P | CC(C)C[C@H.... |
139 | 1APV | Ki = 1 nM | IVA VAL VAL DFO NME | n/a | n/a |
140 | 1IZE | - | IVA VAL VAL STA ALA STA | n/a | n/a |
141 | 3EMY | - | IVA VAL VAL STA ALA STA | n/a | n/a |
No: | PDB id | Binding Data | Representative ligand | Formula | Smiles |
---|---|---|---|---|---|
The Class containing this family consists of a total of 1 families. | |||||
1 | 1E81 | - | M91 | C34 H49 N5 O6 S | CSC[C@@H](.... |
2 | 4ZEA | - | IMI | C10 H17 N3 O2 S | C1[C@H]2[C.... |
3 | 3ER3 | Ki = 81 nM | 0EL | C51 H78 N8 O9 | NULL |
4 | 4Y4D | - | CFF | C8 H10 N4 O2 | Cn1cnc2c1C.... |
5 | 5LWT | - | 7B3 | C10 H13 N3 O | Cc1c2cnnc(.... |
6 | 1EPM | - | THR PHE GLN ALA PSA LEU ARG GLU | n/a | n/a |
7 | 1EED | Ki = 16.2 uM | 0EO | C34 H55 N3 O8 | CC(C)C[C@@.... |
8 | 3PMY | - | 41L | C15 H13 N3 O | c1ccc(cc1).... |
9 | 1OEX | - | BOC HIS PRO PHE ALA LOV ILE HIS | n/a | n/a |
10 | 4ER4 | Ki = 160 nM | PRO HIS PRO PHE HIS LAV ILE HIS LYS | n/a | n/a |
11 | 4LBT | Ki = 6 uM | 1TZ | C21 H24 N4 O | Cc1cc(c(c(.... |
12 | 3PWW | - | ROC | C38 H50 N6 O5 | CC(C)(C)NC.... |
13 | 4Y38 | Kd = 4 mM | 0A9 | C10 H13 N O2 | COC(=O)[C@.... |
14 | 2JJJ | - | 0QS | C36 H56 F2 N7 O8 S | CC(C)(C)S(.... |
15 | 1GVV | - | 0GM | C51 H61 N5 O6 | CC(C)C[C@H.... |
16 | 3PMU | - | F7L | C14 H20 F N O2 | c1ccc(c(c1.... |
17 | 5OJE | Ki = 6.1 uM | VSK | C22 H27 N3 O | Cc1cc(c(c(.... |
18 | 1GVT | - | 2ZS | C31 H48 N4 O7 S | CC(C)OC(=O.... |
19 | 1EPR | - | 0QS | C36 H56 F2 N7 O8 S | CC(C)(C)S(.... |
20 | 5MB5 | - | 46P | C8 H10 N4 S | Cc1c(sc(n1.... |
21 | 5MB7 | - | 4AV | C8 H9 Cl N2 O2 | CNCc1cc(cc.... |
22 | 4Y4G | - | GGB | C5 H12 N4 O3 | [H]/N=C(N).... |
23 | 3ER5 | Ki = 1 nM | PRO HIS PRO PHE HIS STA VAL ILE HIS LYS | n/a | n/a |
24 | 3URL | - | HIS SER LEU PHE HIS PUK THR PRO | n/a | n/a |
25 | 3PCZ | - | BAM | C7 H9 N2 | c1ccc(cc1).... |
26 | 2V00 | Kd = 0.22 mM | V15 | C12 H13 N3 O | c1ccc(cc1).... |
27 | 5LWR | - | 7B2 | C27 H29 Cl N9 O | Cc1c2cnn3c.... |
28 | 3PLL | - | F06 | C8 H9 Cl N2 S | [H]/N=C(N).... |
29 | 4ER2 | Ki = 0.5 nM | IVA VAL VAL STA ALA STA | n/a | n/a |
30 | 4LP9 | ic50 = 0.62 uM | SER LEU PHE HIS 22G THR PRO | n/a | n/a |
31 | 3PRS | - | RIT | C37 H48 N6 O5 S2 | CC(C)c1nc(.... |
32 | 1ENT | Ki = 110 nM | 0EM | C32 H52 N6 O7 P | NULL |
33 | 1E80 | - | 0GQ | C41 H64 N10 O6 | CC[C@H](C).... |
34 | 5LWS | - | 7B2 | C27 H29 Cl N9 O | Cc1c2cnn3c.... |
35 | 3PBD | - | F05 | C8 H8 N2 | c1ccc2c(c1.... |
36 | 1OD1 | - | 0QS | C36 H56 F2 N7 O8 S | CC(C)(C)S(.... |
37 | 3WZ6 | Ki = 1.1 uM | IXZ | C27 H25 N3 O2 S | c1ccc(cc1).... |
38 | 5ER1 | Ki = 960 nM | 0HT | C28 H48 N4 O5 | CC[C@H](C).... |
