1
|
1E81
|
- |
M91
|
C34 H49 N5 O6 S
|
CSC[C@@H](....
|
2
|
4ZEA
|
- |
IMI
|
C10 H17 N3 O2 S
|
C1[C@H]2[C....
|
3
|
3ER3
|
Ki
=
81
nM |
0EL
|
C51 H78 N8 O9
|
NULL
|
4
|
4Y4D
|
- |
CFF
|
C8 H10 N4 O2
|
Cn1cnc2c1C....
|
5
|
5LWT
|
- |
7B3
|
C10 H13 N3 O
|
Cc1c2cnnc(....
|
6
|
1EPM
|
- |
THR PHE GLN ALA PSA LEU ARG GLU
|
n/a
|
n/a
|
7
|
1EED
|
Ki
=
16.2
uM |
0EO
|
C34 H55 N3 O8
|
CC(C)C[C@@....
|
8
|
3PMY
|
- |
41L
|
C15 H13 N3 O
|
c1ccc(cc1)....
|
9
|
1OEX
|
- |
BOC HIS PRO PHE ALA LOV ILE HIS
|
n/a
|
n/a
|
10
|
4ER4
|
Ki
=
160
nM |
PRO HIS PRO PHE HIS LAV ILE HIS LYS
|
n/a
|
n/a
|
11
|
4LBT
|
Ki
=
6
uM |
1TZ
|
C21 H24 N4 O
|
Cc1cc(c(c(....
|
12
|
3PWW
|
- |
ROC
|
C38 H50 N6 O5
|
CC(C)(C)NC....
|
13
|
4Y38
|
Kd
=
4
mM |
0A9
|
C10 H13 N O2
|
COC(=O)[C@....
|
14
|
2JJJ
|
- |
0QS
|
C36 H56 F2 N7 O8 S
|
CC(C)(C)S(....
|
15
|
1GVV
|
- |
0GM
|
C51 H61 N5 O6
|
CC(C)C[C@H....
|
16
|
3PMU
|
- |
F7L
|
C14 H20 F N O2
|
c1ccc(c(c1....
|
17
|
5OJE
|
Ki
=
6.1
uM |
VSK
|
C22 H27 N3 O
|
Cc1cc(c(c(....
|
18
|
1GVT
|
- |
2ZS
|
C31 H48 N4 O7 S
|
CC(C)OC(=O....
|
19
|
1EPR
|
- |
0QS
|
C36 H56 F2 N7 O8 S
|
CC(C)(C)S(....
|
20
|
5MB5
|
- |
46P
|
C8 H10 N4 S
|
Cc1c(sc(n1....
|
21
|
5MB7
|
- |
4AV
|
C8 H9 Cl N2 O2
|
CNCc1cc(cc....
|
22
|
4Y4G
|
- |
GGB
|
C5 H12 N4 O3
|
[H]/N=C(N)....
|
23
|
3ER5
|
Ki
=
1
nM |
PRO HIS PRO PHE HIS STA VAL ILE HIS LYS
|
n/a
|
n/a
|
24
|
3URL
|
- |
HIS SER LEU PHE HIS PUK THR PRO
|
n/a
|
n/a
|
25
|
3PCZ
|
- |
BAM
|
C7 H9 N2
|
c1ccc(cc1)....
|
26
|
2V00
|
Kd
=
0.22
mM |
V15
|
C12 H13 N3 O
|
c1ccc(cc1)....
|
27
|
5LWR
|
- |
7B2
|
C27 H29 Cl N9 O
|
Cc1c2cnn3c....
|
28
|
3PLL
|
- |
F06
|
C8 H9 Cl N2 S
|
[H]/N=C(N)....
|
29
|
4ER2
|
Ki
=
0.5
nM |
IVA VAL VAL STA ALA STA
|
n/a
|
n/a
|
30
|
4LP9
|
ic50
=
0.62
uM |
SER LEU PHE HIS 22G THR PRO
|
n/a
|
n/a
|
31
|
3PRS
|
- |
RIT
|
C37 H48 N6 O5 S2
|
CC(C)c1nc(....
