Searching for Source: 'HUMAN IMMUNODEFICIENCY VIRUS 1';
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Molecular Weight (Da)
3UCB 1.38 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 017 Kd = 41 nM 547.664
4LL3 1.95 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 017 Kd = 2.7 pM 547.664
4NJT 1.95 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME HYDROLASES 017 547.664
5KQY 1.65 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 017 Ki = 0.51 nM 547.664
5KR1 1.6 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 017 Ki = 0.32 nM 547.664
5T2Z 1.5 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME HYDROLASES 017 547.664
6DH0 1.9 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 017 Ki = 25.6 pM 547.664
6OPS 2.08 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 017 547.664
6OPU 1.94 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME HYDROLASES 017 547.664
6OPV 1.91 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME HYDROLASES 017 Ki = 12.8 nM 547.664
6OPX 2.03 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME HYDROLASES 017 Ki = 172.7 nM 547.664
6OPY 2.13 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME HYDROLASES 017 Ki = 156.4 nM 547.664
6OPZ 2.2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME HYDROLASES 017 Ki = 759.2 nM 547.664
6DGX 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 017, SO4 Ki < 5 pM 547.664, 96.063
6DH3 1.91 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 017, SO4 Ki < 5 pM 547.664, 96.063
6DH6 1.97 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 017, SO4 Ki = 117.2 pM 547.664, 96.063
6OOS 1.9 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 017, SO4 547.664, 96.063
6OOU 2.13 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 017, SO4 547.664, 96.063
6OPT 1.96 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 017, SO4 547.664, 96.063
6OPW 2.1 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME HYDROLASES 017, SO4 Ki = 23.2 nM 547.664, 96.063
4J55 1.31 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 031 601.711
1ODW 2.1 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 0E8 Ki = 100 nM 543.695
1ODX 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 0E8 543.695
4DJR 1.55 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 0KJ, PO4 Ki = 0.003 nM 588.739, 94.971
4DVS 2.1 HUMAN IMMUNODEFICIENCY VIRUS 1 NON-ENZYME OTHER 0LY, NAG, EPE 382.295, 221.208, 238.305
4DVT 2.4 HUMAN IMMUNODEFICIENCY VIRUS 1 NON-ENZYME OTHER 0LZ, NAG, EPE 361.798, 221.208, 238.305
4DVW 2.2 HUMAN IMMUNODEFICIENCY VIRUS 1 NON-ENZYME OTHER 0M4, EPE, NAG 339.792, 238.305, 221.208
4DVX 2.4 HUMAN IMMUNODEFICIENCY VIRUS 1 NON-ENZYME OTHER 0M5, NAG, EPE 339.792, 221.208, 238.305
4E92 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 NON-ENZYME OTHER 0OG, 0OE 535.55, 522.985
1A8K 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 0Q4 833.053
1A94 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 0Q4 Ki = 14 nM 833.053
1DAZ 1.55 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 0Q4 833.053
1DW6 1.88 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 0Q4 833.053
1EBK 2.06 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 0Q4 833.053
1FFF 1.9 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 0Q4 833.053
1FG8 1.85 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 0Q4 833.053
1K1U 1.55 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 0Q4 833.053
1K2B 1.7 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 0Q4 833.053
1K2C 2.2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 0Q4 833.053
5KQZ 1.7 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 0Q4 833.053
6O5X 1.7 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME HYDROLASES 0Q4, NA, CL Ki = 22 nM 833.053, 22.99, 35.453
1ZLF 2.3 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 0ZR Ki = 1000 nM 702.84
1ZSF 1.98 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 0ZS Ki = 0.12 nM 703.824
1ZJ7 1.93 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 0ZT Ki = 86 nM 703.824
1ZSR 2.06 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 0ZT Ki = 0.15 nM 703.824
1BWB 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 146 Ki = 3.8 nM 824.924
1QBT 2.1 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 146 Ki = 0.024 nM 824.924
1XL5 1.73 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 190, CL Ki = 45 nM 634.597, 35.453
2CEJ 2.5 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 1AH Ki = 2.4 nM 681.617
2XDE 1.4 HUMAN IMMUNODEFICIENCY VIRUS 1 NON-ENZYME OTHER 1B0 Kd = 3.42 uM 425.522
4XRQ 1.95 HUMAN IMMUNODEFICIENCY VIRUS 1 NON-ENZYME OTHER 1B0 Kd = 0.232 uM 425.522
4EJD 1.1 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 1F1, IVA VAL VAL STA ALA STA, GOL, BME Kd = 14.5 uM 161.157, 696.992, 92.094, 78.133
2BPV 1.9 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 1IN Ki = 21.2 nM 621.81
4J93 1.74 HUMAN IMMUNODEFICIENCY VIRUS 1 NON-ENZYME OTHER 1JR, 0OE 276.293, 522.985
1OHR 2.1 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 1UN Ki = 2 nM 567.782
2PYM 1.9 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 1UN Kd = 150 nM 567.782
2PYN 1.85 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 1UN Kd = 27 nM 567.782
2Q63 2.2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 1UN Kd = 66 nM 567.782
2Q64 2.5 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 1UN Kd = 3 nM 567.782
2R5Q 2.3 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 1UN Ki = 2.7 nM 567.782
1HIV 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 1ZK Ki < 1 nM 813.016
1HWR 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 216 Ki = 4.7 nM 406.517
2CEM 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 2AH Ki = 12 nM 679.804
1FEJ 1.78 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 2NC 770.983
1FF0 1.85 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 2NC 770.983
1FFI 1.7 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 2NC 770.983
1FG6 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 2NC 770.983
1FGC 1.9 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 2NC 770.983
4HVP 2.3 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 2NC Ki = 0.78 uM 770.983
6O57 1.71 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME HYDROLASES 2NC, FMT Ki = 514 nM 770.983, 46.025
4CEC 1.75 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 2SS, ACT, CL, GOL, SO4 522.589, 59.044, 35.453, 92.094, 96.063
1A8G 2.5 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 2Z4 Ki = 7.4 nM 825.989
2FDD 1.58 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 385 ic50 = 4.8 nM 703.823
4U7Q 1.7 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 3EM Ki = 180 pM 797.959
4CF2 1.95 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 3GM, SO4 482.526, 96.063
1C6X 2.5 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 3IN 727.336
2BPY 1.9 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 3IN Ki = 39.8 nM 727.336
2BPZ 2.5 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 3IN Ki = 39.8 nM 727.336
1NPA 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 3NH ic50 = 2 nM 629.743
2AZ8 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 3TL ic50 = 6 nM 909.077
2AZ9 2.5 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 3TL ic50 = 22 nM 909.077
2AZB 2.03 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 3TL ic50 = 64 nM 909.077
2AZC 2.01 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 3TL ic50 = 183 nM 909.077
2P3A 1.75 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 3TL Ki = 11 nM 909.077
2P3B 2.1 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 3TL Ki = 3.3 nM 909.077
4TVH 2.2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 3TL, BME, K97 909.077, 78.133, 260.288
1HPV 1.9 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 478 Ki = 0.6 nM 505.627
4J5J 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 478, CL Ka = 5610000 M^-1 505.627, 35.453