39 | 1OEW | - | SER THR | n/a | n/a |
40 | 1EPQ | Ki = 6.5 nM | 0QF | C31 H52 N4 O7 S2 | CCS[C@@H](.... |
41 | 5MB3 | - | 5GL | C13 H20 N2 O S | CCCN1C2=C(.... |
42 | 2JJI | - | 0QS | C36 H56 F2 N7 O8 S | CC(C)(C)S(.... |
43 | 3PCW | - | FBF | C8 H7 F3 N2 | [H]/N=C(/c.... |
44 | 3PGI | - | F41 | C14 H18 N2 O3 | c1cc2c(cc1.... |
45 | 4Y3J | Kd = 6.8 mM | HIC | C7 H11 N3 O2 | Cn1cc(nc1).... |
46 | 1GVW | Ki = 110 nM | 0EM | C32 H52 N6 O7 P | NULL |
47 | 5ER2 | Ki = 0.27 uM | 0EK | C50 H77 N9 O9 | NULL |
48 | 1EPP | Ki = 69 nM | 1Z1 | C32 H57 N7 O6 S2 | CC[C@H](C).... |
49 | 2ER7 | ic50 = 0.7 nM | BOC HIS PRO PHE HIS LOV ILE HIS | n/a | n/a |
50 | 4KUP | Ki = 6 uM | 1TZ | C21 H24 N4 O | Cc1cc(c(c(.... |
51 | 3WZ7 | Ki = 1.8 uM | IXY | C28 H30 N4 O2 S | c1ccc(cc1).... |
52 | 1EPO | Ki = 11 nM | 2Z3 | C32 H49 F2 N5 O7 | NULL |
53 | 1ER8 | - | DHI PRO PHE HIS LEU LEU VAL TYR | n/a | n/a |
54 | 3WZ8 | Ki = 1.5 uM | IXV | C27 H25 N3 O2 S | c1ccc(cc1).... |
55 | 3PI0 | - | F91 | C14 H14 N2 O2 | c1cc2c(cc1.... |
56 | 1GVU | Ki = 1 nM | PRO HIS PRO PHE HIS STA VAL ILE HIS LYS | n/a | n/a |
57 | 1EPL | - | PRO LEU GLU PSA ARG LEU | n/a | n/a |
58 | 4Y3Y | Kd = 4.5 mM | DCL | C6 H15 N O | CC(C)C[C@@.... |
59 | 1E5O | - | 3AI | C23 H38 N4 O4 S | CC[C@H](C).... |
60 | 3PLD | - | F90 | C8 H9 Cl N2 S | [H]/N=C(N).... |
61 | 5MB0 | Kd = 1.4 mM | F91 | C14 H14 N2 O2 | c1cc2c(cc1.... |
62 | 2ER6 | Ki = 60 nM | PRO THR GLU PUK ARG GLU | n/a | n/a |
63 | 3URI | - | HIS PRO HIS LEU SER 13E ALA HIS | n/a | n/a |
64 | 4LHH | Ki = 6 uM | 1TZ | C21 H24 N4 O | Cc1cc(c(c(.... |
65 | 4Y48 | - | GLY PRO | n/a | n/a |
66 | 1E82 | - | M90 | C34 H49 N5 O6 S | CSC[C@@H](.... |
67 | 1EPN | - | 2ZS | C31 H48 N4 O7 S | CC(C)OC(=O.... |
68 | 2ER9 | Ki = 40 nM | BOC HIS PRO PHE HIS STA LEU PHE | n/a | n/a |
69 | 4Y4J | Kd = 3.4 mM | LNR | C8 H11 N O3 | c1cc(c(cc1.... |
70 | 1GVX | Ki = 60 nM | PRO THR GLU PUK ARG GLU | n/a | n/a |
71 | 3PM4 | - | F5N | C15 H13 N3 O | c1ccc(cc1).... |
72 | 3PB5 | - | F63 | C11 H12 N2 O2 | CNCc1ccc(o.... |
73 | 4ZE6 | Kd = 3.3 mM | 011 | C7 H15 N O2 | C(CCCN)CCC.... |
74 | 3PBZ | - | F02 | C11 H17 N3 O | CCN(CC)c1c.... |
75 | 4ER1 | Ki = 0.24 uM | 0ZP | C51 H68 N5 O4 | CC[C@H](C).... |
76 | 3OWN | Ki = 34 nM | 3OX | C37 H48 N4 O7 S | CC(C)CNC(=.... |
77 | 2G21 | - | L1B | C19 H24 N5 O | CCc1c(c(nc.... |
78 | 4RYC | ic50 = 0.08 uM | 3ZK | C27 H39 N3 O6 S | Cc1ccc(cc1.... |
79 | 3D91 | Kd = 131 pM | REM | C33 H50 N4 O6 S | CC(C)(C)S(.... |
80 | 1BIL | ic50 = 0.5 nM | 0IU | C34 H53 N5 O5 S | NULL |