|
32
|
1ENT
|
Ki
=
110
nM |
0EM
|
C32 H52 N6 O7 P
|
NULL
|
33
|
1E80
|
- |
0GQ
|
C41 H64 N10 O6
|
CC[C@H](C)....
|
34
|
5LWS
|
- |
7B2
|
C27 H29 Cl N9 O
|
Cc1c2cnn3c....
|
35
|
3PBD
|
- |
F05
|
C8 H8 N2
|
c1ccc2c(c1....
|
36
|
1OD1
|
- |
0QS
|
C36 H56 F2 N7 O8 S
|
CC(C)(C)S(....
|
37
|
3WZ6
|
Ki
=
1.1
uM |
IXZ
|
C27 H25 N3 O2 S
|
c1ccc(cc1)....
|
38
|
5ER1
|
Ki
=
960
nM |
0HT
|
C28 H48 N4 O5
|
CC[C@H](C)....
|
39
|
1OEW
|
- |
SER THR
|
n/a
|
n/a
|
40
|
1EPQ
|
Ki
=
6.5
nM |
0QF
|
C31 H52 N4 O7 S2
|
CCS[C@@H](....
|
41
|
5MB3
|
- |
5GL
|
C13 H20 N2 O S
|
CCCN1C2=C(....
|
42
|
2JJI
|
- |
0QS
|
C36 H56 F2 N7 O8 S
|
CC(C)(C)S(....
|
43
|
3PCW
|
- |
FBF
|
C8 H7 F3 N2
|
[H]/N=C(/c....
|
44
|
3PGI
|
- |
F41
|
C14 H18 N2 O3
|
c1cc2c(cc1....
|
45
|
4Y3J
|
Kd
=
6.8
mM |
HIC
|
C7 H11 N3 O2
|
Cn1cc(nc1)....
|
46
|
1GVW
|
Ki
=
110
nM |
0EM
|
C32 H52 N6 O7 P
|
NULL
|
47
|
5ER2
|
Ki
=
0.27
uM |
0EK
|
C50 H77 N9 O9
|
NULL
|
48
|
1EPP
|
Ki
=
69
nM |
1Z1
|
C32 H57 N7 O6 S2
|
CC[C@H](C)....
|
49
|
2ER7
|
ic50
=
0.7
nM |
BOC HIS PRO PHE HIS LOV ILE HIS
|
n/a
|
n/a
|
50
|
4KUP
|
Ki
=
6
uM |
1TZ
|
C21 H24 N4 O
|
Cc1cc(c(c(....
|
51
|
3WZ7
|
Ki
=
1.8
uM |
IXY
|
C28 H30 N4 O2 S
|
c1ccc(cc1)....
|
52
|
1EPO
|
Ki
=
11
nM |
2Z3
|
C32 H49 F2 N5 O7
|
NULL
|
53
|
1ER8
|
- |
DHI PRO PHE HIS LEU LEU VAL TYR
|
n/a
|
n/a
|
54
|
3WZ8
|
Ki
=
1.5
uM |
IXV
|
C27 H25 N3 O2 S
|
c1ccc(cc1)....
|
55
|
3PI0
|
- |
F91
|
C14 H14 N2 O2
|
c1cc2c(cc1....
|
56
|
1GVU
|
Ki
=
1
nM |
PRO HIS PRO PHE HIS STA VAL ILE HIS LYS
|
n/a
|
n/a
|
57
|
1EPL
|
- |
PRO LEU GLU PSA ARG LEU
|
n/a
|
n/a
|
58
|
4Y3Y
|
Kd
=
4.5
mM |
DCL
|
C6 H15 N O
|
CC(C)C[C@@....
|
59
|
1E5O
|
- |
3AI
|
C23 H38 N4 O4 S
|
CC[C@H](C)....