5KR0 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 478, GOL Ki = 0.71 nM 505.627, 92.094
2CEN 1.7 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 4AH Ki = 5 nM 679.804
4CJP 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 4D2, CL, SO4 384.426, 35.453, 96.063
5COK 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 52U 576.701
5CON 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 52W 592.701
5COO 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 52Z 622.727
5COP 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 53F 607.716
1WBK 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 568 620.689
5DGW 1.62 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 5B5, NA, CL Ki = 0.009 nM 619.769, 22.99, 35.453
1C1C 2.5 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.49 612 326.454
5HRP 1.81 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 65P, CAC, EDO, SO4 534.594, 136.989, 62.068, 96.063
5HRN 1.75 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.49 65P, CAC, SO4, EDO 534.594, 136.989, 96.063, 62.068
5IVS 1.46 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 6EF, CL ic50 = 6.1 nM 650.763, 35.453
5IVR 1.5 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 6EG, CL 566.69, 35.453
5IVQ 1.57 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 6EH, CL 425.521, 35.453
5JFP 1.49 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 6KK, CL, NA Ki = 0.48 nM 620.797, 35.453, 22.99
5JFU 1.7 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 6KQ, CL Ki = 8.5 nM 654.813, 35.453
5JG1 1.16 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 6KR, GOL, NA, CL Ki = 1.9 nM 634.824, 92.094, 22.99, 35.453
5KRT 1.65 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 6W6 262.113
4CFC 1.9 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 7NV, CL, ACT, SO4 441.477, 35.453, 59.044, 96.063
5TYR 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 7O7 ic50 = 0.26 nM 670.839
5TYS 2.01 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 7OA ic50 = 0.019 nM 706.82
6MKL 1.7 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME HYDROLASES 7OA 706.82
5KGW 2.34 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 7SK, SO4 393.475, 96.063
1QBU 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 846 Ki = 0.058 nM 596.739
5UOV 1.33 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 8FP, NA, GOL, CL, ACT Ki = 0.025 nM 704.898, 22.99, 92.094, 35.453, 59.044
5YOJ 1.5 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 8Z0, GOL 756.907, 92.094
5YOK 0.85 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 8Z0, GOL 756.907, 92.094
4CED 1.75 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 9NS, CL, SO4, GOL 534.557, 35.453, 96.063, 92.094
4CJL 1.77 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 9PA, ACT, SO4, CL 378.463, 59.044, 96.063, 35.453
5OIA 2.2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 9VK, SO4, MG ic50 = 0.17 uM 413.573, 96.063, 24.305
5OI8 2.35 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 9VN, SO4, MG ic50 = 0.21 uM 413.573, 96.063, 24.305
2BQV 2.1 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 A1A Ki = 9 nM 588.694
6DH8 1.95 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 A60, SO4 Ki = 146.2 pM 575.717, 96.063
1HVL 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 A76 Ki = 1000 pM 794.981
1HVI 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 A77 Ki = 84 pM 794.981
1HVS 2.25 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 A77 Ki = 50 pM 794.981
1HVJ 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 A78 Ki = 4 pM 780.998
1HVC 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 A79 794.981
1HVK 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 A79 Ki = 77 pM 794.981
1ZPA 2.02 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 A83 Ki = 4 nM 720.878
1PRO 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 A88 Ki = 5 pM 583.674
1VRU 2.4 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.49 AAP ic50 = 0.1 uM 351.227
2A4F 1.9 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 AAU 641.71
4L1A 1.9 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME HYDROLASES AB1 ic50 = 5.39 nM 628.801
6DJ1 1.26 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 AB1, CL, NA Ki = 0.031 nM 628.801, 35.453, 22.99
6DJ2 1.36 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 AB1, CL, NA Ki = 4.5 nM 628.801, 35.453, 22.99
6PJB 1.98 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 AB1, SO4 628.801, 96.063
1ZP8 2.02 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 AB2 Ki = 1.7 nM 663.784
7HVP 2.4 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 ACE SER LEU ASN JG3 ILE VME Ki = 0.24 nM 818.006
1YTH 2.2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 ACE SER LEU ASN PHE 520.563
3LZS 1.95 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 ACT, 017 Kd = 0.0109 nM 59.044, 547.664
3LZU 1.76 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 ACT, 017 Kd = 0.087 nM 59.044, 547.664
4DQE 1.3 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 ACT, 017 59.044, 547.664
4Q1W 1.85 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 ACT, 017, PO4 Ki = 2 pM 59.044, 547.664, 94.971
4Q1Y 1.5 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 ACT, 017, PO4 Ki = 45 pM 59.044, 547.664, 94.971
1T7J 2.2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 ACT, 478 Kd = 0.000000064 M 59.044, 505.627
4CJ5 1.95 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 ACT, 4VW, CL, SO4 Kd = 200 uM 59.044, 398.452, 35.453, 96.063
5DGU 1.22 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 ACT, 5B7, NA, CL Ki = 0.0045 nM 59.044, 606.727, 22.99, 35.453
5IVT 1.15 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 ACT, CL, 6EE ic50 = 0.8 nM 59.044, 35.453, 674.034
6BZ2 1.67 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 ACT, CL, 7OA, NA Ki = 14 pM 59.044, 35.453, 706.82, 22.99
4CHP 1.9 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 ACT, EDO, IMV, SO4 59.044, 62.068, 311.289, 96.063
4J54 1.55 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 ACT, G52, IOD 59.044, 604.712, 126.904
4E43 1.54 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 ACT, GOL, DMS, BME, ASN LEU LEU GLN LYS LYS 59.044, 92.094, 78.133, 78.133, 729.945
6CDL 1.25 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 ACT, GOL, GR5, CL, NA Ki = 0.012 nM 59.044, 92.094, 720.847, 35.453, 22.99
5WLO 1.27 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 ACT, GR7, GOL, CL, NA Ki = 0.015 nM 59.044, 630.749, 92.094, 35.453, 22.99
4CJV 1.95 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 ACT, IV2, SO4, GOL 59.044, 198.673, 96.063, 92.094
4CJU 1.7 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 ACT, JNS, SO4 59.044, 268.264, 96.063
2QCI 1.2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 ACT, NA, 065, CL Ki = 4.6 nM 59.044, 22.99, 576.658, 35.453
4CFB 1.95 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 ACT, OM3, SO4 59.044, 439.524, 96.063
3S56 1.88 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 ACT, ROC Ki = 0.24 nM 59.044, 670.841
4CEO 1.9 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 ACT, SO4, G0T, CL 59.044, 96.063, 548.584, 35.453
2P3C 2.1 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 ACY, 3TL Ki = 24 nM 60.052, 909.077
4CHY 1.7 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 ACY, EDO, SO4, C5Q 60.052, 62.068, 96.063, 295.289
4CEA 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 ACY, GOL, CL, ZSW, SO4 60.052, 92.094, 35.453, 511.587, 96.063
4CGH 1.76 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 ACY, LOZ, SO4 60.052, 396.436, 96.063
1AJX 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 AH1 Ki = 12.2 nM 538.633
1G35 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 AHF Ki = 7.3 nM 664.765
2BB9 1.35 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 AKC ic50 = 0.44 nM 625.711
1HEF 2.2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 ALA ALA PJJ VAL VME Ki = 1 nM