81 | 3KM4 | ic50 = 1.3 nM | 22X | C28 H45 Cl N4 O3 | CC(=O)NCCC.... |
82 | 2G24 | - | 7IG | C19 H19 F2 N5 | CCc1c(c(nc.... |
83 | 2IL2 | Kd = 79 nM | LIX | C32 H38 N6 O5 S | CCc1c(c(nc.... |
84 | 5SY3 | ic50 = 43 uM | 74Z | C15 H15 N3 O S | c1cc(oc1)C.... |
85 | 4Q1N | ic50 = 0.2 nM | 2Y9 | C26 H42 N4 O4 | CCOC[C@@H].... |
86 | 2I4Q | ic50 = 0.007 uM | UA4 | C25 H27 F2 N5 O3 | CCc1c(c(nc.... |
87 | 2BKS | ic50 = 37 nM | PZ1 | C34 H41 N3 O6 | COc1ccccc1.... |
88 | 4S1G | Ki = 0.6 nM | 43T | C24 H29 F N4 O2 | C[C@@H](c1.... |
89 | 4XX3 | Ki = 56 nM | 70X | C23 H28 N4 O2 | [H]/N=C1/N.... |
90 | 2G1S | - | 4IG | C24 H25 F2 N5 O3 | CCc1c(c(nc.... |
91 | 2G20 | - | L1A | C33 H50 N6 O7 S2 | CC(C)C[C@@.... |
92 | 5SXN | ic50 = 11 uM | 74U | C19 H15 N3 O | c1ccc(cc1).... |
93 | 3G70 | ic50 = 0.4 nM | A5T | C33 H32 Cl3 F2 N3 O2 | c1cc(c(c(c.... |
94 | 2G1Y | - | 5IG | C20 H27 N5 O3 | CCc1c(c(nc.... |
95 | 2G1R | - | 3IG | C20 H26 N6 O3 | CCc1c(c(nc.... |
96 | 4GJC | ic50 = 0.09 uM | 0MJ | C27 H29 N3 O4 S | Cc1ccc(cc1.... |
97 | 4GJ8 | - | 0LW | C20 H23 N O S | c1ccc2c(c1.... |
98 | 5SY2 | ic50 = 11 uM | 74V | C18 H25 N5 O2 | CCN([C@H]1.... |
99 | 5KOS | ic50 = 1.5 nM | 6VS | C27 H46 N6 O4 | CC(C)CN([C.... |
100 | 3G72 | ic50 = 0.8 nM | A6T | C33 H32 Cl3 F2 N3 O2 | c1cc(c(c(c.... |
101 | 3G6Z | ic50 = 0.2 nM | A7T | C35 H39 Cl2 N3 O3 | Cc1cccc(c1.... |
102 | 3GW5 | ic50 = 0.47 nM | 72X | C28 H46 Cl N3 O3 | CNC[C@H](C.... |
103 | 3SFC | ic50 = 0.003 uM | S53 | C32 H29 F N4 O2 | Cc1ccc(cc1.... |
104 | 2IKO | Kd = 3571 nM | 7IG | C19 H19 F2 N5 | CCc1c(c(nc.... |
105 | 3K1W | - | BFX | C31 H31 Br Cl F N2 O2 | c1ccc(c(c1.... |
106 | 4XX4 | Ki = 44 nM | 70Y | C25 H30 N4 O2 | [H]/N=C1/N.... |
107 | 2FS4 | ic50 = 37 nM | PZ1 | C34 H41 N3 O6 | COc1ccccc1.... |
108 | 2BKT | ic50 = 23 nM | RPF | C31 H37 N3 O5 | COc1ccccc1.... |
109 | 4GJ5 | - | 0LR | C22 H23 N O | c1ccc(cc1).... |
110 | 2G22 | - | 6IG | C27 H35 N5 O | CCc1c(c(nc.... |
111 | 1RNE | ic50 = 2 nM | C60 | C39 H63 N5 O6 S | CCCCNC(=O).... |
112 | 2G26 | - | 3LG | C32 H35 N3 O7 | COc1ccccc1.... |
113 | 4Y6M | - | 48Q | C39 H52 N4 O4 | CCCN(CCC)C.... |
114 | 5YIE | Ki = 5.6 nM | 8VF | C39 H51 N5 O6 S | CCN(CCN)c1.... |
115 | 5YID | Ki = 4 nM | K95 | C37 H44 N4 O6 S2 | CC1([C@H](.... |
116 | 2IGX | - | A1T | C41 H49 N5 O2 | CCCCCc1ccc.... |
117 | 5YIC | Ki = 1.3 nM | 8VO | C37 H45 N5 O6 S2 | CC1([C@H](.... |
118 | 4CKU | ic50 = 0.15 uM | P2F | C38 H52 N4 O6 S | CCCN(CCC)C.... |
119 | 1XDH | - | IVA VAL VAL STA ALA STA | n/a | n/a |
120 | 1LF2 | - | R37 | C32 H41 N3 O4 | Cc1cccc(c1.... |
121 | 5YIB | Ki = 3.3 nM | 8VC | C40 H53 N5 O6 S | Cc1cc(cc(c.... |
