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5DGU | 1.22 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 5B7, NA, CL, ACT | Ki = 0.0045 nM | 606.727, 22.99, 35.453, 59.044 |
1C1C | 2.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.49 | 612 | 326.454 | |
5HRP | 1.81 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | 65P, CAC, EDO, SO4 | 534.594, 136.989, 62.068, 96.063 | |
5HRN | 1.75 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.49 | 65P, CAC, SO4, EDO | 534.594, 136.989, 96.063, 62.068 | |
5IVS | 1.46 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 6EF, CL | ic50 = 6.1 nM | 650.763, 35.453 |
5IVR | 1.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 6EG, CL | 566.69, 35.453 | |
5IVQ | 1.57 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 6EH, CL | 425.521, 35.453 | |
5JFP | 1.49 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 6KK, CL, NA | Ki = 0.48 nM | 620.797, 35.453, 22.99 |
5JFU | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 6KQ, CL | Ki = 8.5 nM | 654.813, 35.453 |
5JG1 | 1.16 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 6KR, GOL, NA, CL | Ki = 1.9 nM | 634.824, 92.094, 22.99, 35.453 |
5KRT | 1.65 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | 6W6 | 262.113 | |
4CFC | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | 7NV, CL, ACT, SO4 | 441.477, 35.453, 59.044, 96.063 | |
5TYR | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 7O7 | ic50 = 0.26 nM | 670.839 |
5TYS | 2.01 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 7OA | ic50 = 0.019 nM | 706.82 |
6MKL | 1.7 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME HYDROLASES | 7OA | 706.82 | |
5KGW | 2.34 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | 7SK, SO4 | 393.475, 96.063 | |
5U6E | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | NON-ENZYME OTHER | 82M, EPE, NAG | 408.878, 238.305, 221.208 | |
1QBU | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 846 | Ki = 0.058 nM | 596.739 |
5UOV | 1.33 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 8FP, NA, GOL, CL, ACT | Ki = 0.025 nM | 704.898, 22.99, 92.094, 35.453, 59.044 |
5YOJ | 1.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 8Z0, GOL | 756.907, 92.094 | |
5YOK | 0.85 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | 8Z0, GOL | 756.907, 92.094 | |
4CED | 1.75 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | 9NS, CL, SO4, GOL | 534.557, 35.453, 96.063, 92.094 | |
4CJL | 1.77 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | 9PA, ACT, SO4, CL | 378.463, 59.044, 96.063, 35.453 | |
5OIA | 2.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | 9VK, SO4, MG | ic50 = 0.17 uM | 413.573, 96.063, 24.305 |
5OI8 | 2.35 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.7 | 9VN, SO4, MG | ic50 = 0.21 uM | 413.573, 96.063, 24.305 |
2BQV | 2.1 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | A1A | Ki = 9 nM | 588.694 |
6DH5 | 2.01 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | A60, SO4 | 575.717, 96.063 | |
6DH8 | 1.95 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | A60, SO4 | Ki = 146.2 pM | 575.717, 96.063 |
1HVL | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | A76 | Ki = 1000 pM | 794.981 |
1HVI | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | A77 | Ki = 84 pM | 794.981 |
1HVS | 2.25 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | A77 | Ki = 50 pM | 794.981 |
1HVJ | 2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | A78 | Ki = 4 pM | 780.998 |
1HVC | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | A79 | 794.981 | |
1HVK | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | A79 | Ki = 77 pM | 794.981 |
1ZPA | 2.02 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | A83 | Ki = 4 nM | 720.878 |
1PRO | 1.8 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | A88 | Ki = 5 pM | 583.674 |
1VRU | 2.4 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 2.7.7.49 | AAP | ic50 = 0.1 uM | 351.227 |
2A4F | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | AAU | 641.71 | |
4L1A | 1.9 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME HYDROLASES | AB1 | ic50 = 5.39 nM | 628.801 |
6DJ1 | 1.26 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | AB1, CL, NA | Ki = 0.031 nM | 628.801, 35.453, 22.99 |
6DJ2 | 1.36 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | AB1, CL, NA | Ki = 4.5 nM | 628.801, 35.453, 22.99 |
6PJB | 1.98 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | AB1, SO4 | 628.801, 96.063 | |
1ZP8 | 2.02 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | AB2 | Ki = 1.7 nM | 663.784 |
7HVP | 2.4 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | ACE SER LEU ASN JG3 ILE VME | Ki = 0.24 nM | 818.006 |
1YTH | 2.2 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | ACE SER LEU ASN PHE | 520.563 | |
3LZS | 1.95 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | ACT, 017 | Kd = 0.0109 nM | 59.044, 547.664 |
3LZU | 1.76 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | ACT, 017 | Kd = 0.087 nM | 59.044, 547.664 |
4DQE | 1.3 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | ACT, 017 | 59.044, 547.664 | |
4Q1W | 1.85 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | ACT, 017, PO4 | Ki = 2 pM | 59.044, 547.664, 94.971 |
4Q1Y | 1.5 | HUMAN IMMUNODEFICIENCY VIRUS 1 | ENZYME 3.4.23.16 | ACT, 017, PO4 | Ki = 45 pM | 59.044, 547.664, 94.971 |
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