5TKK 1.55 HUMAN IMMUNODEFICIENCY VIRUS 1 NON-ENZYME OTHER ALA VAL GLY ILE GLY ALA VAL PHE 471.579
1KJF 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 ARG PRO GLY ASN PHE LEU GLN SER ARG PRO, ACT 975.119, 59.044
4QJ2 2.13 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 ARG PRO GLY ASN PHE LEU GLN SER ARG PRO, PO4, GOL, SO4 975.119, 94.971, 92.094, 96.063
3OUD 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME HYDROLASES ARG VAL LEU PHE GLU ALA MET 849.044
6BXQ 1.58 HUMAN IMMUNODEFICIENCY VIRUS 1 NON-ENZYME IMMUNE ARG VAL LYS GLU LYS TYR GLN HIS LEU TRP 1098.3
3AID 2.5 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 ARQ Ki = 137 nM 504.64
1B6J 1.85 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 ASN RTY PRO ILE VAL NH2, SO4 Ki = 12 nM 689.855, 96.063
4CEE 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 B0T, ACT, CL, SO4 484.541, 59.044, 35.453, 96.063
1VIJ 2.4 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 BAY ic50 = 0.3 nM 1131.49
1VIK 2.4 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 BAY ic50 = 0.3 nM 1131.49
1EBY 2.29 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 BEB Ki = 0.2 nM 652.733
1EBZ 2.01 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 BEC Ki = 0.4 nM 633.731
1EC0 1.79 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 BED Ki = 3.2 nM 688.714
1EC1 2.1 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 BEE Ki = 1.2 nM 778.977
1EBW 1.81 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 BEI Ki = 0.9 nM 642.783
1EC2 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 BEJ Ki = 0.1 nM 768.898
1T7K 2.1 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 BH0 Ki = 1.37 nM 598.669
1WBM 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 BLL 648.787
3U7S 2.05 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 BME, 017 Ki = 3700 pM 78.133, 547.664
1LZQ 2.2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 BME, 0ZQ Ki = 4.1 nM 78.133, 687.825
4U7V 1.38 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 BME, 3EN Ki = 3.2 uM 78.133, 524.675
3KFR 1.3 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 BME, 3TL, 1F1 78.133, 909.077, 161.157
4K4Q 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 BME, 3TL, DMS, 06B, NO3 78.133, 909.077, 78.133, 261.069, 62.005
1DIF 1.7 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 BME, A85 Ki = 22 pM 78.133, 830.962
6C8Y 1.94 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 BVR, CL, GOL 575.459, 35.453, 92.094
6C8X 1.61 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 BVR, GOL, CL Ki = 0.5 pM 575.459, 92.094, 35.453
1HIH 2.2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 C20, BME Ki = 9 nM 573.767, 78.133
1ZTZ 2.15 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 CB5, ALA GLY ALA ALA Ki = 66 nM 323.749, 273.313
4CJW 1.95 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 CBJ, ACT, SO4 418.195, 59.044, 96.063
3VQ8 1.6 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 CD, BCU, CL, SO4 112.411, 164.201, 35.453, 96.063
3VQ5 1.7 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 CD, CL, SO4, MMJ 112.411, 35.453, 96.063, 218.318
6B36 1.63 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 CKD, CL 607.686, 35.453
6B38 1.48 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 CKM, CL 621.712, 35.453
6B3F 1.46 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 CKV, CL 621.712, 35.453
6B3G 1.5 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 CKY, CL 621.712, 35.453
3MWS 1.09 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 CL, 017 35.453, 547.664
3BVB 1.3 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 CL, 017, NA, GOL Ka = 3170000 M^-1 35.453, 547.664, 22.99, 92.094
3M9F 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 CL, 595 ic50 = 0.007 nM 35.453, 650.828
4CHQ 1.95 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 CL, ACT, CWU, SO4, EDO 35.453, 59.044, 312.317, 96.063, 62.068
4CJ4 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 CL, ACT, S3G, SO4 Kd = 432 uM 35.453, 59.044, 384.426, 96.063
4CFD 2.15 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 CL, ACT, S8Y, SO4 35.453, 59.044, 441.477, 96.063
3NF6 1.9 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 CL, ACY, SO4, IMV, EDO ic50 = 295 uM 35.453, 60.052, 96.063, 311.289, 62.068
3AO4 1.95 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 CL, CD, 833, SO4 Kd = 8.5 mM 35.453, 112.411, 217.224, 96.063
6B3C 1.6 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 CL, CKS 35.453, 621.712
6B3H 1.62 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 CL, CN4 35.453, 571.654
3VQP 2.1 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 CL, DBJ, SO4, CD 35.453, 166.174, 96.063, 112.411
4CGG 1.75 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 CL, EDO, K5Q, SO4 35.453, 62.068, 409.389, 96.063
4CJF 1.9 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 CL, EDO, RVN, SO4, DMS, ACT 35.453, 62.068, 309.273, 96.063, 78.133, 59.044
6IXD 1 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 CL, GOL, B0F, SO4 Ki = 0.16 nM 35.453, 92.094, 873.092, 96.063
4CIF 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 CL, JDX, ACT, SO4 35.453, 448.511, 59.044, 96.063
4CJS 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 CL, L0Y, ACT, SO4 35.453, 452.543, 59.044, 96.063
5ULT 1.53 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 CL, NA, 8FM Ki = 0.014 nM 35.453, 22.99, 588.712
6VKV 2.22 HUMAN IMMUNODEFICIENCY VIRUS 1 NON-ENZYME OTHER CL, QNG, IOD 35.453, 968.282, 126.904
4CEF 1.7 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 D0T, CL, SO4, GOL 518.558, 35.453, 96.063, 92.094
2I4U 1.5 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 DJR Ki = 2.7 pM 562.675
2I4V 1.5 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 DJR Ki = 6.3 pM 562.675
3I7E 1.7 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 DJR Ki = 14 pM 562.675
1MES 1.9 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 DMP Ki = 20 nM 566.687
1MET 1.9 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 DMP Ki = 0.4 nM 566.687
1MEU 1.9 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 DMP Ki = 0.8 uM 566.687
1QBS 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 DMP Ki = 0.34 nM 566.687
1DMP 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 DMQ Ki = 0.28 nM 536.664
1MER 1.9 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 DMQ Ki = 10 nM 536.664
5KRS 1.7 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 DMS, 6XI 78.133, 193.222
4CEQ 1.7 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 DMS, ACT, CL, QCH, SO4 78.133, 59.044, 35.453, 524.605, 96.063
3KFP 1.77 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 DMS, BME, 3TL 78.133, 78.133, 909.077
3KFS 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 DMS, BME, 3TL, 2FX 78.133, 78.133, 909.077, 192.234
2HS1 0.84 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 DMS, CL, 017 Ki = 3.3 nM 78.133, 35.453, 547.664
2HS2 1.22 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 DMS, CL, 017 Ki = 4.9 nM 78.133, 35.453, 547.664
2AQU 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 DR7 Ki = 0.48 nM 704.855
2O4K 1.6 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 DR7, CL Kd = 35 pM 704.855, 35.453
5HGM 2.04 HUMAN IMMUNODEFICIENCY VIRUS 1 NON-ENZYME OTHER DTP 491.182
4CJ3 1.7 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 E4F, SO4, ACT 410.463, 96.063, 59.044
4EJ8 2.35 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 EDO, 1F1, DMS Kd = 4.1 uM 62.068, 161.157, 78.133
5HRR 1.88 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 EDO, 65P, CAC, SO4 62.068, 534.594, 136.989, 96.063
4CGD 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 EDO, 8P3, ACY, SO4, CL, GOL 62.068, 267.279, 60.052, 96.063, 35.453, 92.094
4CF9 2.1 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 EDO, ACT, EE2, 5EY, SO4 62.068, 59.044, 396.39, 396.39, 96.063