122 | 1LEE | - | R36 | C32 H41 N3 O4 | Cc1cccc(c1.... |
123 | 5YIA | Ki = 3 nM | 8V9 | C37 H44 N4 O7 S2 | CC1([C@H](.... |
124 | 1XE5 | - | 5FE | C29 H47 F6 N5 O9 | C[C@@H](C(.... |
125 | 5RBV | - | RQD | C10 H12 F N O2 | COC(=O)[C@.... |
126 | 5RCG | - | REG | C11 H20 N2 O2 | C1CCC(C1)N.... |
127 | 5R1U | - | T9G | C9 H13 N O | CC[C@H](c1.... |
128 | 5RC3 | - | RAY | C11 H14 F N O3 | COCCOCC(=O.... |
129 | 5R21 | - | R9Y | C11 H16 N2 | CN1CCCc2c1.... |
130 | 5RCE | - | RE4 | C11 H13 N5 | Cc1cc(nc(n.... |
131 | 5RBS | - | R8V | C9 H9 N O2 | CN1[C@H](c.... |
132 | 5RBU | - | R97 | C10 H10 N2 S | Cc1csc(n1).... |
133 | 5R2C | - | RE4 | C11 H13 N5 | Cc1cc(nc(n.... |
134 | 5R20 | - | R9V | C14 H19 N O | c1ccc(cc1).... |
135 | 5RCC | - | RDV | C12 H22 N2 O | C1CCC(C1)C.... |
136 | 5RC4 | - | RB7 | C11 H16 Br N O2 S | Cc1cc(ccc1.... |
137 | 5R25 | - | RBJ | C8 H11 N O | CNCc1ccc(c.... |
138 | 5HCT | Ki = 0.0254 uM | 61P | C30 H30 N8 O2 | c1ccc2c(c1.... |
139 | 5R1W | - | R8Y | C10 H13 N O3 S | CCN(CCC(=O.... |
140 | 5R23 | - | RAY | C11 H14 F N O3 | COCCOCC(=O.... |
141 | 5RC5 | - | RBG | C10 H20 N2 O | CC(C)(C)NC.... |
142 | 5RCB | - | RDM | C12 H15 N O3 | CC(=O)N[C@.... |
143 | 5RC6 | - | RBJ | C8 H11 N O | CNCc1ccc(c.... |
144 | 5RBQ | - | R8P | C8 H9 N O3 | C[C@@H](c1.... |
145 | 5R1V | - | R8S | C5 H8 N4 O | COc1ccnc(n.... |
146 | 5R1Z | - | R9M | C6 H7 N O2 S | c1csc(n1)C.... |
147 | 5R2B | - | RDY | C12 H15 N O4 | C[C@@H](C(.... |
148 | 5RC7 | - | AES | C8 H10 F N O2 S | c1cc(ccc1C.... |
149 | 5RBO | - | R8A | C6 H8 N2 O | c1cc(c(nc1.... |
150 | 5R26 | - | RCV | C10 H13 N O3 | COC(=O)COc.... |
151 | 5R1Y | - | R9J | C11 H15 N O2 | Cc1ccc(cc1.... |
152 | 5RBZ | - | R9S | C9 H11 N O | Cc1ccccc1C.... |
153 | 5R1X | - | RQD | C10 H12 F N O2 | COC(=O)[C@.... |
154 | 5RC8 | - | RCV | C10 H13 N O3 | COC(=O)COc.... |
155 | 5RC9 | - | RD4 | C9 H12 N2 O | [H]/N=C(c1.... |
156 | 5RBY | - | R9M | C6 H7 N O2 S | c1csc(n1)C.... |
157 | 5RCF | - | RE7 | C13 H16 F N3 | C[C@H](c1c.... |
158 | 5R24 | - | RB7 | C11 H16 Br N O2 S | Cc1cc(ccc1.... |
159 | 5R28 | - | RDJ | C9 H15 N3 O2 S | CCNC(=O)CS.... |
160 | 5RBT | - | RA7 | C8 H12 N2 O2 S | c1c(sc(n1).... |
161 | 5RCD | - | RDY | C12 H15 N O4 | C[C@@H](C(.... |
162 | 5RBR | - | R8S | C5 H8 N4 O | COc1ccnc(n.... |
163 | 5R2D | - | REG | C11 H20 N2 O2 | C1CCC(C1)N.... |
164 | 5RC0 | - | R9V | C14 H19 N O | c1ccc(cc1).... |
165 | 5R29 | - | RDM | C12 H15 N O3 | CC(=O)N[C@.... |
166 | 5R1T | - | R8A | C6 H8 N2 O | c1cc(c(nc1.... |
167 | 5R2A | - | RDV | C12 H22 N2 O | C1CCC(C1)C.... |