|
60
|
3PLD
|
- |
F90
|
C8 H9 Cl N2 S
|
[H]/N=C(N)....
|
61
|
5MB0
|
Kd
=
1.4
mM |
F91
|
C14 H14 N2 O2
|
c1cc2c(cc1....
|
62
|
2ER6
|
Ki
=
60
nM |
PRO THR GLU PUK ARG GLU
|
n/a
|
n/a
|
63
|
3URI
|
- |
HIS PRO HIS LEU SER 13E ALA HIS
|
n/a
|
n/a
|
64
|
4LHH
|
Ki
=
6
uM |
1TZ
|
C21 H24 N4 O
|
Cc1cc(c(c(....
|
65
|
4Y48
|
- |
GLY PRO
|
n/a
|
n/a
|
66
|
1E82
|
- |
M90
|
C34 H49 N5 O6 S
|
CSC[C@@H](....
|
67
|
1EPN
|
- |
2ZS
|
C31 H48 N4 O7 S
|
CC(C)OC(=O....
|
68
|
2ER9
|
Ki
=
40
nM |
BOC HIS PRO PHE HIS STA LEU PHE
|
n/a
|
n/a
|
69
|
4Y4J
|
Kd
=
3.4
mM |
LNR
|
C8 H11 N O3
|
c1cc(c(cc1....
|
70
|
1GVX
|
Ki
=
60
nM |
PRO THR GLU PUK ARG GLU
|
n/a
|
n/a
|
71
|
3PM4
|
- |
F5N
|
C15 H13 N3 O
|
c1ccc(cc1)....
|
72
|
3PB5
|
- |
F63
|
C11 H12 N2 O2
|
CNCc1ccc(o....
|
73
|
4ZE6
|
Kd
=
3.3
mM |
011
|
C7 H15 N O2
|
C(CCCN)CCC....
|
74
|
3PBZ
|
- |
F02
|
C11 H17 N3 O
|
CCN(CC)c1c....
|
75
|
4ER1
|
Ki
=
0.24
uM |
0ZP
|
C51 H68 N5 O4
|
CC[C@H](C)....
|
76
|
3OWN
|
Ki
=
34
nM |
3OX
|
C37 H48 N4 O7 S
|
CC(C)CNC(=....
|
77
|
2G21
|
- |
L1B
|
C19 H24 N5 O
|
CCc1c(c(nc....
|
78
|
4RYC
|
ic50
=
0.08
uM |
3ZK
|
C27 H39 N3 O6 S
|
Cc1ccc(cc1....
|
79
|
3D91
|
Kd
=
131
pM |
REM
|
C33 H50 N4 O6 S
|
CC(C)(C)S(....
|
80
|
1BIL
|
ic50
=
0.5
nM |
0IU
|
C34 H53 N5 O5 S
|
NULL
|
81
|
3KM4
|
ic50
=
1.3
nM |
22X
|
C28 H45 Cl N4 O3
|
CC(=O)NCCC....
|
82
|
2G24
|
- |
7IG
|
C19 H19 F2 N5
|
CCc1c(c(nc....
|
83
|
2IL2
|
Kd
=
79
nM |
LIX
|
C32 H38 N6 O5 S
|
CCc1c(c(nc....
|
84
|
5SY3
|
ic50
=
43
uM |
74Z
|
C15 H15 N3 O S
|
c1cc(oc1)C....
|
85
|
4Q1N
|
ic50
=
0.2
nM |
2Y9
|
C26 H42 N4 O4
|
CCOC[C@@H]....
|
86
|
2I4Q
|
ic50
=
0.007
uM |
UA4
|
C25 H27 F2 N5 O3
|
CCc1c(c(nc....
|
87
|
2BKS
|
ic50
=
37
nM |
PZ1
|
C34 H41 N3 O6
|
COc1ccccc1....