4CEB 1.75 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 EDO, ACY, SO4, ZSV, GOL Kd = 1080 uM 62.068, 60.052, 96.063, 575.629, 92.094
1FK9 2.5 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.49 EFZ 315.675
6ONF 1.84 HUMAN IMMUNODEFICIENCY VIRUS 1 NON-ENZYME OTHER EPE, MW4, NAG 238.305, 328.766, 221.208
6ONH 2.24 HUMAN IMMUNODEFICIENCY VIRUS 1 NON-ENZYME OTHER EPE, MWD, NAG 238.305, 341.808, 221.208
6OOO 2.4 HUMAN IMMUNODEFICIENCY VIRUS 1 NON-ENZYME OTHER EPE, MXJ, NAG 238.305, 356.823, 221.208
4RZ8 1.9 HUMAN IMMUNODEFICIENCY VIRUS 1 NON-ENZYME OTHER EPE, NAG, 3ZM ic50 ~ 270 nM 238.305, 221.208, 444.978
5U6E 2.1 HUMAN IMMUNODEFICIENCY VIRUS 1 NON-ENZYME OTHER EPE, NAG, 82M 238.305, 221.208, 408.878
6USW 2.5 HUMAN IMMUNODEFICIENCY VIRUS 1 NON-ENZYME OTHER EPE, O51, NAG 238.305, 342.796, 221.208
3ZPS 1.55 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 EQM, CL 730.732, 35.453
3VQ9 1.9 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 FBB 168.191
3VQB 2.1 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 FBG, SO4, CD 198.148, 96.063, 112.411
3VQE 1.7 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 FMQ, CD, CL, SO4 206.216, 112.411, 35.453, 96.063
6OTG 1.5 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 FMT, 4UY, GOL Ki = 31.4 nM 46.025, 591.716, 92.094
6E9A 1.22 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 FMT, CL, J0S, NA Ki = 0.0012 nM 46.025, 35.453, 575.674, 22.99
6O48 1.46 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 FMT, GOL, 0Q4, NA, CL Ki = 75 nM 46.025, 92.094, 833.053, 22.99, 35.453
6D0E 1.95 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 FQ1 612.682
6D0D 1.85 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 FQ4 594.692
4CJR 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 FYM, ACT, CL, SO4 Kd = 793 uM 492.52, 59.044, 35.453, 96.063
4NJS 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME HYDROLASES G08 575.674
2PQZ 1.55 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 G0G, CL Ki = 2.15 uM 561.715, 35.453
1HTF 2.2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 G26 ic50 = 148 nM 574.734
1HTG 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 G37 ic50 = 3.8 nM 761.931
2R3W 1.92 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 G3G, CL Ki = 0.128 uM 591.744, 35.453
5KAO 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 G43 627.146
2R38 1.81 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 G4G, CL Ki = 0.036 uM 647.764, 35.453
2R3T 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 G4G, CL Ki = 1.4 uM 647.764, 35.453
4KB9 1.29 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 G79, GOL, NA, CL, ACT Ki = 0.01 nM 616.765, 92.094, 22.99, 35.453, 59.044
1HBV 2.3 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 GAN Ki = 430 nM 585.778
1C1B 2.5 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.49 GCA 330.421
3GGA 2.5 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 GGW 703.867
3VQ7 1.63 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 GLC FRU, CD, SO4, SNU 340.281, 112.411, 96.063, 158.2
3VQA 1.9 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 GLC FRU, MWP, SO4, CD 340.281, 181.212, 96.063, 112.411
2BE2 2.43 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.49 GLC FRU, R22, MN, GOL ic50 = 0.002 uM 340.281, 481.347, 54.938, 92.094
3VQQ 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 GLC FRU, SO4, BTE, CD 340.281, 96.063, 151.189, 112.411
3AO5 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 GLC FRU, SO4, CL, CD, BBY Kd = 5.9 mM 340.281, 96.063, 35.453, 112.411, 296.12
3OVN 1.95 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 GLC FRU, SO4, MPV, CD Kd = 2.8 mM 340.281, 96.063, 179.242, 112.411
3OTS 1.7 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 GLN ASN TYR PRO ILE VAL GLN 803.915
3OUB 1.6 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 GLN VAL ASN PHE LEU GLY LYS 789.932
1A30 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 GLU ASP LEU Ki = 50 uM 373.362
5YRS 1.76 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 GLU THR HPH TYR VAL ASP 788.808
3OTY 1.75 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 GLU THR PHE TYR VAL ASP GLY 827.845
1KJG 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 GLY ALA GLU THR PHE TYR VAL ASP GLY ALA, ACT 968.995, 59.044
3OUA 1.7 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 GLY ASN PHE LEU GLN SER ARG 821.914
4DQH 1.79 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 GOL, 017 92.094, 547.664
4NPT 1.66 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME HYDROLASES GOL, 017 92.094, 547.664
2PK5 1.9 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 GOL, 075 Kd = 20 pM 92.094, 803.943
1M0B 2.45 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 GOL, 0ZQ Ki = 1.53 nM 92.094, 687.825
1IIQ 1.83 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 GOL, 0ZR Ki = 33 nM 92.094, 702.84
3BVA 1.05 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 GOL, 2NC Ka = 3300000 M^-1 92.094, 770.983
6O5A 1.67 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME HYDROLASES GOL, 2NC Ki = 514 nM 92.094, 770.983
2RKG 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 GOL, AB1 Ki = 8.2 nM 92.094, 628.801
6DV4 1.14 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 GOL, ACT, GA5, CL, NA Ki = 1.6 nM 92.094, 59.044, 695.865, 35.453, 22.99
4DJO 1.78 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 GOL, ACT, PO4, MK5 Ki = 0.003 nM 92.094, 59.044, 94.971, 618.57
2AVM 1.1 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 GOL, ACY, 2NC Ki = 2 uM 92.094, 60.052, 770.983
2FLE 1.9 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 GOL, AI Ki = 14 nM 92.094, 801.029
1XL2 1.5 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 GOL, CL, 189 Ki = 1.5 uM 92.094, 35.453, 577.777
5UPZ 1.27 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 GOL, CL, 8HD, NA Ki = 0.63 nM 92.094, 35.453, 662.796, 22.99
2O4S 1.54 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 GOL, CL, AB1 Kd = 31 pM 92.094, 35.453, 628.801
4CF8 1.65 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 GOL, EDO, CL, ACY, SO4, V7H 92.094, 62.068, 35.453, 60.052, 96.063, 504.531
4OVL 1.7 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 GOL, EDO, SO4, 1TD, ACY 92.094, 62.068, 96.063, 265.263, 60.052
6DJ7 1.31 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 GOL, G10, ACT, CL, NA Ki = 1.9 nM 92.094, 583.645, 59.044, 35.453, 22.99
2PWC 1.78 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 GOL, G3G, CL Ki = 0.27 uM 92.094, 591.744, 35.453
2R43 1.58 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 GOL, G3G, CL Ki = 1 uM 92.094, 591.744, 35.453
2PWR 1.5 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 GOL, G4G, CL Ki = 0.26 uM 92.094, 647.764, 35.453
6VCE 1.18 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 GOL, G6R, NA, CL ic50 = 79 pM 92.094, 704.847, 22.99, 35.453
6DV0 1.2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 GOL, GA8, CL, NA Ki = 0.38 nM 92.094, 697.904, 35.453, 22.99
4FLG 1.31 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 GOL, GLN ILE ILE, CL, ASP GLN ILE ILE, NA, ILE GLU ILE 92.094, 315.414, 35.453, 386.493, 22.99, 315.37
6DJ5 1.75 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 GOL, NA, G52, CL 92.094, 22.99, 604.712, 35.453
2I0A 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 GOL, PO4, MUI Ki = 0.004 nM 92.094, 94.971, 637.743
2O4N 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 GOL, TPV Kd = 15010 pM 92.094, 602.664
4CJK 1.75 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 H39, CL, SO4, ACT 386.442, 35.453, 96.063, 59.044
4CHZ 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 H75, EDO, ACT, CL, SO4 293.159, 62.068, 59.044, 35.453, 96.063
2BBB 1.7 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 HH1 ic50 = 2.4 nM 623.738
2UXZ 1.75 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 HI1 Ki = 3.3 nM 709.67
4CJT 1.71 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 HLR, GOL, SO4, ACT 134.135, 92.094, 96.063, 59.044