168 | 5R27 | - | RD4 | C9 H12 N2 O | [H]/N=C(c1.... |
169 | 5RBX | - | R9J | C11 H15 N O2 | Cc1ccc(cc1.... |
170 | 5RC1 | - | R9Y | C11 H16 N2 | CN1CCCc2c1.... |
171 | 5RCA | - | RDJ | C9 H15 N3 O2 S | CCNC(=O)CS.... |
172 | 5R22 | - | RA7 | C8 H12 N2 O2 S | c1c(sc(n1).... |
173 | 5RC2 | - | R8Y | C10 H13 N O3 S | CCN(CCC(=O.... |
174 | 5RBW | - | R9G | C12 H15 N O2 | COc1cccc(c.... |
175 | 5RBP | - | SYG | C9 H13 N O | CC[C@@H](c.... |
176 | 1PPM | Ki = 1600 nM | 0P1 | C29 H40 N3 O9 P | C[C@@H](C(.... |
177 | 2WED | Ki = 0.8 uM | PP6 | C29 H32 N2 O7 P | CC(C)[C@H].... |
178 | 1APU | Ki = 1.6 nM | IVA VAL VAL 32L | n/a | n/a |
179 | 2WEC | Ki = 110 uM | PP5 | C28 H32 N2 O7 P | CC(C)[C@@H.... |
180 | 1APW | Ki = 10 nM | IVA VAL VAL DFI NME | n/a | n/a |
181 | 1PPL | Ki = 2.8 nM | 1Z7 | C30 H50 N3 O8 P | CC(C)C[C@H.... |
182 | 2WEB | Ki = 7.6 uM | PP4 | C28 H32 N2 O7 P | CC(C)[C@@H.... |
183 | 2WEA | - | PP6 | C29 H32 N2 O7 P | CC(C)[C@H].... |
184 | 1BXO | Ki = 0.1 nM | PP7 | C30 H47 N4 O9 P | CC(C)C[C@@.... |
185 | 1APT | - | IVA VAL VAL LTA | n/a | n/a |
186 | 1PPK | Ki = 22 nM | IVV | C24 H46 N3 O7 P | CCOC(=O)C[.... |
187 | 1BXQ | Ki = 42 nM | PP8 | C29 H47 N4 O9 P | CC(C)C[C@H.... |
188 | 1APV | Ki = 1 nM | IVA VAL VAL DFO NME | n/a | n/a |
189 | 1SMR | - | PIV HIS PRO PHE HIS LPL TYR TYR SER | n/a | n/a |
190 | 1QRP | - | HH0 | C36 H60 N5 O10 P | C[C@@H](C(.... |
191 | 1PSO | - | IVA VAL VAL STA ALA STA | n/a | n/a |
192 | 2QZX | ic50 = 6 nM | IVA VAL VAL STA ALA STA | n/a | n/a |
193 | 2JXR | Ki = 90 nM | 2Z3 | C32 H49 F2 N5 O7 | NULL |
194 | 1FQ5 | Ki = 4 nM | 0GM | C51 H61 N5 O6 | CC(C)C[C@H.... |
195 | 1QS8 | - | IVA VAL VAL STA ALA STA | n/a | n/a |
196 | 1ZAP | Ki = 0.17 nM | A70 | C42 H70 N6 O5 | CCCC[C@@H].... |
197 | 1IZE | - | IVA VAL VAL STA ALA STA | n/a | n/a |
198 | 1WKR | - | IVA VAL VAL STA ALA STA | n/a | n/a |
199 | 5N7Q | - | IVA VAL VAL STA ALA STA | n/a | n/a |
200 | 5N70 | Kd ~ 3 nM | ALA PHE ARG ILE PRO LEU THR ARG | n/a | n/a |
201 | 3EMY | - | IVA VAL VAL STA ALA STA | n/a | n/a |
202 | 2H6T | Ki = 60 nM | IVA VAL VAL STA ALA STA | n/a | n/a |
203 | 3FV3 | Ki = 0.3 nM | IVA VAL VAL STA ALA STA | n/a | n/a |
204 | 3QVI | - | K95 | C37 H44 N4 O6 S2 | CC1([C@H](.... |
205 | 3APR | - | DHI PRO PHE HIS PUK VAL TYR | n/a | n/a |
206 | 6APR | Ki < 17 nM | IVA VAL VAL STA ALA STA | n/a | n/a |
207 | 5APR | Ki < 17 nM | HIS PRO PHE CYS STA LEU PHE DHL | n/a | n/a |
208 | 4APR | Ki = 200 nM | IVA HIS PRO PHE HIS STA LEU PHE | n/a | n/a |
209 | 1CZI | - | PRO PHI SMC NOR | n/a | n/a |
No: | Ligand | Similarity coefficient |
---|---|---|