|
88
|
4S1G
|
Ki
=
0.6
nM |
43T
|
C24 H29 F N4 O2
|
C[C@@H](c1....
|
89
|
4XX3
|
Ki
=
56
nM |
70X
|
C23 H28 N4 O2
|
[H]/N=C1/N....
|
90
|
2G1S
|
- |
4IG
|
C24 H25 F2 N5 O3
|
CCc1c(c(nc....
|
91
|
2G20
|
- |
L1A
|
C33 H50 N6 O7 S2
|
CC(C)C[C@@....
|
92
|
5SXN
|
ic50
=
11
uM |
74U
|
C19 H15 N3 O
|
c1ccc(cc1)....
|
93
|
3G70
|
ic50
=
0.4
nM |
A5T
|
C33 H32 Cl3 F2 N3 O2
|
c1cc(c(c(c....
|
94
|
2G1Y
|
- |
5IG
|
C20 H27 N5 O3
|
CCc1c(c(nc....
|
95
|
2G1R
|
- |
3IG
|
C20 H26 N6 O3
|
CCc1c(c(nc....
|
96
|
4GJC
|
ic50
=
0.09
uM |
0MJ
|
C27 H29 N3 O4 S
|
Cc1ccc(cc1....
|
97
|
4GJ8
|
- |
0LW
|
C20 H23 N O S
|
c1ccc2c(c1....
|
98
|
5SY2
|
ic50
=
11
uM |
74V
|
C18 H25 N5 O2
|
CCN([C@H]1....
|
99
|
5KOS
|
ic50
=
1.5
nM |
6VS
|
C27 H46 N6 O4
|
CC(C)CN([C....
|
100
|
3G72
|
ic50
=
0.8
nM |
A6T
|
C33 H32 Cl3 F2 N3 O2
|
c1cc(c(c(c....
|
101
|
3G6Z
|
ic50
=
0.2
nM |
A7T
|
C35 H39 Cl2 N3 O3
|
Cc1cccc(c1....
|
102
|
3GW5
|
ic50
=
0.47
nM |
72X
|
C28 H46 Cl N3 O3
|
CNC[C@H](C....
|
103
|
3SFC
|
ic50
=
0.003
uM |
S53
|
C32 H29 F N4 O2
|
Cc1ccc(cc1....
|
104
|
2IKO
|
Kd
=
3571
nM |
7IG
|
C19 H19 F2 N5
|
CCc1c(c(nc....
|
105
|
3K1W
|
- |
BFX
|
C31 H31 Br Cl F N2 O2
|
c1ccc(c(c1....
|
106
|
4XX4
|
Ki
=
44
nM |
70Y
|
C25 H30 N4 O2
|
[H]/N=C1/N....
|
107
|
2FS4
|
ic50
=
37
nM |
PZ1
|
C34 H41 N3 O6
|
COc1ccccc1....
|
108
|
2BKT
|
ic50
=
23
nM |
RPF
|
C31 H37 N3 O5
|
COc1ccccc1....
|
109
|
4GJ5
|
- |
0LR
|
C22 H23 N O
|
c1ccc(cc1)....
|
110
|
2G22
|
- |
6IG
|
C27 H35 N5 O
|
CCc1c(c(nc....
|
111
|
1RNE
|
ic50
=
2
nM |
C60
|
C39 H63 N5 O6 S
|
CCCCNC(=O)....
|
112
|
2G26
|
- |
3LG
|
C32 H35 N3 O7
|
COc1ccccc1....
|
113
|
4Y6M
|
- |
48Q
|
C39 H52 N4 O4
|
CCCN(CCC)C....
|
114
|
5YIE
|
Ki
=
5.6
nM |
8VF
|
C39 H51 N5 O6 S
|
CCN(CCN)c1....
|
115
|
5YID
|
Ki
=
4
nM |
K95
|
C37 H44 N4 O6 S2
|
CC1([C@H](....