2UY0 1.76 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 HV1 Ki = 120 nM 723.653
6E7J 1.3 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 HWY, NA, CL Ki = 0.33 nM 651.77, 22.99, 35.453
6ES8 1.9 HUMAN IMMUNODEFICIENCY VIRUS 1 NON-ENZYME OTHER IHP 660.035
1KJH 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 ILE ARG LYS ILE LEU PHE LEU ASP GLY ILE, ACT 1146.42, 59.044
4GZF 2.05 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 ILO VAL DC0 GLU ALA NLE ic50 = 4.4 nM 832.057
4GYE 2.27 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 ILO VAL PUK GLU ALA NLE 866.074
1BDQ 2.5 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 IM1 Ki = 460 nM 534.69
1TCX 2.3 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 IM1 Ki = 112 nM 534.69
7UPJ 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 INU Ki = 3.2 nM 479.588
4E91 1.7 HUMAN IMMUNODEFICIENCY VIRUS 1 NON-ENZYME OTHER IOD, 0OF, 0OE 126.904, 517.498, 522.985
3NU9 1.85 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 IOD, 478 Ki = 0.9 nM 126.904, 505.627
3NUJ 1.5 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 IOD, 478 Ki = 0.41 nM 126.904, 505.627
3NUO 1.35 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 IOD, 478 Ki = 0.16 nM 126.904, 505.627
3S43 1.26 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 IOD, GOL, 478 Ki = 2.53 nM 126.904, 92.094, 505.627
4EJL 2.45 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 IOP, DMS, GOL, PEG Kd = 7.2 uM 189.211, 78.133, 92.094, 106.12
4EJK 1.79 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 IOP, IVA VAL VAL STA ALA STA Kd = 5.3 uM 189.211, 696.992
4CF1 1.9 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 IY7, ACT, SO4 496.552, 59.044, 96.063
6EB1 2.2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 J3M ic50 = 4.65 uM 467.556
6EB2 2.49 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 J3P ic50 = 0.48 uM 547.644
6MCS 1.52 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 JDV 688.83
6MCR 1.48 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 JDY, EDO 688.83, 62.068
6OGT 1.21 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME HYDROLASES JDY, EDO, GOL ic50 = 31 nM 688.83, 62.068, 92.094
1MSM 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 JE2 Kd = 33 pM 575.718
1MSN 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 JE2 Kd < 1 nM 575.718
3KF0 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 K, DMS, BME, 4DX, 3TL 39.098, 78.133, 78.133, 114.185, 909.077
3KFN 1.77 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 K, DMS, BME, 4DX, 3TL 39.098, 78.133, 78.133, 114.185, 909.077
6DH4 1.94 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 K13, SO4 Ki < 5 pM 561.69, 96.063
4CK3 1.79 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 K1T, SO4, ACT Kd = 268 uM 364.436, 96.063, 59.044
1MRW 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 K57 Kd = 0.2 nM 527.675
1MRX 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 K57 Kd = 55 nM 527.675
4TVG 2.18 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 K97, IVA VAL VAL STA ALA STA, GOL 260.288, 696.992, 92.094
2I4W 1.55 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 KGQ Ki = 2.6 pM 728.787
2I4X 1.55 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 KGQ Ki = 1.9 pM 728.787
4M8X 2.05 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 KGQ Ki = 0.063 nM 728.787
4M8Y 2.22 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 KGQ Ki = 0.11 nM 728.787
1U8G 2.2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 KI2 PHE GLU GLU NH2 732.767
6NCJ 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 KJJ, SO4, EDO ic50 = 0.024 uM 572.709, 96.063, 62.068
1HPX 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 KNI Ki = 5.5 pM 667.839
3FX5 0.93 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 KNI, GOL Ki < 1 nM 667.839, 92.094
3A2O 0.88 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 KNJ, GOL Ki = 0.83 nM 568.727, 92.094
6KMP 1.31 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 KVS 800.986
1NPV 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 L27 ic50 = 5.7 nM 595.685
6NUJ 2.1 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 L3D 442.506
1C70 2.5 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 L75 Ki = 0.05 nM 652.822
3OU3 1.7 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 LEU ASN PHE PRO ILE SER PRO 786.928
1NPW 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 LGZ ic50 = 2 nM 625.711
1F7A 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 LYS ALA ARG VAL LEU ALA GLU ALA MET SER, ACT 916.136, 59.044
1MT8 2.15 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 LYS ALA ARG VAL LEU ALA GLU ALA MET SER, ACT 916.136, 59.044
3OU1 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME HYDROLASES LYS VAL LEU PHE LEU ASP GLY 790.96
3ZPU 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 M8B, CL Ki = 4.2 nM 742.743, 35.453
3ZPT 1.54 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 M8Y, CL Ki = 3.1 nM 728.716, 35.453
1QS4 2.1 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 MG, 100 ic50 = 2.3 uM 24.305, 289.677
5OI5 2.4 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 MG, 9VK ic50 = 0.19 uM 24.305, 413.573
4LH5 2.19 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 MG, LF0 ic50 = 0.23 uM 24.305, 405.486
6OGP 1.53 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 MJD, EDO ic50 = 0.055 uM 692.77, 62.068
1C6Y 2.5 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 MK1 Ki = 0.31 nM 613.789
1HSG 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 MK1 Ki = 0.38 nM 613.789
1HSH 1.9 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 MK1 Ki = 2.45 nM 613.789
1SGU 1.9 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 MK1 Ki = 4235 nM 613.789
1K6C 2.2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 MK1, ACT Kd = 33 nM 613.789, 59.044
1SDT 1.3 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 MK1, CL Ki = 540 pM 613.789, 35.453
1SDV 1.4 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 MK1, CL Ki = 1810 pM 613.789, 35.453
2AVV 1.5 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 MK1, CL, ACY Ki = 0.55 nM 613.789, 35.453, 60.052
1EC3 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 MS3 Ki = 0.92 nM 768.898
2Q54 1.85 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 MU1, ACT, PO4 Ki = 0.98 nM 656.768, 59.044, 94.971
6ONE 2.2 HUMAN IMMUNODEFICIENCY VIRUS 1 NON-ENZYME OTHER MVY, EPE, NAG 314.74, 238.305, 221.208
4INB 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 NON-ENZYME OTHER NA, 1F6 ic50 = 0.89 uM 22.99, 419.397
2IEO 1.53 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 NA, CL, 017 Ki = 3.2 nM 22.99, 35.453, 547.664
3NU4 1.2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 NA, CL, 478 Ki = 1.5 nM 22.99, 35.453, 505.627
3PWM 1.46 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 NA, CL, ACT, 017 22.99, 35.453, 59.044, 547.664
2QD6 1.28 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 NA, CL, ACT, 065 Ki = 2.1 nM 22.99, 35.453, 59.044, 576.658
2QD8 1.35 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 NA, CL, ACT, 065 Ki = 0.85 nM 22.99, 35.453, 59.044, 576.658
2Z4O 1.6 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 NA, CL, ACT, 065 Ki = 0.27 nM 22.99, 35.453, 59.044, 576.658
3NU5 1.29 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 NA, CL, ACT, 478 Ki = 4.5 nM 22.99, 35.453, 59.044, 505.627
3NU6 1.16 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 NA, CL, ACT, 478 Ki = 0.5 nM 22.99, 35.453, 59.044, 505.627
6U7P 1.13 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 NA, FMT, B4R, CL, GOL 22.99, 46.025, 590.493, 35.453, 92.094
6B4N 1.3 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 NA, G53, CL Ki = 27.9 pM 22.99, 657.731, 35.453
2F81 1.25 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 NA, GOL, CL, 017 Ki = 0.03 nM 22.99, 92.094, 35.453, 547.664