1 | LEU | 0.9596 |
2 | LMR | 0.9576 |
3 | CMS | 0.9553 |
4 | JYD | 0.9543 |
5 | ASN | 0.9519 |
6 | ASP | 0.9517 |
7 | MLA | 0.9512 |
8 | MLI | 0.9501 |
9 | COI | 0.9495 |
10 | P2D | 0.9493 |
11 | MLT | 0.9477 |
12 | IVA | 0.9463 |
13 | DMG | 0.9456 |
14 | 1SP | 0.9445 |
15 | 3HL | 0.9436 |
16 | AAE | 0.9428 |
17 | KG7 | 0.9407 |
18 | IHG | 0.9371 |
19 | CIZ | 0.9368 |
20 | SGL | 0.9358 |
21 | DPR | 0.9357 |
22 | 2PC | 0.9357 |
23 | PRO | 0.9356 |
24 | ITN | 0.9346 |
25 | 60P | 0.9337 |
26 | CRN | 0.9336 |
27 | XLS | 0.9328 |
28 | FW5 | 0.9328 |
29 | 23W | 0.9326 |
30 | C5J | 0.9322 |
31 | IOM | 0.9321 |
32 | 2KT | 0.9320 |
33 | MLM | 0.9319 |
34 | 3PY | 0.9307 |
35 | 98J | 0.9306 |
36 | ODV | 0.9294 |
37 | SSN | 0.9280 |
38 | 6PC | 0.9279 |
39 | T2C | 0.9276 |
40 | OAA | 0.9276 |
41 | 273 | 0.9275 |
42 | IPU | 0.9270 |
43 | HZP | 0.9269 |
44 | PYC | 0.9268 |
45 | XBT | 0.9266 |
46 | 3HR | 0.9259 |
47 | ROR | 0.9256 |
48 | HDA | 0.9253 |
49 | HSE | 0.9252 |
50 | BEN | 0.9249 |
51 | MLE | 0.9243 |
52 | 5AC | 0.9239 |
53 | 40E | 0.9236 |
54 | MRY | 0.9230 |
55 | LLQ | 0.9229 |
56 | PZA | 0.9215 |
57 | SS2 | 0.9215 |
58 | BEZ | 0.9212 |
59 | FQI | 0.9209 |
60 | GAG | 0.9208 |
61 | 2RA | 0.9207 |
62 | CYS | 0.9206 |
63 | S0H | 0.9200 |
64 | NCA | 0.9200 |
65 | PBC | 0.9199 |
66 | BAM | 0.9198 |
67 | A3B | 0.9194 |
68 | PRS | 0.9193 |
69 | THE | 0.9193 |
70 | PG3 | 0.9190 |
71 | ABU | 0.9189 |
72 | DSN | 0.9183 |
73 | ILE | 0.9177 |
74 | NIO | 0.9172 |
75 | LEA | 0.9172 |
76 | HY3 | 0.9172 |
77 | TFB | 0.9165 |
78 | LER | 0.9162 |
79 | DTL | 0.9154 |
80 | AL0 | 0.9152 |
81 | MPD | 0.9151 |
82 | YCP | 0.9150 |
83 | UY7 | 0.9148 |
84 | GBD | 0.9148 |
85 | TB6 | 0.9148 |
86 | HCS | 0.9144 |
87 | FOA | 0.9144 |
88 | KIV | 0.9143 |
89 | 2RH | 0.9142 |
90 | BAL | 0.9142 |
91 | UGC | 0.9140 |
92 | JZ5 | 0.9136 |
93 | FUM | 0.9136 |
94 | BXO | 0.9135 |
95 | SER | 0.9135 |
96 | OXQ | 0.9133 |
97 | ABA | 0.9126 |
98 | TAR | 0.9124 |
99 | 2AS | 0.9122 |
100 | SIN | 0.9121 |
101 | TP5 | 0.9120 |
102 | THR | 0.9110 |
103 | UYA | 0.9108 |
104 | G2H | 0.9107 |
105 | ORN | 0.9100 |
106 | VAH | 0.9099 |
107 | GLY CYS | 0.9096 |
108 | HV2 | 0.9093 |
109 | BNS | 0.9091 |
110 | 9YL | 0.9091 |
111 | PAE | 0.9090 |
112 | GLY ALA | 0.9090 |
113 | TZE | 0.9086 |
114 | BU4 | 0.9085 |
115 | DXX | 0.9083 |
116 | XUL | 0.9082 |
117 | C21 | 0.9082 |
118 | SAL | 0.9076 |
119 | C2N | 0.9069 |
120 | O7U | 0.9066 |
121 | CP | 0.9064 |
122 | VAL | 0.9058 |
123 | TZL | 0.9055 |
124 | ZBT | 0.9055 |
125 | HYP | 0.9054 |
126 | MEV | 0.9052 |
127 | 51F | 0.9047 |
128 | NXA | 0.9047 |