|
116
|
2IGX
|
- |
A1T
|
C41 H49 N5 O2
|
CCCCCc1ccc....
|
117
|
5YIC
|
Ki
=
1.3
nM |
8VO
|
C37 H45 N5 O6 S2
|
CC1([C@H](....
|
118
|
4CKU
|
ic50
=
0.15
uM |
P2F
|
C38 H52 N4 O6 S
|
CCCN(CCC)C....
|
119
|
1XDH
|
- |
IVA VAL VAL STA ALA STA
|
n/a
|
n/a
|
120
|
1LF2
|
- |
R37
|
C32 H41 N3 O4
|
Cc1cccc(c1....
|
121
|
5YIB
|
Ki
=
3.3
nM |
8VC
|
C40 H53 N5 O6 S
|
Cc1cc(cc(c....
|
122
|
1LEE
|
- |
R36
|
C32 H41 N3 O4
|
Cc1cccc(c1....
|
123
|
5YIA
|
Ki
=
3
nM |
8V9
|
C37 H44 N4 O7 S2
|
CC1([C@H](....
|
124
|
1XE5
|
- |
5FE
|
C29 H47 F6 N5 O9
|
C[C@@H](C(....
|
125
|
5RBV
|
- |
RQD
|
C10 H12 F N O2
|
COC(=O)[C@....
|
126
|
5RCG
|
- |
REG
|
C11 H20 N2 O2
|
C1CCC(C1)N....
|
127
|
5R1U
|
- |
T9G
|
C9 H13 N O
|
CC[C@H](c1....
|
128
|
5RC3
|
- |
RAY
|
C11 H14 F N O3
|
COCCOCC(=O....
|
129
|
5R21
|
- |
R9Y
|
C11 H16 N2
|
CN1CCCc2c1....
|
130
|
5RCE
|
- |
RE4
|
C11 H13 N5
|
Cc1cc(nc(n....
|
131
|
5RBS
|
- |
R8V
|
C9 H9 N O2
|
CN1[C@H](c....
|
132
|
5RBU
|
- |
R97
|
C10 H10 N2 S
|
Cc1csc(n1)....
|
133
|
5R2C
|
- |
RE4
|
C11 H13 N5
|
Cc1cc(nc(n....
|
134
|
5R20
|
- |
R9V
|
C14 H19 N O
|
c1ccc(cc1)....
|
135
|
5RCC
|
- |
RDV
|
C12 H22 N2 O
|
C1CCC(C1)C....
|
136
|
5RC4
|
- |
RB7
|
C11 H16 Br N O2 S
|
Cc1cc(ccc1....
|
137
|
5R25
|
- |
RBJ
|
C8 H11 N O
|
CNCc1ccc(c....
|
138
|
5HCT
|
Ki
=
0.0254
uM |
61P
|
C30 H30 N8 O2
|
c1ccc2c(c1....
|
139
|
5R1W
|
- |
R8Y
|
C10 H13 N O3 S
|
CCN(CCC(=O....
|
140
|
5R23
|
- |
RAY
|
C11 H14 F N O3
|
COCCOCC(=O....
|
141
|
5RC5
|
- |
RBG
|
C10 H20 N2 O
|
CC(C)(C)NC....
|
142
|
5RCB
|
- |
RDM
|
C12 H15 N O3
|
CC(=O)N[C@....
|
143
|
5RC6
|
- |
RBJ
|
C8 H11 N O
|
CNCc1ccc(c....
|
144
|
5RBQ
|
- |
R8P
|
C8 H9 N O3
|
C[C@@H](c1....
|
145
|
5R1V
|
- |
R8S
|
C5 H8 N4 O
|
COc1ccnc(n....
|
146
|
5R1Z
|
- |
R9M
|
C6 H7 N O2 S
|
c1csc(n1)C....
|
147
|
5R2B
|
- |
RDY
|
C12 H15 N O4
|
C[C@@H](C(....