3NU3 1.02 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 NA, GOL, CL, 478 Ki = 0.15 nM 22.99, 92.094, 35.453, 505.627
3S54 1.42 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 NA, GOL, CL, ACT, 017 Ki = 0.23 nM 22.99, 92.094, 35.453, 59.044, 547.664
2F8G 1.22 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 NA, GOL, CL, ACY, 017 Ki = 2 nM 22.99, 92.094, 35.453, 60.052, 547.664
2IEN 1.3 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 NA, GOL, CL, ACY, 017 Ki = 1 nM 22.99, 92.094, 35.453, 60.052, 547.664
3OK9 1.27 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 NA, GOL, G52, CL Ki = 5.9 pM 22.99, 92.094, 604.712, 35.453
6CDJ 1.13 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 NA, GR8, ACT, CL, GOL Ki = 2 pM 22.99, 720.847, 59.044, 35.453, 92.094
2HB3 1.35 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 NA, GRL, GOL, CL Ki = 0.0045 nM 22.99, 560.702, 92.094, 35.453
2A1E 1.3 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 NA, IPF, GOL, DMS, CL, ACT 22.99, 905.092, 92.094, 78.133, 35.453, 59.044
2R5P 2.3 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 NA, MK1, CL Ki = 3.3 nM 22.99, 613.789, 35.453
6VOD 1.25 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 NA, T1R, CL, GOL, FMT ic50 = 38 nM 22.99, 588.712, 35.453, 92.094, 46.025
6MTJ 2.34 HUMAN IMMUNODEFICIENCY VIRUS 1 NON-ENZYME OTHER NAG NAG BMA MAN MAN MAN MAN MAN MAN MAN, NAG NAG BMA, NAG NAG BMA MAN MAN MAN, 83G, NAG, NAG NAG 1721.53, 570.545, 406.434, 221.208, 408.404
6MU7 2.5 HUMAN IMMUNODEFICIENCY VIRUS 1 NON-ENZYME OTHER NAG NAG BMA MAN MAN MAN MAN MAN MAN MAN, NAG NAG BMA, NAG NAG BMA MAN MAN MAN, NAG, NAG NAG, JYY Kd = 0.002 uM 1721.53, 570.545, 221.208, 408.404, 572.635
6MTN 2.5 HUMAN IMMUNODEFICIENCY VIRUS 1 NON-ENZYME OTHER NAG NAG BMA MAN MAN MAN MAN MAN MAN MAN, NAG NAG BMA, NAG NAG, NAG NAG BMA MAN MAN MAN, NAG, JYJ 1721.53, 570.545, 408.404, 221.208, 374.884
4DVV 1.94 HUMAN IMMUNODEFICIENCY VIRUS 1 NON-ENZYME OTHER NAG, 0M1, EPE 221.208, 359.78, 238.305
6L1Y 2.47 HUMAN IMMUNODEFICIENCY VIRUS 1 NON-ENZYME OTHER NAG, EPE 221.208, 238.305
6OXU 1.86 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 NE7, SO4 590.728, 96.063
6OXT 1.86 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 NEJ, SO4 590.728, 96.063
6OXV 1.99 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 NF4 604.755
6OXX 1.96 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 NF7 592.701
6OXW 1.98 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 NFJ 604.755
4CES 1.85 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 NFW, CL, SO4 508.52, 35.453, 96.063
6OXS 1.99 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 NJ4 576.701
6OY0 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 NJ7, SO4 606.727, 96.063
6OXR 2.04 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 NJA 576.701
6OXZ 1.96 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 NJG, SO4 606.727, 96.063
6OY2 1.99 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 NJJ, SO4 620.754, 96.063
6OXO 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 NJM, SO4 562.675, 96.063
6OYR 1.54 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 NJY ic50 = 0.29 nM 674.78
6OYD 1.46 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 NKA ic50 = 0.12 nM 674.78
1G2K 1.95 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 NM1 Ki = 11 nM 631.738
1AJV 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 NMB Ki = 19.1 nM 574.687
1VRT 2.2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.49 NVP, MG ic50 = 0.08 uM 266.298, 24.305
4CK2 1.85 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 NVU, SO4, ACT 177.157, 96.063, 59.044
4CGI 2.07 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 NZL, ACT, SO4 Kd = 752 uM 424.49, 59.044, 96.063
4CGJ 2.15 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 NZL, ACT, SO4 424.49, 59.044, 96.063
2PK6 1.45 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 O33, GOL Kd = 13 pM 771.945, 92.094
4CE9 2.1 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 O3N, ACY, SO4, GOL 550.643, 60.052, 96.063, 92.094
4CEZ 1.7 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 O3N, CL, SO4, GOL 550.643, 35.453, 96.063, 92.094
4CF0 1.85 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 O5U, ACT, SO4 510.579, 59.044, 96.063
4CK1 1.75 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 OM1, CL, EDO, ACT, SO4 449.476, 35.453, 62.068, 59.044, 96.063
4CHN 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 ONZ, ACT, EDO, GOL, SO4 223.182, 59.044, 62.068, 92.094, 96.063
6PJI 1.9 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 OO4, SO4 Ki = 0.571 nM 595.683, 96.063
6PJF 1.94 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 OP7, SO4 Ki = 0.235 nM 623.736, 96.063
6PJE 1.92 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 OPJ, SO4 Ki = 46 nM 609.71, 96.063
6PJO 1.95 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 OQ7, SO4 Ki = 0.161 nM 623.736, 96.063
6PJK 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 OQD, SO4 Ki = 0.055 nM 611.726, 96.063
6PJN 1.98 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 OQP, SO4 Ki = 7.3 nM 609.71, 96.063
6PJM 1.93 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 OQV, SO4 Ki = 0.013 nM 611.726, 96.063
6PJG 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 ORV Ki = 0.019 nM 569.646
6PU8 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 P3V 563.663
6UM8 2.33 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 PEG, 1PE, SO4, QCG Ki = 0.17 uM 106.12, 238.278, 96.063, 503.565
6OGQ 1.41 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME HYDROLASES PEG, GOL, JDV, SO4 ic50 = 26 nM 106.12, 92.094, 688.83, 96.063
3OU4 1.6 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME HYDROLASES PHE ASN PHE PRO GLN ILE THR 865.986
1HOS 2.3 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 PHP Ki = 2.8 nM 770.85
1T3R 1.2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 PO4, 017 Ki = 14 pM 94.971, 547.664
4Q1X 1.9 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 PO4, 017, GOL Ki = 7 pM 94.971, 547.664, 92.094
3R4B 1.9 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 PO4, 74T 94.971, 755.987
2Q5K 1.95 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 PO4, AB1 Ki = 0.005 nM 94.971, 628.801
1T7I 1.35 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 PO4, ACT, 017 94.971, 59.044, 547.664
2FNS 1.85 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 PO4, ARG GLN ALA ASN PHE LEU GLY LYS ILE ASN, ACT 94.971, 647.754, 59.044
2FNT 1.44 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 PO4, ARG GLN VAL ASN PHE LEU GLY LYS ILE ASN, ACT 94.971, 675.808, 59.044
1MT9 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 PO4, ARG PRO GLY ASN PHE LEU GLN SER ARG PRO 94.971, 975.119
3GI6 1.84 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 PO4, D78 Ki = 0.006 nM 94.971, 663.704
4DQB 1.5 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 PO4, EDO, DMS, 017 94.971, 62.068, 78.133, 547.664
4DQC 1.94 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 PO4, GOL, 017 94.971, 92.094, 547.664
2QD7 1.11 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 PO4, GOL, DMS, 065 Ki = 0.8 nM 94.971, 92.094, 78.133, 576.658
2IDW 1.1 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 PO4, GOL, DMS, CL, ACY, 017 Ki = 1.3 nM 94.971, 92.094, 78.133, 35.453, 60.052, 547.664
3S53 1.5 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 PO4, IOD, 017 Ki = 0.23 nM 94.971, 126.904, 547.664
3GI4 1.85 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 PO4, K60, ACT Ki = 0.016 nM 94.971, 677.688, 59.044
3GI5 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 PO4, K62 Ki = 0.006 nM 94.971, 651.727
4DJP 1.4 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 PO4, M73 Ki = 0.028 nM 94.971, 564.691
4DJQ 1.4 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 PO4, M86 Ki = 0.048 nM 94.971, 576.705
2Q55 1.9 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 PO4, MU0 Ki = 2.04 nM 94.971, 655.783