129 | FCN | 0.9045 |
130 | AHB | 0.9045 |
131 | SHF | 0.9041 |
132 | AOA | 0.9041 |
133 | PPV | 0.9039 |
134 | TEO | 0.9034 |
135 | 7VD | 0.9031 |
136 | KPL | 0.9027 |
137 | SC2 | 0.9026 |
138 | FBJ | 0.9025 |
139 | GLU | 0.9022 |
140 | NVA | 0.9020 |
141 | PEP | 0.9017 |
142 | 54D | 0.9016 |
143 | BVC | 0.9015 |
144 | DPF | 0.9014 |
145 | DAS | 0.9012 |
146 | PZI | 0.9012 |
147 | BMD | 0.9006 |
148 | PYJ | 0.9002 |
149 | 7WG | 0.9001 |
150 | BUA | 0.9001 |
151 | PEQ | 0.8997 |
152 | 8X3 | 0.8997 |
153 | DBB | 0.8996 |
154 | APY | 0.8994 |
155 | 4MV | 0.8994 |
156 | PCT | 0.8993 |
157 | DGY | 0.8993 |
158 | 2PN | 0.8991 |
159 | SAT | 0.8991 |
160 | ALO | 0.8989 |
161 | SS1 | 0.8988 |
162 | QSC | 0.8984 |
163 | 2HE | 0.8984 |
164 | OEM | 0.8983 |
165 | RBL | 0.8980 |
166 | PCA | 0.8977 |
167 | GG6 | 0.8973 |
168 | HYA | 0.8971 |
169 | EGD | 0.8970 |
170 | MAE | 0.8970 |
171 | ABN | 0.8970 |
172 | MET | 0.8969 |
173 | 1DQ | 0.8969 |
174 | RB0 | 0.8969 |
175 | RB5 | 0.8969 |
176 | XYL | 0.8969 |
177 | POA | 0.8959 |
178 | OPE | 0.8958 |
179 | IT2 | 0.8956 |
180 | HVQ | 0.8955 |
181 | M58 | 0.8955 |
182 | MZ0 | 0.8955 |
183 | SYN | 0.8954 |
184 | B24 | 0.8952 |
185 | NMG | 0.8949 |
186 | 1DU | 0.8948 |
187 | BUB | 0.8946 |
188 | GZ3 | 0.8945 |
189 | 3BB | 0.8944 |
190 | POP | 0.8944 |
191 | HX2 | 0.8939 |
192 | DCY | 0.8939 |
193 | 3SL | 0.8938 |
194 | PGA | 0.8938 |
195 | HBX | 0.8930 |
196 | PIS | 0.8930 |
197 | CHT | 0.8928 |
198 | PPR | 0.8927 |
199 | R67 | 0.8927 |
200 | ES6 | 0.8927 |
201 | PRI | 0.8925 |
202 | GLN | 0.8925 |
203 | DE2 | 0.8922 |
204 | 2EH | 0.8919 |
205 | PUT | 0.8918 |
206 | MSF | 0.8916 |
207 | OHG | 0.8912 |
208 | VX | 0.8912 |
209 | JBN | 0.8912 |
210 | BTL | 0.8910 |
211 | SKG | 0.8909 |
212 | 9CL | 0.8906 |
213 | ISZ | 0.8905 |
214 | AC5 | 0.8904 |
215 | GXV | 0.8896 |
216 | SAR | 0.8894 |
217 | 0V5 | 0.8894 |
218 | PE9 | 0.8894 |
219 | ETM | 0.8892 |
220 | HIU | 0.8891 |
221 | PPF | 0.8891 |
222 | P7I | 0.8887 |
223 | FJO | 0.8886 |
224 | BHO | 0.8885 |
225 | XPO | 0.8884 |
226 | HIO | 0.8883 |
227 | BVG | 0.8882 |
228 | 03W | 0.8881 |
229 | HPY | 0.8878 |
230 | COM | 0.8878 |
231 | SPV | 0.8874 |
232 | HL5 | 0.8873 |
233 | NVI | 0.8873 |
234 | PLU | 0.8870 |
235 | FEH | 0.8870 |
236 | 2EZ | 0.8867 |
237 | AMC | 0.8865 |
238 | CSS | 0.8861 |
239 | SRT | 0.8860 |
240 | FPI | 0.8859 |
241 | SMB | 0.8857 |
242 | PAF | 0.8857 |
243 | DSS | 0.8856 |
244 | 4SD | 0.8856 |
245 | ETX | 0.8851 |
246 | 69O | 0.8851 |
247 | 1GP | 0.8848 |
248 | 9X7 | 0.8846 |
249 | 2PG | 0.8845 |
250 | 3GR | 0.8843 |
251 | TAU | 0.8842 |
252 | HSM | 0.8839 |