|
148
|
5RC7
|
- |
AES
|
C8 H10 F N O2 S
|
c1cc(ccc1C....
|
149
|
5RBO
|
- |
R8A
|
C6 H8 N2 O
|
c1cc(c(nc1....
|
150
|
5R26
|
- |
RCV
|
C10 H13 N O3
|
COC(=O)COc....
|
151
|
5R1Y
|
- |
R9J
|
C11 H15 N O2
|
Cc1ccc(cc1....
|
152
|
5RBZ
|
- |
R9S
|
C9 H11 N O
|
Cc1ccccc1C....
|
153
|
5R1X
|
- |
RQD
|
C10 H12 F N O2
|
COC(=O)[C@....
|
154
|
5RC8
|
- |
RCV
|
C10 H13 N O3
|
COC(=O)COc....
|
155
|
5RC9
|
- |
RD4
|
C9 H12 N2 O
|
[H]/N=C(c1....
|
156
|
5RBY
|
- |
R9M
|
C6 H7 N O2 S
|
c1csc(n1)C....
|
157
|
5RCF
|
- |
RE7
|
C13 H16 F N3
|
C[C@H](c1c....
|
158
|
5R24
|
- |
RB7
|
C11 H16 Br N O2 S
|
Cc1cc(ccc1....
|
159
|
5R28
|
- |
RDJ
|
C9 H15 N3 O2 S
|
CCNC(=O)CS....
|
160
|
5RBT
|
- |
RA7
|
C8 H12 N2 O2 S
|
c1c(sc(n1)....
|
161
|
5RCD
|
- |
RDY
|
C12 H15 N O4
|
C[C@@H](C(....
|
162
|
5RBR
|
- |
R8S
|
C5 H8 N4 O
|
COc1ccnc(n....
|
163
|
5R2D
|
- |
REG
|
C11 H20 N2 O2
|
C1CCC(C1)N....
|
164
|
5RC0
|
- |
R9V
|
C14 H19 N O
|
c1ccc(cc1)....
|
165
|
5R29
|
- |
RDM
|
C12 H15 N O3
|
CC(=O)N[C@....
|
166
|
5R1T
|
- |
R8A
|
C6 H8 N2 O
|
c1cc(c(nc1....
|
167
|
5R2A
|
- |
RDV
|
C12 H22 N2 O
|
C1CCC(C1)C....
|
168
|
5R27
|
- |
RD4
|
C9 H12 N2 O
|
[H]/N=C(c1....
|
169
|
5RBX
|
- |
R9J
|
C11 H15 N O2
|
Cc1ccc(cc1....
|
170
|
5RC1
|
- |
R9Y
|
C11 H16 N2
|
CN1CCCc2c1....
|
171
|
5RCA
|
- |
RDJ
|
C9 H15 N3 O2 S
|
CCNC(=O)CS....
|
172
|
5R22
|
- |
RA7
|
C8 H12 N2 O2 S
|
c1c(sc(n1)....
|
173
|
5RC2
|
- |
R8Y
|
C10 H13 N O3 S
|
CCN(CCC(=O....
|
174
|
5RBW
|
- |
R9G
|
C12 H15 N O2
|
COc1cccc(c....
|
175
|
5RBP
|
- |
SYG
|
C9 H13 N O
|
CC[C@@H](c....
|
176
|
1PPM
|
Ki
=
1600
nM |
0P1
|
C29 H40 N3 O9 P
|
C[C@@H](C(....
|
177
|
2WED
|
Ki
=
0.8
uM |
PP6
|
C29 H32 N2 O7 P
|
CC(C)[C@H]....
|
178
|
1APU
|
Ki
=
1.6
nM |
IVA VAL VAL 32L
|
n/a
|
n/a
|
179
|
2WEC
|
Ki
=
110
uM |
PP5
|
C28 H32 N2 O7 P
|
CC(C)[C@@H....