2I0D 1.95 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 PO4, MUT, ACT Ki = 0.0008 nM 94.971, 637.743, 59.044
2PSU 1.93 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 PO4, MUU, ACT Ki = 24 nM 94.971, 517.638, 59.044
2PSV 1.75 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 PO4, MUV, ACT Ki = 58 nM 94.971, 477.574, 59.044
2Q3K 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 PO4, MUW, ACT 94.971, 638.817, 59.044
2QHY 1.85 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 PO4, MZ1, ACT Ki = 33 nM 94.971, 583.643, 59.044
2QHZ 1.85 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 PO4, MZ2 Ki = 53 nM 94.971, 606.6
2QI0 2.1 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 PO4, MZ3 Ki = 42 nM 94.971, 582.706
2QI1 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 PO4, MZ4 Ki = 50 nM 94.971, 582.688
2QI3 1.95 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 PO4, MZ5 Ki = 0.063 nM 94.971, 547.73
2QI4 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 PO4, MZ6, ACT Ki = 0.036 nM 94.971, 567.719, 59.044
2QI5 1.85 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 PO4, MZ7 Ki = 0.014 nM 94.971, 588.782
2QI6 1.85 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 PO4, MZ8 Ki = 0.027 nM 94.971, 553.693
2QI7 1.85 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 PO4, MZ9, ACT Ki = 0.062 nM 94.971, 532.692, 59.044
2HND 2.5 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.49 PO4, NVP, MG 94.971, 266.298, 24.305
2HNY 2.5 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.49 PO4, NVP, MG ic50 = 1165 nM 94.971, 266.298, 24.305
2WHH 1.69 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 PPN, GLU 210.187, 147.129
1KJ7 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 PRO ALA THR ILE MET MET GLN ARG GLY ASN, ACT 892.138, 59.044
1YTG 2.3 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 PRO ILE VAL NH2 328.457
1AAQ 2.5 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 PSI Ki = 3 nM 577.713
1HEG 2.2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 PSI Ki = 18 nM 577.713
6U7O 1.33 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 Q1D, NA, FMT, CL, GOL Ki = 15.5 uM 602.504, 22.99, 46.025, 35.453, 92.094
4CJE 1.9 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 Q31, CL, ACT, SO4 387.43, 35.453, 59.044, 96.063
1IZH 1.9 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 Q50 Ki = 0.02 uM 685.809
1IZI 2.15 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 Q50, CL Ki = 0.26 nM 685.809, 35.453
1HVH 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 Q82 Ki = 11 nM 590.711
2I4D 1.5 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 QFI Ki = 2.1 pM 672.681
2QNN 1.48 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 QN1, GOL, CL Ki = 0.07 uM 783.76, 92.094, 35.453
2QNP 1.41 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 QN2, CL Ki = 0.39 uM 813.508, 35.453
2QNQ 2.3 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 QN3, CL Ki = 0.77 uM 630.605, 35.453
1MTB 2.5 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 QNC ASN HPH DIQ NTB 670.855
2FGU 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 QNC ASN HPH DIQ NTB, PO4 Kd = 0.66 nM 670.855, 94.971
2FGV 1.5 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 QNC ASN HPH DIQ NTB, PO4 Kd = 760 nM 670.855, 94.971
6V2F 2 HUMAN IMMUNODEFICIENCY VIRUS 1 NON-ENZYME OTHER QNG Kd = 240 pM 968.282
6VLM 2.32 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 R2D ic50 = 10 uM 342.799
1HXW 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 RIT Ki = 15 pM 720.944
1N49 2.2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 RIT 720.944
1RL8 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 RIT 720.944
1SH9 2.5 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 RIT Ki = 932 nM 720.944
4EYR 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 RIT ic50 = 237 nM 720.944
4NJV 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME HYDROLASES RIT 720.944
2F3K 1.6 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 RO1, PO4 Kd = 0.95 nM 711.911, 94.971
1C6Z 2.5 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 ROC 670.841
5KQX 2.4 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 ROC Ki = 3.6 nM 670.841
5KR2 1.78 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 ROC Ki = 3.3 nM 670.841
3PWR 1.45 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 ROC, GOL, CL 670.841, 92.094, 35.453
2NNK 1.25 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 ROC, NA, GOL, CL, ACY 670.841, 22.99, 92.094, 35.453, 60.052
3CYX 1.2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 ROC, PO4, NA, GOL, ACY Ki = 10 nM 670.841, 94.971, 22.99, 92.094, 60.052
3R0W 1.7 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 RSY ic50 = 30.3 uM 631.163
3R0Y 1.65 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 RSZ ic50 = 14.53 uM 597.704
1HPS 2.3 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 RUN Ki = 0.6 nM 638.796
1EP4 2.5 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.49 S11 451.369
6BRA 1.11 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 SER GLY ILE PHE LEU GLU THR SER, CL 854.956, 35.453
3NF7 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 SO4 EDO, SO4, EDO, CIW, ACY ic50 = 340 uM 96.063, 62.068, 345.734, 60.052
6OOT 1.82 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 SO4, 017 96.063, 547.664
3VQ4 1.9 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 SO4, 0NX, CD 96.063, 175.184, 112.411
1K1T 1.2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 SO4, 0Q4 96.063, 833.053
3UHL 2.2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 SO4, 2NC 96.063, 770.983
5OI2 2.2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 SO4, 9VN, MG ic50 = 0.17 uM 96.063, 413.573, 24.305
6DGZ 1.99 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 SO4, A60 Ki < 5 pM 96.063, 575.717
6DH2 1.98 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 SO4, A60 Ki = 12.8 pM 96.063, 575.717
6DH5 2.01 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 SO4, A60 96.063, 575.717
3VQ6 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 SO4, BCK, CD 96.063, 188.226, 112.411
3NFA 1.95 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 SO4, CBJ, ACY ACY, ACY 96.063, 418.195, 60.052
3AO1 1.9 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 SO4, CD, BZX Kd = 5.5 mM 96.063, 112.411, 138.121
3L3V 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 SO4, CD, GLC FRU 96.063, 112.411, 340.281
3NF8 1.9 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 SO4, CDQ, ACY 96.063, 359.76, 60.052
2F80 1.45 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 SO4, CL, 017 Ki = 6.6 nM 96.063, 35.453, 547.664
3AO3 1.9 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 SO4, CL, CD, BMC 96.063, 35.453, 112.411, 246.219
2FXD 1.6 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 SO4, DR7, ACT ic50 = 12 nM 96.063, 704.855, 59.044
5HRS 1.86 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 SO4, EDO, 65P, CAC 96.063, 62.068, 534.594, 136.989
3NF9 1.95 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 SO4, EDO, CD9, ACY ic50 = 290 uM 96.063, 62.068, 345.734, 60.052
6OXQ 1.89 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 SO4, F53 96.063, 590.728
2RKF 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 SO4, GOL, AB1 Ki = 0.83 nM 96.063, 92.094, 628.801
2J9K 1.2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 SO4, GOL, ACT, 2NC 96.063, 92.094, 59.044, 770.983
2J9J 1.04 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 SO4, GOL, ACT, ACE SER LEU ASN JG3 ILE VME 96.063, 92.094, 59.044, 818.006
2JE4 1.07 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 SO4, GOL, ACT, ACE SER LEU ASN JG3 ILE VME 96.063, 92.094, 59.044, 818.006
2FXE 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 SO4, GOL, DR7, ACT 96.063, 92.094, 704.855, 59.044
4DQF 1.9 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 SO4, GOL, EDO, 017 96.063, 92.094, 62.068, 547.664