253 | 3U4 | 0.8836 |
254 | H95 | 0.8836 |
255 | NIZ | 0.8829 |
256 | PBE | 0.8825 |
257 | 6JN | 0.8822 |
258 | FBM | 0.8822 |
259 | FLA | 0.8821 |
260 | PAH | 0.8820 |
261 | MRZ | 0.8820 |
262 | JKE | 0.8818 |
263 | IP0 | 0.8817 |
264 | 4CS | 0.8813 |
265 | ITU | 0.8813 |
266 | ONL | 0.8811 |
267 | G3H | 0.8809 |
268 | G3P | 0.8809 |
269 | CFI | 0.8808 |
270 | AML | 0.8807 |
271 | NLE | 0.8806 |
272 | 4HA | 0.8804 |
273 | HIS | 0.8804 |
274 | QFH | 0.8803 |
275 | DTU | 0.8802 |
276 | AKB | 0.8802 |
277 | AC0 | 0.8802 |
278 | XAP | 0.8801 |
279 | ACH | 0.8799 |
280 | DAB | 0.8798 |
281 | XSP | 0.8796 |
282 | FSG | 0.8794 |
283 | IZC | 0.8792 |
284 | 1MR | 0.8792 |
285 | 192 | 0.8790 |
286 | 1P3 | 0.8790 |
287 | F9P | 0.8789 |
288 | URP | 0.8784 |
289 | TLA | 0.8783 |
290 | CXF | 0.8781 |
291 | IQ0 | 0.8776 |
292 | BP9 | 0.8776 |
293 | MTG | 0.8772 |
294 | DAL | 0.8770 |
295 | HY1 | 0.8768 |
296 | A8C | 0.8766 |
297 | 23B | 0.8754 |
298 | 9SB | 0.8754 |
299 | DPJ | 0.8753 |
300 | 271 | 0.8751 |
301 | 39J | 0.8751 |
302 | JZ7 | 0.8747 |
303 | EFS | 0.8746 |
304 | HTX | 0.8745 |
305 | GOL | 0.8743 |
306 | DMV | 0.8740 |
307 | 13P | 0.8739 |
308 | AG2 | 0.8738 |
309 | 278 | 0.8738 |
310 | MED | 0.8734 |
311 | DYA | 0.8730 |
312 | 6NA | 0.8729 |
313 | PYR | 0.8728 |
314 | DGL | 0.8724 |
315 | 2IT | 0.8724 |
316 | PG0 | 0.8721 |
317 | GGL | 0.8720 |
318 | H3M | 0.8719 |
319 | QDK | 0.8714 |
320 | SLP | 0.8710 |
321 | FPY | 0.8710 |
322 | BAE | 0.8708 |
323 | 1DJ | 0.8708 |
324 | BHH | 0.8705 |
325 | 282 | 0.8704 |
326 | 7N0 | 0.8702 |
327 | RSO | 0.8698 |
328 | DTT | 0.8697 |
329 | WTZ | 0.8694 |
330 | 3SS | 0.8694 |
331 | GUA | 0.8690 |
332 | MDN | 0.8688 |
333 | 9J3 | 0.8684 |
334 | 285 | 0.8680 |
335 | HBR | 0.8670 |
336 | 8EZ | 0.8668 |
337 | YHO | 0.8665 |
338 | 1AC | 0.8665 |
339 | HUI | 0.8659 |
340 | R1X | 0.8654 |
341 | R2B | 0.8654 |
342 | PEL | 0.8646 |
343 | DCD | 0.8643 |
344 | 280 | 0.8640 |
345 | PEA | 0.8639 |
346 | PEZ | 0.8634 |
347 | 8EW | 0.8632 |
348 | MUC | 0.8631 |
349 | ISU | 0.8628 |
350 | ICF | 0.8621 |
351 | LNO | 0.8619 |
352 | SD4 | 0.8618 |
353 | I1E | 0.8610 |
354 | 4SV | 0.8609 |
355 | SYM | 0.8601 |
356 | EDG | 0.8595 |
357 | 3PG | 0.8593 |
358 | 0OC | 0.8593 |
359 | 7WV | 0.8591 |
360 | MNN | 0.8584 |
361 | HBS | 0.8571 |
362 | 9TY | 0.8562 |
363 | M6W | 0.8544 |
364 | KOJ | 0.8539 |
365 | 3V4 | 0.8525 |
366 | DYT | 0.8520 |
This union binding pocket(no: 1) in the query (biounit: 4er2.bio1) has 39 residues | |||
---|---|---|---|
No: | Leader PDB | Ligand | Sequence Similarity |
1 | 1J71 | THR ILE THR SER | 42.4242 |