|
180
|
1APW
|
Ki
=
10
nM |
IVA VAL VAL DFI NME
|
n/a
|
n/a
|
181
|
1PPL
|
Ki
=
2.8
nM |
1Z7
|
C30 H50 N3 O8 P
|
CC(C)C[C@H....
|
182
|
2WEB
|
Ki
=
7.6
uM |
PP4
|
C28 H32 N2 O7 P
|
CC(C)[C@@H....
|
183
|
2WEA
|
- |
PP6
|
C29 H32 N2 O7 P
|
CC(C)[C@H]....
|
184
|
1BXO
|
Ki
=
0.1
nM |
PP7
|
C30 H47 N4 O9 P
|
CC(C)C[C@@....
|
185
|
1APT
|
- |
IVA VAL VAL LTA
|
n/a
|
n/a
|
186
|
1PPK
|
Ki
=
22
nM |
IVV
|
C24 H46 N3 O7 P
|
CCOC(=O)C[....
|
187
|
1BXQ
|
Ki
=
42
nM |
PP8
|
C29 H47 N4 O9 P
|
CC(C)C[C@H....
|
188
|
1APV
|
Ki
=
1
nM |
IVA VAL VAL DFO NME
|
n/a
|
n/a
|
189
|
1SMR
|
- |
PIV HIS PRO PHE HIS LPL TYR TYR SER
|
n/a
|
n/a
|
190
|
1QRP
|
- |
HH0
|
C36 H60 N5 O10 P
|
C[C@@H](C(....
|
191
|
1PSO
|
- |
IVA VAL VAL STA ALA STA
|
n/a
|
n/a
|
192
|
2QZX
|
ic50
=
6
nM |
IVA VAL VAL STA ALA STA
|
n/a
|
n/a
|
193
|
2JXR
|
Ki
=
90
nM |
2Z3
|
C32 H49 F2 N5 O7
|
NULL
|
194
|
1FQ5
|
Ki
=
4
nM |
0GM
|
C51 H61 N5 O6
|
CC(C)C[C@H....
|
195
|
1QS8
|
- |
IVA VAL VAL STA ALA STA
|
n/a
|
n/a
|
196
|
1ZAP
|
Ki
=
0.17
nM |
A70
|
C42 H70 N6 O5
|
CCCC[C@@H]....
|
197
|
1IZE
|
- |
IVA VAL VAL STA ALA STA
|
n/a
|
n/a
|
198
|
1WKR
|
- |
IVA VAL VAL STA ALA STA
|
n/a
|
n/a
|
199
|
5N7Q
|
- |
IVA VAL VAL STA ALA STA
|
n/a
|
n/a
|
200
|
5N70
|
Kd
~
3
nM |
ALA PHE ARG ILE PRO LEU THR ARG
|
n/a
|
n/a
|
201
|
3EMY
|
- |
IVA VAL VAL STA ALA STA
|
n/a
|
n/a
|
202
|
2H6T
|
Ki
=
60
nM |
IVA VAL VAL STA ALA STA
|
n/a
|
n/a
|
203
|
3FV3
|
Ki
=
0.3
nM |
IVA VAL VAL STA ALA STA
|
n/a
|
n/a
|
204
|
3QVI
|
- |
K95
|
C37 H44 N4 O6 S2
|
CC1([C@H](....
|
205
|
3APR
|
- |
DHI PRO PHE HIS PUK VAL TYR
|
n/a
|
n/a
|
206
|
6APR
|
Ki
<
17
nM |
IVA VAL VAL STA ALA STA
|
n/a
|
n/a
|
207
|
5APR
|
Ki
<
17
nM |
HIS PRO PHE CYS STA LEU PHE DHL
|
n/a
|
n/a
|
208
|
4APR
|
Ki
=
200
nM |
IVA HIS PRO PHE HIS STA LEU PHE
|
n/a
|
n/a
|
209
|
1CZI
|
- |
PRO PHI SMC NOR
|
n/a
|
n/a
|