6DGY 1.95 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 SO4, K13 Ki < 5 pM 96.063, 561.69
6DH1 1.97 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 SO4, K13 Ki = 26.1 pM 96.063, 561.69
6DH7 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 SO4, K13 Ki = 131.3 pM 96.063, 561.69
6OXP 1.97 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 SO4, K2A 96.063, 576.701
1NH0 1.03 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 SO4, KI2 PHE GLU GLU NH2, BME Ki = 0.18 nM 96.063, 732.767, 78.133
4TSX 1.94 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 SO4, LF0 Kd = 10.3 uM 96.063, 405.486
3AO2 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 SO4, MG, DTV, DTT, CL, CD, AVX Kd = 0.17 mM 96.063, 24.305, 154.251, 154.251, 35.453, 112.411, 296.12
1SDU 1.25 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 SO4, MK1, ACT Ki = 86 pM 96.063, 613.789, 59.044
2AVO 1.1 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 SO4, MK1, GOL, DMS, ACY Ki = 1.4 nM 96.063, 613.789, 92.094, 78.133, 60.052
3VQD 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 SO4, MOK, CD 96.063, 203.194, 112.411
3VQC 2.3 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 SO4, MPK, CD 96.063, 189.211, 112.411
6OXY 1.96 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 SO4, NG4 96.063, 592.701
6OY1 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 SO4, NJ1 96.063, 620.754
6PJL 1.99 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 SO4, OQA Ki = 0.027 nM 96.063, 611.726
6PJH 1.85 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 SO4, OQG Ki = 0.074 nM 96.063, 597.699
6PJD 1.89 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 SO4, OQY Ki = 0.018 nM 96.063, 611.726
6PJC 1.97 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 SO4, OR1 Ki = 0.017 nM 96.063, 602.717
1B6L 1.75 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 SO4, PI4 Ki = 5 nM 96.063, 545.671
1B6K 1.85 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 SO4, PI5 Ki = 1.8 nM 96.063, 679.846
1B6M 1.85 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 SO4, PI6 Ki = 4 nM 96.063, 596.757
1MTR 1.75 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 SO4, PI6 Ki = 4 nM 96.063, 596.757
1B6P 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 SO4, PI7 Ki = 3 nM 96.063, 667.835
2AVS 1.1 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 SO4, PO4, MK1, DMS, ACY Ki = 27 nM 96.063, 94.971, 613.789, 78.133, 60.052
2NMZ 0.97 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 SO4, ROC 96.063, 670.841
3OXC 1.16 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 SO4, ROC, FMT Ki = 3.9 nM 96.063, 670.841, 46.025
2NNP 1.2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 SO4, ROC, GOL, ACY 96.063, 670.841, 92.094, 60.052
2NMY 1.1 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 SO4, ROC, NA, CL 96.063, 670.841, 22.99, 35.453
4CGF 1.7 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 SO4, UJ6, EDO, ACT 96.063, 311.289, 62.068, 59.044
3BGR 2.1 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.49 T27, EDO 366.419, 62.068
2ZD1 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.49 T27, SO4, EDO 366.419, 96.063, 62.068
6VOE 1.3 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 T2R, ACT, NA, CL ic50 = 0.3 nM 656.789, 59.044, 22.99, 35.453
1AID 2.2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 THK, CL Ki = 15 uM 452.048, 35.453
2AID 1.9 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 THK, CL Ki = 15 uM 452.048, 35.453
3OUC 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 THR ILE MET MET GLN ARG GLY 837.058
1D4S 2.5 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 TPV Ki = 0.008 nM 602.664
1D4Y 1.97 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 TPV Ki = 0.008 nM 602.664
4NJU 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME HYDROLASES TPV 602.664
6DIL 1.48 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 TPV, CL, GOL, ACT, NA Ki = 7.6 nM 602.664, 35.453, 92.094, 59.044, 22.99
2O4P 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 TPV, GOL Kd = 19 pM 602.664, 92.094
2O4L 1.33 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 TPV, GOL, CL Kd = 608 pM 602.664, 92.094, 35.453
6DIF 1.2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 TPV, GOL, CL, NA Ki = 0.019 nM 602.664, 92.094, 35.453, 22.99
2RKI 2.3 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.49 TT1, SO4, MG, GOL, CL 397.944, 96.063, 24.305, 92.094, 35.453
1HYV 1.7 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 TTA, SO4, CL ic50 > 5 mM 383.337, 96.063, 35.453
1HYZ 2.3 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 TTO, SO4, CL ic50 = 380 uM 415.336, 96.063, 35.453
4FL8 1.2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 TYR ASP GLN ILE IL0 ILE GLU, GOL, GLN ILE IL0 ILE GLU ILE ALA, CL 801.916, 92.094, 743.944, 35.453
4FM6 1.4 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 TYR ASP GLN ILE ILE ILE, NA, GOL, CL 485.582, 22.99, 92.094, 35.453
1SP5 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 TYR ASP GLN ILE LEU, DMS, CL, BME 649.722, 78.133, 35.453, 78.133
2NPH 1.65 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 TYR VAL ASP GLY ALA, ALA GLU THR PHE 522.535, 465.483
1UPJ 2.22 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 U01 373.24
1RTH 2.2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.49 U05 ic50 = 0.4 uM 298.297
1A9M 2.3 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 U0E Ki = 119 nM 596.762
1AXA 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 U0E 596.762
1GNM 2.3 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 U0E Ki = 560 nM 596.762
1GNN 2.3 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 U0E Ki = 2100 nM 596.762
1GNO 2.3 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 U0E Ki = 20 nM 596.762
4CHO 1.7 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 U2Z, EDO, ACT, GOL, SO4 217.267, 62.068, 59.044, 92.094, 96.063
1S1T 2.4 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.49 UC1, PO4 335.848, 94.971
1HPO 2.5 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 UNI Ki = 0.6 nM 504.597
4PHV 2.1 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 VAC ic50 = 0.67 nM 618.761
8HVP 2.5 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 VAL SER GLN ASN LOV ILE VAL Ki < 1 nM 872.075
1MT7 1.9 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 VAL SER GLN ASN TYR PRO ILE VAL GLN ASN, ACT 904.056, 59.044
4CER 1.7 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 VL4, CL, SO4 496.552, 35.453, 96.063
4CJQ 1.7 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 VXO, SO4, ACT Kd = 256 uM 436.5, 96.063, 59.044
4CFA 2.05 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 WOP, SO4 475.493, 96.063
4CIG 1.7 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 X0P, ACT, SO4 Kd = 214 uM 498.57, 59.044, 96.063
1HVR 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 XK2 Ki = 0.31 nM 606.752
1K6T 2.25 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 XN1, ACT Kd = 24 nM 627.816, 59.044
1K6V 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 XN2, ACT Kd = 120 nM 670.837, 59.044
1K6P 2.2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 XN3, ACT Kd = 44 nM 656.811, 59.044
1BV7 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 XV6 Ki = 0.5 nM 758.908
1BV9 2 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 XV6 Ki = 1.1 nM 758.908
1BWA 1.9 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 XV6 Ki = 2.5 nM 758.908
1QBR 1.8 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 XV6 Ki = 0.027 nM 758.908
4CIE 1.7 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 2.7.7.7 Y7N, ACY, CL, SO4 422.474, 60.052, 35.453, 96.063
2ZGA 1.65 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 YDP Ki = 0.48 uM 603.753
3CKT 1.65 HUMAN IMMUNODEFICIENCY VIRUS 1 ENZYME 3.4.23.16 YDP, CL Ki = 0.48 uM 603.753, 35.453
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